DK1663243T3 - Farmaceutisk formulering omfattende et pyrimidin-a-on-derivat coatet med en enterisk polymer - Google Patents

Farmaceutisk formulering omfattende et pyrimidin-a-on-derivat coatet med en enterisk polymer

Info

Publication number
DK1663243T3
DK1663243T3 DK04764689T DK04764689T DK1663243T3 DK 1663243 T3 DK1663243 T3 DK 1663243T3 DK 04764689 T DK04764689 T DK 04764689T DK 04764689 T DK04764689 T DK 04764689T DK 1663243 T3 DK1663243 T3 DK 1663243T3
Authority
DK
Denmark
Prior art keywords
pyrimidine
pharmaceutical formulation
enteric polymer
derivative coated
derivative
Prior art date
Application number
DK04764689T
Other languages
Danish (da)
English (en)
Inventor
Schie Dirk Marinus J Van
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of DK1663243T3 publication Critical patent/DK1663243T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2886Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK04764689T 2003-09-02 2004-08-31 Farmaceutisk formulering omfattende et pyrimidin-a-on-derivat coatet med en enterisk polymer DK1663243T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0320522.6A GB0320522D0 (en) 2003-09-02 2003-09-02 Formulation
PCT/EP2004/009726 WO2005021002A1 (fr) 2003-09-02 2004-08-31 Preparation pharmaceutique comprenant un derive de la pyrimidine-a-one enrobe d'un polymere enterique

Publications (1)

Publication Number Publication Date
DK1663243T3 true DK1663243T3 (da) 2009-05-04

Family

ID=28686767

Family Applications (1)

Application Number Title Priority Date Filing Date
DK04764689T DK1663243T3 (da) 2003-09-02 2004-08-31 Farmaceutisk formulering omfattende et pyrimidin-a-on-derivat coatet med en enterisk polymer

Country Status (30)

Country Link
US (2) US20060287346A1 (fr)
EP (1) EP1663243B1 (fr)
JP (1) JP4892346B2 (fr)
KR (1) KR101115984B1 (fr)
CN (2) CN1874778B (fr)
AR (1) AR045547A1 (fr)
AT (1) ATE422889T1 (fr)
AU (1) AU2004268376B2 (fr)
BR (1) BRPI0414038A (fr)
CA (1) CA2537178C (fr)
CY (1) CY1108953T1 (fr)
DE (1) DE602004019547D1 (fr)
DK (1) DK1663243T3 (fr)
ES (1) ES2319124T3 (fr)
GB (1) GB0320522D0 (fr)
HR (1) HRP20090147T3 (fr)
IL (1) IL173910A (fr)
IS (1) IS2677B (fr)
MA (1) MA28033A1 (fr)
MX (1) MXPA06002436A (fr)
MY (1) MY139165A (fr)
NO (1) NO333744B1 (fr)
NZ (1) NZ545453A (fr)
PL (1) PL1663243T3 (fr)
PT (1) PT1663243E (fr)
RU (1) RU2359660C2 (fr)
SI (1) SI1663243T1 (fr)
TW (1) TWI343257B (fr)
WO (1) WO2005021002A1 (fr)
ZA (1) ZA200601599B (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0320522D0 (en) * 2003-09-02 2003-10-01 Glaxo Group Ltd Formulation
EP2155225B1 (fr) 2007-05-11 2015-07-08 The Trustees of the University of Pennsylvania Procédés de traitement des ulcères de la peau
WO2008140449A1 (fr) 2007-05-11 2008-11-20 Thomas Jefferson University Méthodes de traitement et de prévention de maladies et de troubles neurodégénératifs
MA33295B1 (fr) 2009-04-24 2012-05-02 Iceutica Pty Ltd Nouvelle formulation de diclofénac
WO2012080497A2 (fr) 2010-12-17 2012-06-21 Glaxo Group Limited Procédés de traitement et de prévention de maladies oculaires
US9173884B2 (en) 2011-11-30 2015-11-03 Trustees Of Boston College Inhibitors of phosphodiesterase 11 (PDE11)
US9526734B2 (en) 2014-06-09 2016-12-27 Iceutica Pty Ltd. Formulation of meloxicam
ES2744339T3 (es) 2014-07-22 2020-02-24 Glaxosmithkline Ip Dev Ltd Compuestos

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3619570C1 (en) 1986-06-11 1987-10-29 Kneipp Werke Kneipp Mittel Zen Coated garlic tablet
US4971805A (en) * 1987-12-23 1990-11-20 Teysan Pharmaceuticals Co., Ltd. Slow-releasing granules and long acting mixed granules comprising the same
IT1227899B (it) * 1988-12-23 1991-05-14 Poli Ind Chimica Spa Rivestimento totale o parziale di principi attivi farmaceutici e relative composizioni
TW209174B (fr) * 1991-04-19 1993-07-11 Takeda Pharm Industry Co Ltd
JPH07223970A (ja) * 1994-02-10 1995-08-22 Tanabe Seiyaku Co Ltd 消化管内適所放出製剤
JP2917799B2 (ja) * 1994-03-11 1999-07-12 田辺製薬株式会社 消化管内適所放出型製剤
SG80553A1 (en) 1995-07-20 2001-05-22 Tanabe Seiyaku Co Pharmaceutical preparation in form of coated capsule releasable at lower part of digestive tract
JP3185206B2 (ja) * 1995-07-20 2001-07-09 田辺製薬株式会社 消化管下部放出型被覆カプセル製剤
WO1997046224A1 (fr) * 1996-06-06 1997-12-11 Bifodan A/S Revetement gastro-resistant comprenant de l'acide alginique pour preparation a administrer par voie orale
DE59702733D1 (de) * 1996-08-15 2001-01-11 Losan Pharma Gmbh Gut schluckbare orale arzneiform
US6296876B1 (en) * 1997-10-06 2001-10-02 Isa Odidi Pharmaceutical formulations for acid labile substances
JP3746167B2 (ja) * 1998-05-18 2006-02-15 武田薬品工業株式会社 医薬製剤
DE69939485D1 (de) * 1998-11-12 2008-10-16 Smithkline Beecham Plc Arzneimittel zur gesteuerten freisetzung eines insulin sensibilisators und metformin
US6268385B1 (en) * 1999-08-26 2001-07-31 Robert R. Whittle Dry blend pharmaceutical formulations
ATE437862T1 (de) * 2000-02-16 2009-08-15 Smithkline Beecham Plc Pyrimidin-5-onderivate als ldl-pla2 inhibitoren
AUPQ672800A0 (en) * 2000-04-06 2000-05-04 Natraherbal Pty Ltd Garlic supplement for deodoriser
NZ522783A (en) * 2000-06-28 2004-07-30 Smithkline Beecham P Wet milling process for pharmaceuticals with agitator or chamber having nylon with internal lubricant
JP5138856B2 (ja) * 2001-06-20 2013-02-06 武田薬品工業株式会社 錠剤の製造方法
EP1405621B1 (fr) 2001-06-20 2011-05-11 Takeda Pharmaceutical Company Limited Procede de fabrication de comprimes
RU2203671C1 (ru) * 2002-03-25 2003-05-10 Общество С Ограниченной Ответственностью "Научно-Технологическая Фармацевтическая Фирма "Полисан" Противовирусный лекарственный препарат для перорального применения
GB0320522D0 (en) * 2003-09-02 2003-10-01 Glaxo Group Ltd Formulation

Also Published As

Publication number Publication date
MY139165A (en) 2009-08-28
NO20061514L (no) 2006-04-03
US20060287346A1 (en) 2006-12-21
NZ545453A (en) 2009-12-24
CY1108953T1 (el) 2014-07-02
ZA200601599B (en) 2007-05-30
CN102204891B (zh) 2013-08-21
IS2677B (is) 2010-09-15
AU2004268376B2 (en) 2010-04-22
KR101115984B1 (ko) 2012-03-13
KR20060118422A (ko) 2006-11-23
US20090306113A1 (en) 2009-12-10
DE602004019547D1 (de) 2009-04-02
EP1663243B1 (fr) 2009-02-18
CA2537178A1 (fr) 2005-03-10
CA2537178C (fr) 2013-03-19
RU2006110546A (ru) 2006-08-10
PT1663243E (pt) 2009-04-27
BRPI0414038A (pt) 2006-10-24
JP4892346B2 (ja) 2012-03-07
TW200517113A (en) 2005-06-01
IL173910A0 (en) 2006-07-05
HRP20090147T3 (hr) 2009-04-30
IS8366A (is) 2006-03-20
HK1091734A1 (en) 2007-01-26
CN1874778A (zh) 2006-12-06
RU2359660C2 (ru) 2009-06-27
CN102204891A (zh) 2011-10-05
JP2007504195A (ja) 2007-03-01
CN1874778B (zh) 2011-06-22
ES2319124T3 (es) 2009-05-04
PL1663243T3 (pl) 2009-07-31
AU2004268376A1 (en) 2005-03-10
MA28033A1 (fr) 2006-07-03
ATE422889T1 (de) 2009-03-15
IL173910A (en) 2010-11-30
TWI343257B (en) 2011-06-11
NO333744B1 (no) 2013-09-09
EP1663243A1 (fr) 2006-06-07
GB0320522D0 (en) 2003-10-01
US8772303B2 (en) 2014-07-08
WO2005021002A1 (fr) 2005-03-10
AR045547A1 (es) 2005-11-02
SI1663243T1 (sl) 2009-06-30
MXPA06002436A (es) 2006-06-20

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