DK1663243T3 - Farmaceutisk formulering omfattende et pyrimidin-a-on-derivat coatet med en enterisk polymer - Google Patents

Farmaceutisk formulering omfattende et pyrimidin-a-on-derivat coatet med en enterisk polymer

Info

Publication number
DK1663243T3
DK1663243T3 DK04764689T DK04764689T DK1663243T3 DK 1663243 T3 DK1663243 T3 DK 1663243T3 DK 04764689 T DK04764689 T DK 04764689T DK 04764689 T DK04764689 T DK 04764689T DK 1663243 T3 DK1663243 T3 DK 1663243T3
Authority
DK
Denmark
Prior art keywords
pyrimidine
pharmaceutical formulation
enteric polymer
derivative coated
derivative
Prior art date
Application number
DK04764689T
Other languages
Danish (da)
English (en)
Inventor
Schie Dirk Marinus J Van
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of DK1663243T3 publication Critical patent/DK1663243T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846—Poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK04764689T 2003-09-02 2004-08-31 Farmaceutisk formulering omfattende et pyrimidin-a-on-derivat coatet med en enterisk polymer DK1663243T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0320522.6A GB0320522D0 (en) 2003-09-02 2003-09-02 Formulation
PCT/EP2004/009726 WO2005021002A1 (fr) 2003-09-02 2004-08-31 Preparation pharmaceutique comprenant un derive de la pyrimidine-a-one enrobe d'un polymere enterique

Publications (1)

Publication Number Publication Date
DK1663243T3 true DK1663243T3 (da) 2009-05-04

Family

ID=28686767

Family Applications (1)

Application Number Title Priority Date Filing Date
DK04764689T DK1663243T3 (da) 2003-09-02 2004-08-31 Farmaceutisk formulering omfattende et pyrimidin-a-on-derivat coatet med en enterisk polymer

Country Status (30)

Country Link
US (2) US20060287346A1 (fr)
EP (1) EP1663243B1 (fr)
JP (1) JP4892346B2 (fr)
KR (1) KR101115984B1 (fr)
CN (2) CN1874778B (fr)
AR (1) AR045547A1 (fr)
AT (1) ATE422889T1 (fr)
AU (1) AU2004268376B2 (fr)
BR (1) BRPI0414038A (fr)
CA (1) CA2537178C (fr)
CY (1) CY1108953T1 (fr)
DE (1) DE602004019547D1 (fr)
DK (1) DK1663243T3 (fr)
ES (1) ES2319124T3 (fr)
GB (1) GB0320522D0 (fr)
HR (1) HRP20090147T3 (fr)
IL (1) IL173910A (fr)
IS (1) IS2677B (fr)
MA (1) MA28033A1 (fr)
MX (1) MXPA06002436A (fr)
MY (1) MY139165A (fr)
NO (1) NO333744B1 (fr)
NZ (1) NZ545453A (fr)
PL (1) PL1663243T3 (fr)
PT (1) PT1663243E (fr)
RU (1) RU2359660C2 (fr)
SI (1) SI1663243T1 (fr)
TW (1) TWI343257B (fr)
WO (1) WO2005021002A1 (fr)
ZA (1) ZA200601599B (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0320522D0 (en) * 2003-09-02 2003-10-01 Glaxo Group Ltd Formulation
BRPI0810336A2 (pt) 2007-05-11 2019-03-19 The Trustees Of The University Of Pennsylvania "método para tratar e/ou prevenir úlceras de pele em um indivíduo"
MX2009012188A (es) 2007-05-11 2010-02-24 Univ Jefferson Métodos de tratamiento y prevención de enfermedades y desórdenes neurodegenerativos.
MA33295B1 (fr) 2009-04-24 2012-05-02 Iceutica Pty Ltd Nouvelle formulation de diclofénac
EP2651403B1 (fr) 2010-12-17 2020-12-02 Glaxo Group Limited Procédés de traitement et de prévention de maladies oculaires
WO2013082275A1 (fr) 2011-11-30 2013-06-06 Trustees Of Boston College Inhibiteurs de phosphodiestérases 11 (pde11) et procédés d'utilisation pour augmenter la production de cortisol
US9526734B2 (en) 2014-06-09 2016-12-27 Iceutica Pty Ltd. Formulation of meloxicam
JP6625604B2 (ja) 2014-07-22 2019-12-25 グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ Ｄｅｖｅｌｏｐｍｅｎｔ Ｌｉｍｉｔｅｄ 化合物

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3619570C1 (en) 1986-06-11 1987-10-29 Kneipp Werke Kneipp Mittel Zen Coated garlic tablet
US4971805A (en) * 1987-12-23 1990-11-20 Teysan Pharmaceuticals Co., Ltd. Slow-releasing granules and long acting mixed granules comprising the same
IT1227899B (it) * 1988-12-23 1991-05-14 Poli Ind Chimica Spa Rivestimento totale o parziale di principi attivi farmaceutici e relative composizioni
TW209174B (fr) * 1991-04-19 1993-07-11 Takeda Pharm Industry Co Ltd
JPH07223970A (ja) * 1994-02-10 1995-08-22 Tanabe Seiyaku Co Ltd 消化管内適所放出製剤
JP2917799B2 (ja) * 1994-03-11 1999-07-12 田辺製薬株式会社 消化管内適所放出型製剤
SG80553A1 (en) 1995-07-20 2001-05-22 Tanabe Seiyaku Co Pharmaceutical preparation in form of coated capsule releasable at lower part of digestive tract
JP3185206B2 (ja) * 1995-07-20 2001-07-09 田辺製薬株式会社 消化管下部放出型被覆カプセル製剤
NZ333182A (en) * 1996-06-06 2000-03-27 Bifodan As Enteric coating comprising alginic acid and a water soluble binding agent for an oral preparation
AU3691297A (en) * 1996-08-15 1998-03-06 Losan Pharma Gmbh Easy to swallow oral medicament composition
US6296876B1 (en) * 1997-10-06 2001-10-02 Isa Odidi Pharmaceutical formulations for acid labile substances
EP1736144B1 (fr) * 1998-05-18 2015-11-11 Takeda Pharmaceutical Company Limited Comprimé à désintégration orale
PT1131070E (pt) * 1998-11-12 2008-11-19 Smithkline Beecham Plc Composição farmacêutica para libertação modificada de um sensibilizador à insulina e de outro agente antidiabético
US6268385B1 (en) * 1999-08-26 2001-07-31 Robert R. Whittle Dry blend pharmaceutical formulations
ES2330552T3 (es) * 2000-02-16 2009-12-11 Smithkline Beecham Plc Derivados de pirimidin-5-ona como inhibidores de ldl-pla2.
AUPQ672800A0 (en) * 2000-04-06 2000-05-04 Natraherbal Pty Ltd Garlic supplement for deodoriser
CZ303572B6 (cs) * 2000-06-28 2012-12-12 Smithkline Beecham P. L. C. Jemne rozmelnený prostredek a zpusob jeho prípravy
JP5138856B2 (ja) * 2001-06-20 2013-02-06 武田薬品工業株式会社 錠剤の製造方法
WO2003000169A1 (fr) 2001-06-20 2003-01-03 Takeda Chemical Industries, Ltd. Procede de fabrication de comprimes
RU2203671C1 (ru) * 2002-03-25 2003-05-10 Общество С Ограниченной Ответственностью "Научно-Технологическая Фармацевтическая Фирма "Полисан" Противовирусный лекарственный препарат для перорального применения
GB0320522D0 (en) * 2003-09-02 2003-10-01 Glaxo Group Ltd Formulation

Also Published As

Publication number Publication date
CN1874778B (zh) 2011-06-22
AU2004268376B2 (en) 2010-04-22
WO2005021002A1 (fr) 2005-03-10
KR101115984B1 (ko) 2012-03-13
US20060287346A1 (en) 2006-12-21
NO333744B1 (no) 2013-09-09
IL173910A (en) 2010-11-30
IL173910A0 (en) 2006-07-05
IS8366A (is) 2006-03-20
AR045547A1 (es) 2005-11-02
ATE422889T1 (de) 2009-03-15
KR20060118422A (ko) 2006-11-23
US20090306113A1 (en) 2009-12-10
TWI343257B (en) 2011-06-11
GB0320522D0 (en) 2003-10-01
EP1663243B1 (fr) 2009-02-18
RU2006110546A (ru) 2006-08-10
BRPI0414038A (pt) 2006-10-24
ES2319124T3 (es) 2009-05-04
AU2004268376A1 (en) 2005-03-10
JP4892346B2 (ja) 2012-03-07
DE602004019547D1 (de) 2009-04-02
CN102204891A (zh) 2011-10-05
RU2359660C2 (ru) 2009-06-27
ZA200601599B (en) 2007-05-30
PT1663243E (pt) 2009-04-27
CN102204891B (zh) 2013-08-21
MXPA06002436A (es) 2006-06-20
HK1091734A1 (en) 2007-01-26
US8772303B2 (en) 2014-07-08
CY1108953T1 (el) 2014-07-02
EP1663243A1 (fr) 2006-06-07
HRP20090147T3 (hr) 2009-04-30
CA2537178C (fr) 2013-03-19
SI1663243T1 (sl) 2009-06-30
MA28033A1 (fr) 2006-07-03
CA2537178A1 (fr) 2005-03-10
MY139165A (en) 2009-08-28
JP2007504195A (ja) 2007-03-01
NZ545453A (en) 2009-12-24
PL1663243T3 (pl) 2009-07-31
NO20061514L (no) 2006-04-03
CN1874778A (zh) 2006-12-06
IS2677B (is) 2010-09-15
TW200517113A (en) 2005-06-01

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