DK1667975T3 - En polymorf form for 3-phenylsulfonyl-8-piperazin-1-yl-quinolin - Google Patents

En polymorf form for 3-phenylsulfonyl-8-piperazin-1-yl-quinolin

Info

Publication number
DK1667975T3
DK1667975T3 DK04765655T DK04765655T DK1667975T3 DK 1667975 T3 DK1667975 T3 DK 1667975T3 DK 04765655 T DK04765655 T DK 04765655T DK 04765655 T DK04765655 T DK 04765655T DK 1667975 T3 DK1667975 T3 DK 1667975T3
Authority
DK
Denmark
Prior art keywords
phenylsulfonyl
piperazin
quinoline
polymorphic form
polymorphic
Prior art date
Application number
DK04765655T
Other languages
Danish (da)
English (en)
Inventor
Asa Elisabeth Gladwin
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of DK1667975T3 publication Critical patent/DK1667975T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • C07D215/40Nitrogen atoms attached in position 8
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Quinoline Compounds (AREA)
DK04765655T 2003-09-26 2004-09-23 En polymorf form for 3-phenylsulfonyl-8-piperazin-1-yl-quinolin DK1667975T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0322629.7A GB0322629D0 (en) 2003-09-26 2003-09-26 Novel compound
PCT/EP2004/010843 WO2005040124A1 (en) 2003-09-26 2004-09-23 A polymorphic form of 3-phenylsulfonyl -8-piperazin-1-yl-quinoline

Publications (1)

Publication Number Publication Date
DK1667975T3 true DK1667975T3 (da) 2008-04-14

Family

ID=29286934

Family Applications (1)

Application Number Title Priority Date Filing Date
DK04765655T DK1667975T3 (da) 2003-09-26 2004-09-23 En polymorf form for 3-phenylsulfonyl-8-piperazin-1-yl-quinolin

Country Status (24)

Country Link
US (1) US20070032504A1 (ja)
EP (1) EP1667975B1 (ja)
JP (1) JP2007506702A (ja)
CN (1) CN1856471A (ja)
AU (1) AU2004283805A1 (ja)
BR (1) BRPI0414678A (ja)
CA (1) CA2540022A1 (ja)
CO (1) CO5680402A2 (ja)
DE (1) DE602004010410T2 (ja)
DK (1) DK1667975T3 (ja)
ES (1) ES2297465T3 (ja)
GB (1) GB0322629D0 (ja)
HK (1) HK1094190A1 (ja)
HR (1) HRP20080055T3 (ja)
IL (1) IL174213A0 (ja)
IS (1) IS8399A (ja)
MA (1) MA28093A1 (ja)
MX (1) MXPA06003375A (ja)
NO (1) NO20061791L (ja)
PL (1) PL1667975T3 (ja)
PT (1) PT1667975E (ja)
RU (1) RU2355681C2 (ja)
WO (1) WO2005040124A1 (ja)
ZA (1) ZA200601453B (ja)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003080580A2 (en) * 2002-03-27 2003-10-02 Glaxo Group Limited Quinoline derivatives and their use as 5-ht6 ligands
CN1826322B (zh) 2003-07-22 2012-04-18 艾尼纳制药公司 用于预防和治疗相关病症而作为5-ht2a血清素受体调节剂的二芳基和芳基杂芳基脲衍生物
NZ542865A (en) 2003-09-18 2009-04-30 Virobay Inc Haloalkyl containing compounds as cysteine protease inhibitors
BRPI0611516A2 (pt) 2005-06-02 2010-09-14 Hoffmann La Roche 3-metanossulfonilquinolinas como realçadores ("enhancers") de gaba-b
GB0519758D0 (en) * 2005-09-28 2005-11-09 Glaxo Group Ltd Novel process
EP2120950B1 (en) * 2007-03-21 2012-07-04 Glaxo Group Limited Use of quinoline derivatives in the treatment of pain
EP2508177A1 (en) 2007-12-12 2012-10-10 Glaxo Group Limited Combinations comprising 3-phenylsulfonyl-8-piperazinyl-1yl-quinoline
US20110021538A1 (en) 2008-04-02 2011-01-27 Arena Pharmaceuticals, Inc. Processes for the preparation of pyrazole derivatives useful as modulators of the 5-ht2a serotonin receptor
WO2010062321A1 (en) 2008-10-28 2010-06-03 Arena Pharmaceuticals, Inc. Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2h-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)-urea and crystalline forms related thereto
AU2016276966A1 (en) 2015-06-12 2018-01-18 Axovant Sciences Gmbh Diaryl and arylheteroaryl urea derivatives useful for the prophylaxis and treatment of REM sleep behavior disorder
TW201720439A (zh) 2015-07-15 2017-06-16 Axovant Sciences Gmbh 用於預防及治療與神經退化性疾病相關的幻覺之作為5-ht2a血清素受體的二芳基及芳基雜芳基脲衍生物
WO2017202206A1 (zh) * 2016-05-27 2017-11-30 深圳市塔吉瑞生物医药有限公司 一种取代的喹啉化合物及其药物组合物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9818916D0 (en) * 1998-08-28 1998-10-21 Smithkline Beecham Plc Use
WO2003080580A2 (en) * 2002-03-27 2003-10-02 Glaxo Group Limited Quinoline derivatives and their use as 5-ht6 ligands
GB0321473D0 (en) * 2003-09-12 2003-10-15 Glaxo Group Ltd Novel compounds

Also Published As

Publication number Publication date
MA28093A1 (fr) 2006-08-01
PL1667975T3 (pl) 2008-04-30
IL174213A0 (en) 2006-08-01
DE602004010410T2 (de) 2008-10-16
RU2355681C2 (ru) 2009-05-20
ZA200601453B (en) 2007-04-25
AU2004283805A1 (en) 2005-05-06
NO20061791L (no) 2006-04-24
EP1667975A1 (en) 2006-06-14
WO2005040124A1 (en) 2005-05-06
BRPI0414678A (pt) 2006-11-28
ES2297465T3 (es) 2008-05-01
RU2006114024A (ru) 2007-11-10
IS8399A (is) 2006-04-05
US20070032504A1 (en) 2007-02-08
HRP20080055T3 (en) 2008-02-29
CO5680402A2 (es) 2006-09-29
JP2007506702A (ja) 2007-03-22
HK1094190A1 (en) 2007-03-23
DE602004010410D1 (en) 2008-01-10
EP1667975B1 (en) 2007-11-28
GB0322629D0 (en) 2003-10-29
PT1667975E (pt) 2008-02-29
CA2540022A1 (en) 2005-05-06
MXPA06003375A (es) 2006-06-08
CN1856471A (zh) 2006-11-01

Similar Documents

Publication Publication Date Title
SE0302305D0 (sv) Novel Compounds
IS8108A (is) Ný efnasambönd
DK1605897T3 (da) Polyethelen-glycol-link-glp-1-forbindelser
HK1093483A1 (en) Polymorphic form of n-
IS8228A (is) Ný asetídínefnasambönd
IS8283A (is) Umbrotsefni kvetíapíns
IS8089A (is) Efnasambönd
IL174213A0 (en) A polymorphic form of 3-phenylsulfonyl-8-piperazin-1-yl-quinoline
IS8292A (is) Ný efnasambönd
ITMI20042238A1 (it) Composti per fluoropolirterei
NO20055097D0 (no) Krystallinske N-formyl-hydroksylaminforbindelser
NO20031736D0 (no) Forbindelser
SE0303452D0 (sv) New compounds
NO20054532D0 (no) Fremgangsmater for a forhindre glukonoylering av proteiner
ITMI20032550A1 (it) Mescole elastomeriche a base di nerofumo
SE0402103D0 (sv) Novel compounds
SI1667975T1 (sl) Polimorfna oblika 3-fenilsulfonil-8-piperazin-1-il-kinolina
SE0302667D0 (sv) Novel Compounds
SE0300388D0 (sv) Novel compounds
SE0300118D0 (sv) Novel Compounds
SE0302369D0 (sv) New compounds
SE0301120D0 (sv) New compounds
SE0302368D0 (sv) New compounds
SE0301246D0 (sv) New compounds
SE0303078D0 (sv) New compounds