DK141996B - Analogifremgangsmåde til fremstilling af triazolobenzodiazepinderivater eller salte heraf. - Google Patents

Analogifremgangsmåde til fremstilling af triazolobenzodiazepinderivater eller salte heraf. Download PDF

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Publication number
DK141996B
DK141996B DK603471AA DK603471A DK141996B DK 141996 B DK141996 B DK 141996B DK 603471A A DK603471A A DK 603471AA DK 603471 A DK603471 A DK 603471A DK 141996 B DK141996 B DK 141996B
Authority
DK
Denmark
Prior art keywords
group
compound
benzodiazepine
triazolo
phenyl
Prior art date
Application number
DK603471AA
Other languages
Danish (da)
English (en)
Other versions
DK141996C (US07413550-20080819-C00001.png
Inventor
Kanji Meguro
Yutaka Kuwada
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of DK141996B publication Critical patent/DK141996B/da
Application granted granted Critical
Publication of DK141996C publication Critical patent/DK141996C/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK603471AA 1970-12-11 1971-12-10 Analogifremgangsmåde til fremstilling af triazolobenzodiazepinderivater eller salte heraf. DK141996B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP11071670 1970-12-11
JP45110716A JPS4932874B1 (US07413550-20080819-C00001.png) 1970-12-11 1970-12-11

Publications (2)

Publication Number Publication Date
DK141996B true DK141996B (da) 1980-08-04
DK141996C DK141996C (US07413550-20080819-C00001.png) 1980-12-15

Family

ID=14542652

Family Applications (1)

Application Number Title Priority Date Filing Date
DK603471AA DK141996B (da) 1970-12-11 1971-12-10 Analogifremgangsmåde til fremstilling af triazolobenzodiazepinderivater eller salte heraf.

Country Status (19)

Country Link
US (1) US4235775A (US07413550-20080819-C00001.png)
JP (1) JPS4932874B1 (US07413550-20080819-C00001.png)
AT (2) AT315181B (US07413550-20080819-C00001.png)
AU (1) AU453008B2 (US07413550-20080819-C00001.png)
BE (1) BE776514A (US07413550-20080819-C00001.png)
CA (1) CA975363A (US07413550-20080819-C00001.png)
CH (2) CH569735A5 (US07413550-20080819-C00001.png)
DE (2) DE2159242A1 (US07413550-20080819-C00001.png)
DK (1) DK141996B (US07413550-20080819-C00001.png)
ES (1) ES397845A1 (US07413550-20080819-C00001.png)
FI (1) FI53128C (US07413550-20080819-C00001.png)
FR (1) FR2118028B1 (US07413550-20080819-C00001.png)
GB (2) GB1374469A (US07413550-20080819-C00001.png)
HU (1) HU164524B (US07413550-20080819-C00001.png)
NL (1) NL173523C (US07413550-20080819-C00001.png)
NO (1) NO132933C (US07413550-20080819-C00001.png)
PH (1) PH10822A (US07413550-20080819-C00001.png)
YU (1) YU35141B (US07413550-20080819-C00001.png)
ZA (1) ZA718044B (US07413550-20080819-C00001.png)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4141902A (en) * 1971-04-28 1979-02-27 The Upjohn Company 1-Halomethyl-6-phenyl-4H-s-[4,3-a][1,4]benzodiazepines
GB1331015A (en) * 1971-04-28 1973-09-19 Upjohn Co 1-substituted-6-phenyl-4h-s-triazolo-4,3-a-1,4-benzodiazepines
GB1377230A (en) * 1971-09-13 1974-12-11 Upjohn Co 4h-s-triazolo -4,3-a- 1,4-benzodiazepines
US3842090A (en) * 1973-02-14 1974-10-15 Upjohn Co Certain 1-aminomethyl-6-phenyl 4h-s-triazolo(4,3-a)(1,4)benzodiazepines
US3894025A (en) * 1974-03-21 1975-07-08 Upjohn Co 1-Piperazino-6-phenyl-4H-s-triazolo{8 4,3-a{9 {8 1,4{9 -benzodiazepine compounds
CA1055490A (en) * 1974-06-19 1979-05-29 Upjohn Company (The) Process for preparing triazolobenzodiazepines
ZA755418B (en) * 1974-09-11 1977-06-29 Hoffmann La Roche Diazepine derivatives
US4021441A (en) * 1975-04-07 1977-05-03 The Upjohn Company 1-[(Allylamino)-methyl]-6-phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines
DE2609486A1 (de) * 1975-08-07 1977-05-12 Hoffmann La Roche Imidazo eckige klammer auf 1,5-a eckige klammer zu eckige klammer auf 1,4 eckige klammer zu diazepin-verbindungen und verfahren zu ihrer herstellung
US4009175A (en) * 1976-03-15 1977-02-22 The Upjohn Company 1-[(Aminooxy)-methyl]-6-substituted-4H-s-triazolo[4,3-a][1,4] benzodiazepines
US4510141A (en) * 1982-09-13 1985-04-09 Ciba-Geigy Corporation Tricyclic polyazaheterocycles for treating depression or anxiety
US4663454A (en) * 1985-04-17 1987-05-05 The Upjohn Company Process to prepare α-chloroalprazolam

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH9315A (en) * 1968-11-05 1975-08-22 K Meguro Triazolo(4,3-a)(1,4)benzodiazepine derivatives
FR2022598A1 (en) * 1969-11-04 1970-07-31 Pakeda Chemical Ind Sedative chloro-phenyl-triazolobenzodiazepines
DE2156472A1 (de) 1970-11-23 1972-05-31 Ciba-Geigy Ag, Basel (Schweiz) Verfahren zur Herstellung von neuen Diazepinderivaten
CH544764A (de) 1971-01-21 1974-01-15 Ciba Geigy Ag Verfahren zur Herstellung von neuen Triazolo-benzodiazepinderivaten
US3681343A (en) * 1971-05-11 1972-08-01 Upjohn Co 6-phenyl-s-triazolo{8 4,3-a{9 {8 1,4{9 {0 benzodiazepines

Also Published As

Publication number Publication date
AT315858B (de) 1974-06-10
CA975363A (en) 1975-09-30
NO132933C (US07413550-20080819-C00001.png) 1976-02-04
FI53128B (US07413550-20080819-C00001.png) 1977-10-31
ZA718044B (en) 1972-08-30
HU164524B (US07413550-20080819-C00001.png) 1974-02-28
CH569735A5 (US07413550-20080819-C00001.png) 1975-11-28
DE2159242A1 (de) 1972-12-07
AT315181B (de) 1974-05-10
YU35141B (en) 1980-09-25
GB1374470A (en) 1974-11-20
CH567022A5 (US07413550-20080819-C00001.png) 1975-09-30
AU453008B2 (en) 1974-09-19
DE2166657C2 (US07413550-20080819-C00001.png) 1988-10-20
US4235775A (en) 1980-11-25
GB1374469A (en) 1974-11-20
DK141996C (US07413550-20080819-C00001.png) 1980-12-15
NL173523C (nl) 1984-02-01
DE2166657A1 (de) 1975-01-23
BE776514A (fr) 1972-04-04
FR2118028A1 (US07413550-20080819-C00001.png) 1972-07-28
ES397845A1 (es) 1975-05-16
DE2159242C2 (US07413550-20080819-C00001.png) 1988-01-28
NL173523B (nl) 1983-09-01
PH10822A (en) 1977-09-08
JPS4932874B1 (US07413550-20080819-C00001.png) 1974-09-03
NO132933B (US07413550-20080819-C00001.png) 1975-10-27
YU309471A (en) 1980-03-15
AU3680271A (en) 1973-06-14
FR2118028B1 (US07413550-20080819-C00001.png) 1975-06-13
NL7116874A (US07413550-20080819-C00001.png) 1972-06-13
FI53128C (US07413550-20080819-C00001.png) 1978-02-10

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PUP Patent expired