DK136713B - Analogous process for the preparation of alpha-aryl-4-substituted piperidinoalkanol derivatives or their acid addition salts. - Google Patents
Analogous process for the preparation of alpha-aryl-4-substituted piperidinoalkanol derivatives or their acid addition salts.Info
- Publication number
- DK136713B DK136713B DK44973AA DK44973A DK136713B DK 136713 B DK136713 B DK 136713B DK 44973A A DK44973A A DK 44973AA DK 44973 A DK44973 A DK 44973A DK 136713 B DK136713 B DK 136713B
- Authority
- DK
- Denmark
- Prior art keywords
- aryl
- alpha
- preparation
- acid addition
- addition salts
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US22182172A | 1972-01-28 | 1972-01-28 |
Publications (2)
Publication Number | Publication Date |
---|---|
DK136713B true DK136713B (en) | 1977-11-14 |
DK136713C DK136713C (en) | 1978-05-01 |
Family
ID=22829539
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK44973AA DK136713B (en) | 1972-01-28 | 1973-01-26 | Analogous process for the preparation of alpha-aryl-4-substituted piperidinoalkanol derivatives or their acid addition salts. |
Country Status (26)
Country | Link |
---|---|
JP (1) | JPS5115035B2 (en) |
AR (1) | AR195314A1 (en) |
AT (2) | AT321917B (en) |
AU (1) | AU467361B2 (en) |
BE (1) | BE794597A (en) |
CA (1) | CA978946A (en) |
CH (2) | CH587820A5 (en) |
CS (1) | CS177834B2 (en) |
DD (1) | DD103239A5 (en) |
DE (1) | DE2303306C3 (en) |
DK (1) | DK136713B (en) |
ES (1) | ES410731A1 (en) |
FR (1) | FR2181690B1 (en) |
GB (1) | GB1413138A (en) |
HU (1) | HU166477B (en) |
IE (1) | IE36983B1 (en) |
IL (1) | IL41060A (en) |
LU (1) | LU66916A1 (en) |
NL (1) | NL175410C (en) |
NO (1) | NO140057C (en) |
PH (1) | PH10264A (en) |
PL (1) | PL89095B1 (en) |
SE (1) | SE382058B (en) |
SU (1) | SU464997A3 (en) |
YU (1) | YU36013B (en) |
ZA (1) | ZA728544B (en) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3941795A (en) | 1974-02-08 | 1976-03-02 | Richardson-Merrell Inc. | α-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES |
US4254129A (en) * | 1979-04-10 | 1981-03-03 | Richardson-Merrell Inc. | Piperidine derivatives |
US4254130A (en) * | 1979-04-10 | 1981-03-03 | Richardson-Merrell Inc. | Piperidine derivatives |
IT1200123B (en) * | 1985-09-27 | 1989-01-05 | Ind Chimica Srl | PROCESS FOR ALPHA PREPARATION |
US4742175A (en) * | 1986-05-07 | 1988-05-03 | Merrell Dow Pharmaceuticals Inc. | Preparation of polymorphically pure terfenadine |
JPS63101760U (en) * | 1986-12-19 | 1988-07-02 | ||
IT1205685B (en) * | 1987-05-26 | 1989-03-31 | Erregierre Spa | PROCESS FOR THE PREPARATION OF ALPHA- (ALCHYLPHENYL) -4- (HYDROXY DIPHENYLMETHYL) -1-PIPERIDINE BUTANOL |
IL93499A0 (en) * | 1989-02-28 | 1990-11-29 | Merrell Dow Pharma | Preparation of the low melting polymorphic form of terfenadine |
ZA903145B (en) * | 1989-05-01 | 1991-02-27 | Merrell Dow Pharma | Process for the preparation of the high melting polymorphic form of terfenadine |
DE3917241A1 (en) * | 1989-05-26 | 1990-11-29 | Schaper & Bruemmer Gmbh | 4- (HYDROXYDIPHENYLMETHYL) -1-PIPERIDYL-PHENYLALKANE DERIVATIVES |
US5466691A (en) * | 1991-08-09 | 1995-11-14 | Yoshitomi Pharmaceutical Industries, Ltd. | Thiophene compound |
JPH11504650A (en) * | 1995-05-08 | 1999-04-27 | ヘキスト・マリオン・ルセル・インコーポレイテツド | Alpha- (substituted alkylphenyl) -4- (hydroxydiphenylmethyl) -1-piperidinebutanol derivatives, their preparation and their use as antihistamines, antiallergic agents and bronchodilators |
ES2216191T3 (en) * | 1997-03-11 | 2004-10-16 | Aventis Pharmaceuticals Inc. | PROCEDURE FOR PREPARING ACID 4- (4- (HYDROXIDIFENYL) -1-PIPERIDINYL) -1-HYDROXIBUTE) -ALFA, ALPHA-DIMETHYLPHENYLACETIC AND PHOSPHORILE DERIVATIVES. |
US7498345B2 (en) * | 2004-09-17 | 2009-03-03 | Albany Molecular Research, Inc. | Process for production of piperidine derivatives |
US8153385B2 (en) | 2004-10-18 | 2012-04-10 | Reverse Proteomics Research Institute Co., Ltd. | Target protein and target gene in drug designing and screening method |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3081303A (en) * | 1961-10-13 | 1963-03-12 | Searle & Co | 1-aminoalkyl-alpha, alpha-diphenylpiperidine-methanols |
GB1242169A (en) * | 1969-04-09 | 1971-08-11 | Ucb Sa | Piperidine derivatives |
-
1972
- 1972-12-04 ZA ZA728544A patent/ZA728544B/en unknown
- 1972-12-05 IE IE1689/72A patent/IE36983B1/en unknown
- 1972-12-08 PH PH14156A patent/PH10264A/en unknown
- 1972-12-11 AU AU49893/72A patent/AU467361B2/en not_active Ceased
- 1972-12-12 IL IL41060A patent/IL41060A/en unknown
- 1972-12-15 GB GB5799572A patent/GB1413138A/en not_active Expired
- 1972-12-20 CH CH1854272A patent/CH587820A5/xx not_active IP Right Cessation
- 1972-12-20 CH CH1381476A patent/CH593259A5/xx not_active IP Right Cessation
- 1972-12-27 JP JP47130136A patent/JPS5115035B2/ja not_active Expired
- 1972-12-29 AT AT1115372A patent/AT321917B/en not_active IP Right Cessation
- 1972-12-29 AT AT246074*1A patent/AT323742B/en not_active IP Right Cessation
-
1973
- 1973-01-08 YU YU34/73A patent/YU36013B/en unknown
- 1973-01-16 CA CA161,413A patent/CA978946A/en not_active Expired
- 1973-01-17 HU HURI498A patent/HU166477B/hu unknown
- 1973-01-18 ES ES410731A patent/ES410731A1/en not_active Expired
- 1973-01-22 NL NLAANVRAGE7300873,A patent/NL175410C/en not_active IP Right Cessation
- 1973-01-24 DE DE2303306A patent/DE2303306C3/en not_active Expired
- 1973-01-24 SE SE7300974A patent/SE382058B/en active Protection Beyond IP Right Term
- 1973-01-24 FR FR7302503A patent/FR2181690B1/fr not_active Expired
- 1973-01-25 DD DD168482A patent/DD103239A5/xx unknown
- 1973-01-26 DK DK44973AA patent/DK136713B/en not_active IP Right Cessation
- 1973-01-26 BE BE794597D patent/BE794597A/en not_active IP Right Cessation
- 1973-01-26 LU LU66916A patent/LU66916A1/xx unknown
- 1973-01-26 PL PL1973160419A patent/PL89095B1/pl unknown
- 1973-01-26 NO NO326/73A patent/NO140057C/en unknown
- 1973-01-26 CS CS630A patent/CS177834B2/cs unknown
- 1973-01-26 AR AR246313A patent/AR195314A1/en active
- 1973-01-27 SU SU1878074A patent/SU464997A3/en active
Also Published As
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PUP | Patent expired |