HRP20080055T3 - A polymorphic form of 3-phenylsulfonyl-8-piperazin-1-yl-quinoline - Google Patents

A polymorphic form of 3-phenylsulfonyl-8-piperazin-1-yl-quinoline

Info

Publication number
HRP20080055T3
HRP20080055T3 HR20080055T HRP20080055T HRP20080055T3 HR P20080055 T3 HRP20080055 T3 HR P20080055T3 HR 20080055 T HR20080055 T HR 20080055T HR P20080055 T HRP20080055 T HR P20080055T HR P20080055 T3 HRP20080055 T3 HR P20080055T3
Authority
HR
Croatia
Prior art keywords
phenylsulfonyl
piperazin
polymorphic form
quinoline
ylquinoline
Prior art date
Application number
HR20080055T
Other languages
English (en)
Croatian (hr)
Inventor
Elisabeth Gladwin Asa
Original Assignee
Glaxo Group Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Publication of HRP20080055T3 publication Critical patent/HRP20080055T3/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • C07D215/40Nitrogen atoms attached in position 8
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Quinoline Compounds (AREA)
HR20080055T 2003-09-26 2008-02-04 A polymorphic form of 3-phenylsulfonyl-8-piperazin-1-yl-quinoline HRP20080055T3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0322629.7A GB0322629D0 (en) 2003-09-26 2003-09-26 Novel compound
PCT/EP2004/010843 WO2005040124A1 (en) 2003-09-26 2004-09-23 A polymorphic form of 3-phenylsulfonyl -8-piperazin-1-yl-quinoline

Publications (1)

Publication Number Publication Date
HRP20080055T3 true HRP20080055T3 (en) 2008-02-29

Family

ID=29286934

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20080055T HRP20080055T3 (en) 2003-09-26 2008-02-04 A polymorphic form of 3-phenylsulfonyl-8-piperazin-1-yl-quinoline

Country Status (24)

Country Link
US (1) US20070032504A1 (ja)
EP (1) EP1667975B1 (ja)
JP (1) JP2007506702A (ja)
CN (1) CN1856471A (ja)
AU (1) AU2004283805A1 (ja)
BR (1) BRPI0414678A (ja)
CA (1) CA2540022A1 (ja)
CO (1) CO5680402A2 (ja)
DE (1) DE602004010410T2 (ja)
DK (1) DK1667975T3 (ja)
ES (1) ES2297465T3 (ja)
GB (1) GB0322629D0 (ja)
HK (1) HK1094190A1 (ja)
HR (1) HRP20080055T3 (ja)
IL (1) IL174213A0 (ja)
IS (1) IS8399A (ja)
MA (1) MA28093A1 (ja)
MX (1) MXPA06003375A (ja)
NO (1) NO20061791L (ja)
PL (1) PL1667975T3 (ja)
PT (1) PT1667975E (ja)
RU (1) RU2355681C2 (ja)
WO (1) WO2005040124A1 (ja)
ZA (1) ZA200601453B (ja)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1497266E (pt) * 2002-03-27 2008-09-10 Glaxo Group Ltd Derivados de quinolina e sua utilização como ligandos 5-ht6
MXPA06000795A (es) 2003-07-22 2006-08-23 Arena Pharm Inc Derivados de diaril y arilheteroaril urea como moduladores del receptor 5-ht2a de serotonina utiles para la profilaxis y tratamiento de desordenes relacionados con el mismo.
SG146658A1 (en) 2003-09-18 2008-10-30 Schering Ag Haloalkyl containing compounds as cysteine protease inhibitors
CN101189208A (zh) 2005-06-02 2008-05-28 弗·哈夫曼-拉罗切有限公司 作为gaba-b增强剂的3-甲磺酰基喹啉
GB0519758D0 (en) * 2005-09-28 2005-11-09 Glaxo Group Ltd Novel process
ES2389958T3 (es) * 2007-03-21 2012-11-05 Glaxo Group Limited Uso de derivados de quinolina en el tratamiento del dolor
EP2508177A1 (en) 2007-12-12 2012-10-10 Glaxo Group Limited Combinations comprising 3-phenylsulfonyl-8-piperazinyl-1yl-quinoline
WO2009123714A2 (en) 2008-04-02 2009-10-08 Arena Pharmaceuticals, Inc. Processes for the preparation of pyrazole derivatives useful as modulators of the 5-ht2a serotonin receptor
WO2010062321A1 (en) 2008-10-28 2010-06-03 Arena Pharmaceuticals, Inc. Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2h-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)-urea and crystalline forms related thereto
EP4119141A1 (en) 2015-06-12 2023-01-18 Axovant Sciences GmbH Nelotanserin for the prophylaxis and treatment of rem sleep behavior disorder
CA2992518A1 (en) 2015-07-15 2017-01-19 Axovant Sciences Gmbh Diaryl and arylheteroaryl urea derivatives as modulators of the 5-ht2a serotonin receptor useful for the prophylaxis and treatment of hallucinations associated with a neurodegenerative disease
CN108290842B (zh) * 2016-05-27 2021-04-06 深圳市塔吉瑞生物医药有限公司 一种取代的喹啉化合物及其药物组合物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9818916D0 (en) * 1998-08-28 1998-10-21 Smithkline Beecham Plc Use
PT1497266E (pt) * 2002-03-27 2008-09-10 Glaxo Group Ltd Derivados de quinolina e sua utilização como ligandos 5-ht6
GB0321473D0 (en) * 2003-09-12 2003-10-15 Glaxo Group Ltd Novel compounds

Also Published As

Publication number Publication date
CN1856471A (zh) 2006-11-01
CO5680402A2 (es) 2006-09-29
ES2297465T3 (es) 2008-05-01
WO2005040124A1 (en) 2005-05-06
MXPA06003375A (es) 2006-06-08
PL1667975T3 (pl) 2008-04-30
EP1667975B1 (en) 2007-11-28
GB0322629D0 (en) 2003-10-29
NO20061791L (no) 2006-04-24
AU2004283805A1 (en) 2005-05-06
MA28093A1 (fr) 2006-08-01
DE602004010410T2 (de) 2008-10-16
RU2006114024A (ru) 2007-11-10
BRPI0414678A (pt) 2006-11-28
IS8399A (is) 2006-04-05
HK1094190A1 (en) 2007-03-23
DK1667975T3 (da) 2008-04-14
EP1667975A1 (en) 2006-06-14
ZA200601453B (en) 2007-04-25
CA2540022A1 (en) 2005-05-06
PT1667975E (pt) 2008-02-29
US20070032504A1 (en) 2007-02-08
DE602004010410D1 (en) 2008-01-10
RU2355681C2 (ru) 2009-05-20
IL174213A0 (en) 2006-08-01
JP2007506702A (ja) 2007-03-22

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