DK1434570T3 - Farmaceutiske formuleringer til kontrolleret frigivelse af 4-amino-6,7-dimethoxy-2-(5-methansulfonamido-1,2,3,4-tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazolin - Google Patents

Farmaceutiske formuleringer til kontrolleret frigivelse af 4-amino-6,7-dimethoxy-2-(5-methansulfonamido-1,2,3,4-tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazolin

Info

Publication number
DK1434570T3
DK1434570T3 DK02775048T DK02775048T DK1434570T3 DK 1434570 T3 DK1434570 T3 DK 1434570T3 DK 02775048 T DK02775048 T DK 02775048T DK 02775048 T DK02775048 T DK 02775048T DK 1434570 T3 DK1434570 T3 DK 1434570T3
Authority
DK
Denmark
Prior art keywords
tetrahydroisoquinol
methanesulfonamido
quinazoline
dimethoxy
pyridyl
Prior art date
Application number
DK02775048T
Other languages
Danish (da)
English (en)
Inventor
John D Davis
Michael J Humphrey
Ross J Macrae
Janet S Smith
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of DK1434570T3 publication Critical patent/DK1434570T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5026Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Urology & Nephrology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK02775048T 2001-10-11 2002-09-30 Farmaceutiske formuleringer til kontrolleret frigivelse af 4-amino-6,7-dimethoxy-2-(5-methansulfonamido-1,2,3,4-tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazolin DK1434570T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0124455.7A GB0124455D0 (en) 2001-10-11 2001-10-11 Pharmaceutical formulations

Publications (1)

Publication Number Publication Date
DK1434570T3 true DK1434570T3 (da) 2005-11-07

Family

ID=9923660

Family Applications (1)

Application Number Title Priority Date Filing Date
DK02775048T DK1434570T3 (da) 2001-10-11 2002-09-30 Farmaceutiske formuleringer til kontrolleret frigivelse af 4-amino-6,7-dimethoxy-2-(5-methansulfonamido-1,2,3,4-tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazolin

Country Status (32)

Country Link
EP (1) EP1434570B8 (no)
JP (1) JP4131471B2 (no)
KR (1) KR20050032510A (no)
CN (1) CN1568180A (no)
AP (1) AP2004003001A0 (no)
AR (1) AR036782A1 (no)
AT (1) ATE303135T1 (no)
BR (1) BR0213196A (no)
CA (1) CA2461168A1 (no)
CO (1) CO5560534A2 (no)
DE (1) DE60205925T2 (no)
DK (1) DK1434570T3 (no)
DO (1) DOP2002000464A (no)
EA (1) EA006168B1 (no)
ES (1) ES2246017T3 (no)
GB (1) GB0124455D0 (no)
GT (1) GT200200184A (no)
HR (1) HRP20040261A2 (no)
HU (1) HUP0600064A3 (no)
IL (1) IL160969A0 (no)
IS (1) IS7179A (no)
MA (1) MA27075A1 (no)
MX (1) MXPA04003293A (no)
NO (1) NO20041520L (no)
OA (1) OA12709A (no)
PA (1) PA8556001A1 (no)
PE (1) PE20030551A1 (no)
PL (1) PL369666A1 (no)
SV (1) SV2004001279A (no)
UY (1) UY27477A1 (no)
WO (1) WO2003032956A1 (no)
ZA (1) ZA200401976B (no)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0317663D0 (en) * 2003-07-29 2003-09-03 Astrazeneca Ab Pharmaceutical composition
HUE046285T2 (hu) 2013-03-14 2020-02-28 Amgen Inc Omecamtiv mecarbil sói és eljárás a só elõállítására
KR101943592B1 (ko) 2017-08-31 2019-01-30 조현우 데이터 마이닝 기법을 이용한 전자가계부 시스템

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69008526T2 (de) * 1990-07-02 1994-08-18 Bend Res Inc Asymmetrische mikroporöse Kügelchen für regulierbare Freigabe.
FR2752737B1 (fr) * 1996-08-29 1998-10-02 Synthelabo Comprime a liberation controlee de chlorhydrate d'alfuzosine
GB9700504D0 (en) * 1997-01-11 1997-02-26 Pfizer Ltd Pharmaceutical compounds
IL141235A (en) * 2000-02-09 2012-04-30 Novartis Int Pharm Ltd Combined use of an alpha-adrenoceptor antagonist and a muscarinic antagonist in the preparation of a drug for the treatment of non-malignant prostatic hyperplasia
UA72311C2 (uk) * 2000-03-03 2005-02-15 Пфайзер Інк. Мезилат 4-аміно-6,7-диметокси-2-(5-метансульфонамідо-1,2,3,4-тетрагідроізохінол-2-іл)-5-(2-піридил)хіназоліну та поліморфні форми

Also Published As

Publication number Publication date
PE20030551A1 (es) 2003-06-26
DE60205925D1 (de) 2005-10-06
EP1434570A1 (en) 2004-07-07
HUP0600064A2 (en) 2006-06-28
HRP20040261A2 (en) 2004-08-31
KR20050032510A (ko) 2005-04-07
SV2004001279A (es) 2004-02-19
OA12709A (en) 2006-06-26
CA2461168A1 (en) 2003-04-24
GT200200184A (es) 2003-05-23
EP1434570B8 (en) 2005-10-26
MA27075A1 (fr) 2004-12-20
NO20041520L (no) 2004-04-05
EA200400431A1 (ru) 2004-08-26
EP1434570B1 (en) 2005-08-31
DE60205925T2 (de) 2006-06-08
AR036782A1 (es) 2004-10-06
BR0213196A (pt) 2004-08-31
CO5560534A2 (es) 2005-09-30
WO2003032956A1 (en) 2003-04-24
GB0124455D0 (en) 2001-12-05
JP2005507909A (ja) 2005-03-24
ATE303135T1 (de) 2005-09-15
IL160969A0 (en) 2004-08-31
CN1568180A (zh) 2005-01-19
HUP0600064A3 (en) 2007-02-28
UY27477A1 (es) 2003-05-30
IS7179A (is) 2004-03-11
DOP2002000464A (es) 2003-04-15
PL369666A1 (en) 2005-05-02
AP2004003001A0 (en) 2004-03-31
JP4131471B2 (ja) 2008-08-13
PA8556001A1 (es) 2003-07-28
ES2246017T3 (es) 2006-02-01
EA006168B1 (ru) 2005-10-27
ZA200401976B (en) 2004-07-12
MXPA04003293A (es) 2004-07-23

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