DK139579B - Analogifremgangsmåde til fremstilling af 4-(2-(4-methyl-5-thiazolcarboxamido)ethyl)benzensulfonylurinstof-forbindelser eller basesalte deraf med farmakologisk acceptable kationer. - Google Patents

Analogifremgangsmåde til fremstilling af 4-(2-(4-methyl-5-thiazolcarboxamido)ethyl)benzensulfonylurinstof-forbindelser eller basesalte deraf med farmakologisk acceptable kationer.

Info

Publication number
DK139579B
DK139579B DK113474AA DK113474A DK139579B DK 139579 B DK139579 B DK 139579B DK 113474A A DK113474A A DK 113474AA DK 113474 A DK113474 A DK 113474A DK 139579 B DK139579 B DK 139579B
Authority
DK
Denmark
Prior art keywords
thiazolecarboxamido
benzenesulfonylurea
ethyl
methyl
compounds
Prior art date
Application number
DK113474AA
Other languages
English (en)
Other versions
DK139579C (da
Inventor
Donald Ernest Kuhla
Hans Eberhardt Wiedermann
Reinhard Sarges
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK139579B publication Critical patent/DK139579B/da
Application granted granted Critical
Publication of DK139579C publication Critical patent/DK139579C/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Hematology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Steroid Compounds (AREA)
DK113474AA 1973-03-07 1974-03-04 Analogifremgangsmåde til fremstilling af 4-(2-(4-methyl-5-thiazolcarboxamido)ethyl)benzensulfonylurinstof-forbindelser eller basesalte deraf med farmakologisk acceptable kationer. DK139579B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US00338965A US3856806A (en) 1973-03-07 1973-03-07 Thiazolecarboxamide sulfonylurea hypoglycemic agents

Publications (2)

Publication Number Publication Date
DK139579B true DK139579B (da) 1979-03-12
DK139579C DK139579C (da) 1979-08-27

Family

ID=23326893

Family Applications (1)

Application Number Title Priority Date Filing Date
DK113474AA DK139579B (da) 1973-03-07 1974-03-04 Analogifremgangsmåde til fremstilling af 4-(2-(4-methyl-5-thiazolcarboxamido)ethyl)benzensulfonylurinstof-forbindelser eller basesalte deraf med farmakologisk acceptable kationer.

Country Status (29)

Country Link
US (1) US3856806A (da)
JP (1) JPS5418258B2 (da)
AR (1) AR201135A1 (da)
AT (1) AT342614B (da)
AU (1) AU458655B2 (da)
BE (1) BE811866A (da)
BG (1) BG25376A3 (da)
CA (1) CA1015362A (da)
CH (1) CH581639A5 (da)
CS (1) CS176268B2 (da)
DD (1) DD110500A5 (da)
DE (1) DE2410003A1 (da)
DK (1) DK139579B (da)
EG (1) EG11270A (da)
ES (1) ES423865A1 (da)
FI (1) FI55034C (da)
FR (1) FR2220259B1 (da)
GB (1) GB1409518A (da)
HU (1) HU167511B (da)
IE (1) IE38955B1 (da)
IL (1) IL44230A (da)
LU (1) LU69565A1 (da)
NL (1) NL7402804A (da)
NO (1) NO140820C (da)
PL (1) PL96884B1 (da)
RO (1) RO69724A (da)
SE (1) SE393984B (da)
SU (1) SU617012A3 (da)
ZA (1) ZA741439B (da)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8714920D0 (en) * 1987-06-25 1987-07-29 Shell Int Research Thiazole derivatives

Also Published As

Publication number Publication date
PL96884B1 (pl) 1978-01-31
AU458655B2 (en) 1975-03-06
NL7402804A (da) 1974-09-10
IE38955L (en) 1974-09-07
ES423865A1 (es) 1976-03-16
CA1015362A (en) 1977-08-09
CH581639A5 (da) 1976-11-15
JPS5029557A (da) 1975-03-25
BG25376A3 (en) 1978-09-15
HU167511B (da) 1975-10-28
AR201135A1 (es) 1975-02-14
JPS5418258B2 (da) 1979-07-06
SE393984B (sv) 1977-05-31
FR2220259B1 (da) 1977-10-28
IE38955B1 (en) 1978-07-05
US3856806A (en) 1974-12-24
NO740532L (no) 1974-09-10
NO140820B (no) 1979-08-13
AT342614B (de) 1978-04-10
IL44230A (en) 1976-12-31
RO69724A (ro) 1981-04-30
FI55034C (fi) 1979-05-10
SU617012A3 (ru) 1978-07-25
FR2220259A1 (da) 1974-10-04
ATA174074A (de) 1977-08-15
BE811866A (fr) 1974-09-05
IL44230A0 (en) 1974-05-16
LU69565A1 (da) 1974-10-09
DK139579C (da) 1979-08-27
GB1409518A (en) 1975-10-08
FI55034B (fi) 1979-01-31
DE2410003A1 (de) 1974-09-26
ZA741439B (en) 1975-02-26
EG11270A (en) 1977-08-15
AU6586474A (en) 1975-03-06
NO140820C (no) 1979-11-21
DD110500A5 (da) 1974-12-20
CS176268B2 (da) 1977-06-30

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