DK154180A - Fremgangsmaade til fremstilling af penem-3-carboxylsyrederivatier - Google Patents

Fremgangsmaade til fremstilling af penem-3-carboxylsyrederivatier

Info

Publication number
DK154180A
DK154180A DK154180A DK154180A DK154180A DK 154180 A DK154180 A DK 154180A DK 154180 A DK154180 A DK 154180A DK 154180 A DK154180 A DK 154180A DK 154180 A DK154180 A DK 154180A
Authority
DK
Denmark
Prior art keywords
carboxylic acid
acid derivatives
penem
preparing penem
preparing
Prior art date
Application number
DK154180A
Other languages
Danish (da)
English (en)
Inventor
E Ohki
S Oida
A Yoshida
T Hayashi
S Sugawara
Original Assignee
Sankyo Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co filed Critical Sankyo Co
Publication of DK154180A publication Critical patent/DK154180A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/09Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/18Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804Compounds having Si-O-C linkages
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/568Four-membered rings
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
DK154180A 1979-04-11 1980-04-10 Fremgangsmaade til fremstilling af penem-3-carboxylsyrederivatier DK154180A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP4405079A JPS55153789A (en) 1979-04-11 1979-04-11 Penem-3-carboxylic acid derivative and its preparation

Publications (1)

Publication Number Publication Date
DK154180A true DK154180A (da) 1980-10-12

Family

ID=12680777

Family Applications (1)

Application Number Title Priority Date Filing Date
DK154180A DK154180A (da) 1979-04-11 1980-04-10 Fremgangsmaade til fremstilling af penem-3-carboxylsyrederivatier

Country Status (16)

Country Link
JP (1) JPS55153789A (enrdf_load_stackoverflow)
AU (1) AU5729180A (enrdf_load_stackoverflow)
BE (1) BE882764A (enrdf_load_stackoverflow)
DD (1) DD152561A5 (enrdf_load_stackoverflow)
DE (1) DE3013997A1 (enrdf_load_stackoverflow)
DK (1) DK154180A (enrdf_load_stackoverflow)
ES (1) ES490510A0 (enrdf_load_stackoverflow)
FI (1) FI801168A7 (enrdf_load_stackoverflow)
FR (1) FR2453862A1 (enrdf_load_stackoverflow)
GB (1) GB2048261A (enrdf_load_stackoverflow)
IT (1) IT8067576A0 (enrdf_load_stackoverflow)
NL (1) NL8002147A (enrdf_load_stackoverflow)
NO (1) NO801046L (enrdf_load_stackoverflow)
PL (1) PL223390A1 (enrdf_load_stackoverflow)
SE (1) SE8002708L (enrdf_load_stackoverflow)
ZA (1) ZA802155B (enrdf_load_stackoverflow)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5625110A (en) * 1978-12-18 1981-03-10 Bristol Myers Co Antibacterial
DE3176517D1 (en) * 1980-04-24 1987-12-17 Beecham Group Plc Beta-lactam compounds, their preparation and use
JPS58198486A (ja) * 1982-05-14 1983-11-18 Sankyo Co Ltd ペネムまたはカルバペネム−3−カルボン酸誘導体およびその製法
JPS5835190A (ja) 1981-08-25 1983-03-01 Sankyo Co Ltd ペネム−3−カルボン酸誘導体
JPS5857360A (ja) * 1981-10-01 1983-04-05 Ajinomoto Co Inc アゼチジノン誘導体
CA1190236A (en) 1981-10-23 1985-07-09 Edward J.J. Grabowski Antibiotic synthesis
AU556854B2 (en) * 1981-12-11 1986-11-20 Farmitalia Carlo Erba S.P.A. Method for preparing penems derivatives
US4431654A (en) * 1982-04-05 1984-02-14 Schering Corporation 6-(Hydroxyethyl)-2-[(heterocyclyl or aryl)thioalkylthio]-penem-3-carboxylates
US4610823A (en) * 1983-01-25 1986-09-09 Merck & Co., Inc. Process for preparing substituted 2-thioxopenams and 2-substituted thiopenems
EP0115308A3 (en) * 1983-01-25 1984-10-10 Merck & Co. Inc. 2-unsaturated alkylthio-pen-2-em-3-carboxylic acids and process for preparing substituted 2-thioxopenams and 2-substituted thiopenems
US4504485A (en) * 1983-04-04 1985-03-12 Schering Corporation 5R,6S,8R-6-(1-Hydroxyethyl)-2-(2-carbamoyloxyethylthio)-penem-3-carboxylic acid
GB8321004D0 (en) * 1983-08-04 1983-09-07 Erba Farmitalia Azetidinones
US5075439A (en) * 1990-08-17 1991-12-24 Pfizer Inc. Processes for (3S,4R)-3-[1(R)-t-butyl-dimethylsilyloxy)-ethyl]-4-[1-oxo-3-thiolanylthio(thiocarbonyl)thio]azetidin-2-ones and intermediates therefor
GB2252769A (en) * 1991-01-18 1992-08-19 Pfizer Improved process for azetidin-2-ones and intermediates therefor
GB9103034D0 (en) * 1991-02-13 1991-03-27 Fujisawa Pharmaceutical Co Processes for preparing carbapenem derivatives
GB9913932D0 (en) * 1999-06-15 1999-08-18 Pfizer Ltd Purine derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3950357A (en) * 1974-11-25 1976-04-13 Merck & Co., Inc. Antibiotics
US4168314A (en) * 1977-11-17 1979-09-18 Merck & Co., Inc. 6-(1'-Hydroxyethyl)-2-aminoethylthio-pen-2-em-3-carboxylic acid
EP0003960B1 (de) * 1978-02-02 1983-06-29 Ciba-Geigy Ag 6-Substituierte Thia-Azaverbindungen, ihre Herstellung und diese enthaltende pharmazeutische Präparate
IL59081A0 (en) * 1979-01-10 1980-05-30 Schering Corp 2-penem compounds and a method for preparing them

Also Published As

Publication number Publication date
ES8202015A1 (es) 1981-04-16
PL223390A1 (enrdf_load_stackoverflow) 1981-01-30
ES490510A0 (es) 1981-04-16
GB2048261A (en) 1980-12-10
ZA802155B (en) 1981-05-27
BE882764A (fr) 1980-10-13
NL8002147A (nl) 1980-10-14
DD152561B2 (de) 1981-12-02
NO801046L (no) 1980-10-13
DD152561A5 (de) 1981-12-02
IT8067576A0 (it) 1980-04-11
JPS55153789A (en) 1980-11-29
AU5729180A (en) 1980-10-16
JPH0372630B2 (enrdf_load_stackoverflow) 1991-11-19
FI801168A7 (fi) 1981-01-01
DE3013997A1 (de) 1980-10-30
SE8002708L (sv) 1980-10-12
FR2453862A1 (fr) 1980-11-07

Similar Documents

Publication Publication Date Title
DK156056C (da) Analogifremgangsmaade til fremstilling af 4-amino-3-quinolin-carboxylsyrederivater
DK478980A (da) Fremgangsmaade til fremstilling af imidazol-5-eddikesyrederivater
DK540080A (da) Fremgangsmaade til fremstilling af 2-amino-4-hydroxyquinazolinderivater
DK149080C (da) Fremgangsmaade til fremstilling af derivater af ml-236b-carboxylsyre
DK157760C (da) Fremgangsmaade til fremstilling af 7-(substitueret)-amino-3-substitueret-thiomethyl-cephemcarboxylsyrer
DK156828C (da) Fremgangsmaade til fremstilling af cyclopropancarboxylsyreesterderivater
DK154180A (da) Fremgangsmaade til fremstilling af penem-3-carboxylsyrederivatier
DK157009C (da) Fremgangsmaade til fremstilling af 1-(3-mercapto-2s-methylpropionyl)-pyrrolidin-2s-carboxylsyre
DK380681A (da) Fremgangsmaade til fremstilling af kinolinkarboxylsyrederivater
DK158669C (da) Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater.
DK99980A (da) Fremgangsmaade til fremstilling af mercaptoacyldihydropyrazolcarboxylsyrederivater
DK396880A (da) Fremgangsmaade til fremstilling af cyclohexancarboxylsyrederivater
DK170382A (da) Fremgangsmaade til fremstilling af phenylaliphatiske carboxylsyrederivater
DK157843C (da) Fremgangsmaade til fremstilling af 2-hydroxynaphthalen-6-carboxylsyre
DK193680A (da) Fremgangsmaade til fremstilling af 2-hydroxy-5-(1-hydroxy-2-piperazinylethyl) benzoesyrederivater
DK157677C (da) Fremgangsmaade til fremstilling af cyclopropancarboxylsyreesterderivater
DK154554C (da) Fremgangsmaade til fremstilling af alfa-methyl-carbazol-2-eddikesyrederivater
DK154085C (da) Fremgangsmaade til fremstilling af 1,1-dioxopenicillansyrederivater
DK444279A (da) Fremgangsmaade til fremstilling af 6-hydroxymethyl-2-(beta-aminoethylthio)-1-carbadethiapen-2-em-3-carboxylsyre
DK429779A (da) Fremgangsmaade til fremstilling af cyklopropancarboxylsyreestere
DK163667C (da) Fremgangsmaade til fremstilling af 7-amino-3-chlor-3-cephem-4-carboxylsyreestere
DK144277C (da) Fremgangsmaade til fremstilling af 6-aminopenicillansyre
DK57381A (da) Fremgansmaade til fremstilling af bifenyloxypropionsyrederivater
DK145741C (da) Fremgangsmaade til fremstilling af 6-chlor-alfa-methyl-carbazol-2-eddikesyre
DK157613C (da) Fremgangsmaade til fremstilling af cyclopropancarboxylsyreesterderivater

Legal Events

Date Code Title Description
PBP Patent lapsed