DK165744C - Thienopyrimidinderivater, fremgangsmaader til fremstilling deraf og farmaceutiske praeparater - Google Patents

Thienopyrimidinderivater, fremgangsmaader til fremstilling deraf og farmaceutiske praeparater

Info

Publication number
DK165744C
DK165744C DK617184A DK617184A DK165744C DK 165744 C DK165744 C DK 165744C DK 617184 A DK617184 A DK 617184A DK 617184 A DK617184 A DK 617184A DK 165744 C DK165744 C DK 165744C
Authority
DK
Denmark
Prior art keywords
sup
carbon atoms
alkyl group
procedures
preparing
Prior art date
Application number
DK617184A
Other languages
Danish (da)
English (en)
Other versions
DK165744B (da
DK617184D0 (da
DK617184A (da
Inventor
Kunihiro Ninomiya
Issei Nitta
Akihiro Tobe
Mitsuo Egawa
Ryoji Kikumoto
Original Assignee
Mitsubishi Chem Ind
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsubishi Chem Ind filed Critical Mitsubishi Chem Ind
Publication of DK617184D0 publication Critical patent/DK617184D0/da
Publication of DK617184A publication Critical patent/DK617184A/da
Publication of DK165744B publication Critical patent/DK165744B/da
Application granted granted Critical
Publication of DK165744C publication Critical patent/DK165744C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK617184A 1984-01-05 1984-12-20 Thienopyrimidinderivater, fremgangsmaader til fremstilling deraf og farmaceutiske praeparater DK165744C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP47984 1984-01-05
JP59000479A JPS60146891A (ja) 1984-01-05 1984-01-05 〔２，３−ｄ〕チエノピリミジン誘導体およびその塩

Publications (4)

Publication Number Publication Date
DK617184D0 DK617184D0 (da) 1984-12-20
DK617184A DK617184A (da) 1985-07-06
DK165744B DK165744B (da) 1993-01-11
DK165744C true DK165744C (da) 1993-06-07

Family

ID=11474905

Family Applications (1)

Application Number Title Priority Date Filing Date
DK617184A DK165744C (da) 1984-01-05 1984-12-20 Thienopyrimidinderivater, fremgangsmaader til fremstilling deraf og farmaceutiske praeparater

Country Status (8)

Country Link
US (1) US4695568A (pt)
EP (1) EP0150469B1 (pt)
JP (1) JPS60146891A (pt)
AT (1) ATE35137T1 (pt)
CA (1) CA1224782A (pt)
DE (1) DE3472106D1 (pt)
DK (1) DK165744C (pt)
HU (1) HU191161B (pt)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1307786C (en) * 1984-12-14 1992-09-22 Keiichi Yokoyama Quinazoline derivatives and antihypertensive preparations containing same as effective components
US4703120A (en) * 1986-04-28 1987-10-27 Ortho Pharmaceutical Corporation Furo(3,4-d)pyrimidine-2,4-dione derivatives and intermediates thereof
GB8912335D0 (en) * 1989-05-30 1989-07-12 Smithkline Beckman Intercredit Compounds
DE19636769A1 (de) * 1996-09-10 1998-03-12 Basf Ag 3-Substituierte Pyrido [4',3':4,5]thieno[2,3-d]pyrimidin-Derivate, ihre Herstellung und Verwendung
JPH10298078A (ja) * 1997-05-06 1998-11-10 Mitsubishi Chem Corp 抗不安薬
GB0112494D0 (en) * 2001-05-22 2001-07-11 Arachnova Therapeutics Ltd New therapeutic use
GB0216027D0 (en) 2002-07-10 2002-08-21 Arachnova Therapeutics Ltd New therapeutic use
EP1519728B1 (en) * 2002-07-10 2009-03-11 Dynogen Pharmaceuticals, Inc. 4-(2-fluorophenyl)-6-methyl-2(1-piperazinyl)thieno(2,3-d) pyrimidine in the treatment of functional bowel disorder
DE10232750A1 (de) * 2002-07-18 2004-02-05 Basf Ag Verfahren zur Herstellung von macrocyclischen Ketonen durch Dieckmann-Kondensation in der Gasphase
EP1539172A1 (en) * 2002-08-29 2005-06-15 Arachnova Therapeutics Ltd. New therapeutic uses of (4-(2-fluorophenyl)-6-methyl-2-(1-piperazinyl) thieno[2,3-d]pyrimidine
DE602004005814T2 (de) * 2003-01-13 2008-01-10 Dynogen Pharmaceuticals Inc., Waltham Verfahren zur behandlung von übelkeit, erbrechen, würgereiz oder jede kombination daraus
WO2004062623A2 (en) * 2003-01-13 2004-07-29 Dynogen Pharmaceuticals, Inc. Method of treating functional bowel disorders
EP1539181B1 (en) * 2003-04-04 2007-06-27 Dynogen Pharmaceuticals Inc. Method of treating lower urinary tract disorders
WO2005002583A1 (en) * 2003-07-07 2005-01-13 Mitsubishi Pharma Corporation Use of thieno`2,3-d ! pyrimidines for the prophylaxis or treatment of hyperactivity disorder
US20060293309A1 (en) * 2005-03-28 2006-12-28 Dynogen Pharmaceuticals, Inc. Method of treating disorders and conditions using peripherally-restricted antagonists and inhibitors
WO2007120445A1 (en) * 2006-03-31 2007-10-25 Dynogen Pharmaceuticals, Inc. SOLUBLE SALTS OF THIENO [2,3-d] PYRIMIDINE DERIVATIVES
EP2016082A2 (en) * 2006-03-31 2009-01-21 Dynogen Pharmaceuticals, Inc. Crystalline forms of 4-(2-fluorophenyl)-6-methyl-2-(piperazin-1-yl)thieno(2,3-d)pyrimidine
EP2947084B8 (en) * 2013-01-18 2021-03-10 Guangzhou Maxinovel Pharmaceuticals Co. Five-and-six-membered heterocyclic compound, and preparation method, pharmaceutical composition and use thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3883651A (en) * 1969-08-08 1975-05-13 Boehringer Sohn Ingelheim Pharmaceutical compositions containing a 2-(aminoalkylamino)-4-amino-thieno{8 3,2-d{9 pyrimidine and method of use
US4054656A (en) * 1975-09-10 1977-10-18 Mead Johnson & Company Thieno[2,3-d]pyrimidine antiallergic agents
GB1570494A (en) * 1975-11-28 1980-07-02 Ici Ltd Thienopyrimidine derivatives and their use as pesticides
ZA782648B (en) * 1977-05-23 1979-06-27 Ici Australia Ltd The prevention,control or eradication of infestations of ixodid ticks
US4471117A (en) * 1979-06-21 1984-09-11 Janssen Pharmaceutica N.V. 3,4-Dihydro-2H-pyrimido(2,1-b)benzothiazoles
JPS5692875A (en) * 1979-12-27 1981-07-27 Dainippon Pharmaceut Co Ltd 2-aminoquinazoline derivative
FI824314L (fi) * 1981-12-16 1983-06-17 Sankyo Co Thienopyrimidin-derivater, deras framstaellning och deras medicinska anvaendning
FR2521144A1 (fr) * 1982-02-08 1983-08-12 Sanofi Sa Nouveaux derives de la piperazinyl-2 phenyl-4 quinazoline possedant des proprietes antidepressives, methode de preparation desdits composes et medicaments en contenant

Also Published As

Publication number Publication date
DE3472106D1 (en) 1988-07-21
DK165744B (da) 1993-01-11
CA1224782A (en) 1987-07-28
JPH0367071B2 (pt) 1991-10-21
ATE35137T1 (de) 1988-07-15
US4695568A (en) 1987-09-22
EP0150469B1 (en) 1988-06-15
HU191161B (en) 1987-01-28
JPS60146891A (ja) 1985-08-02
DK617184D0 (da) 1984-12-20
HUT37435A (en) 1985-12-28
DK617184A (da) 1985-07-06
EP0150469A1 (en) 1985-08-07

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Legal Events

Date Code Title Description
PBP Patent lapsed