DK136654B - Analogifremgangsmade til fremstilling af azepinderivater eller salte deraf - Google Patents

Analogifremgangsmade til fremstilling af azepinderivater eller salte deraf

Info

Publication number
DK136654B
DK136654B DK394071AA DK394071A DK136654B DK 136654 B DK136654 B DK 136654B DK 394071A A DK394071A A DK 394071AA DK 394071 A DK394071 A DK 394071A DK 136654 B DK136654 B DK 136654B
Authority
DK
Denmark
Prior art keywords
salts
preparation
azepin
derivatives
analogical procedure
Prior art date
Application number
DK394071AA
Other languages
English (en)
Other versions
DK136654C (da
Inventor
G Griss
M Kleemann
W Grell
H Ballhause
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE2040510A external-priority patent/DE2040510C3/de
Priority claimed from DE19712127267 external-priority patent/DE2127267A1/de
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of DK136654B publication Critical patent/DK136654B/da
Application granted granted Critical
Publication of DK136654C publication Critical patent/DK136654C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
DK394071A 1970-08-14 1971-08-12 Analogifremgangsmaade til fremstilling af azepinderivater eller salte deraf DK136654C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE2040510A DE2040510C3 (de) 1970-08-14 1970-08-14 Oxazole- und Thiazole eckige Klammer auf 5,4-d] azepin- Derivate
DE19712127267 DE2127267A1 (en) 1971-06-02 1971-06-02 2-amino-4,5,7,8-tetrahydro-6h-thiazolo-or oxazolo(5,4-d) - azepines - as hypotensive, antiphlogistic, sedative and bechic agents

Publications (2)

Publication Number Publication Date
DK136654B true DK136654B (da) 1977-11-07
DK136654C DK136654C (da) 1978-04-10

Family

ID=25759588

Family Applications (1)

Application Number Title Priority Date Filing Date
DK394071A DK136654C (da) 1970-08-14 1971-08-12 Analogifremgangsmaade til fremstilling af azepinderivater eller salte deraf

Country Status (23)

Country Link
US (1) US3804849A (da)
JP (1) JPS5246236B1 (da)
AT (1) AT310174B (da)
AU (1) AU462319B2 (da)
BE (1) BE771330A (da)
BG (3) BG17786A3 (da)
CA (1) CA965423A (da)
CH (1) CH571003A5 (da)
CS (1) CS178084B2 (da)
DK (1) DK136654C (da)
ES (3) ES393881A1 (da)
FI (1) FI54925C (da)
FR (1) FR2102192B1 (da)
GB (1) GB1321509A (da)
HU (1) HU162343B (da)
IE (1) IE35517B1 (da)
IL (1) IL37492A (da)
NL (1) NL168516C (da)
NO (1) NO131887C (da)
PL (1) PL85080B1 (da)
RO (4) RO60635A (da)
SE (1) SE380529B (da)
YU (5) YU35027B (da)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3907996A (en) * 1970-08-14 1975-09-23 Boehringer Sohn Ingelheim Pharmaceutical composition containing a 2-amino-4,5,7,8-tetrahydro-6H-thiazolo or -oxazolo 5,4-D azepine and method of use
BE795257A (fr) * 1972-02-10 1973-08-09 Thomae Gmbh Dr K Nouveaux oxazols
DE2820808A1 (de) * 1978-05-12 1979-11-22 Thomae Gmbh Dr K Arzneimittel mit einer antanginoesen wirksamkeit
US4400378A (en) * 1981-11-02 1983-08-23 Karl Thomae Gesellschaft Mit Beschrankter Haftung Pharmaceutical composition for the treatment of glaucoma
EP0192098B1 (de) 1985-02-06 1991-08-21 Boehringer Ingelheim Kg Verwendung des 2-Amino-6-allyl-5,6,7,8-tetrahydro-4H-thiazolo[4,5-d]azepins zur Herstellung eines zur Behandlung der Parkinsonschen Erkrankung bzw. des Parkinsonismus geeigneten Arzneimittels
US4826686A (en) * 1985-12-14 1989-05-02 Boehringer Ingelheim Kg Therapeutic system
DE3820775A1 (de) * 1988-06-20 1989-12-21 Thomae Gmbh Dr K Neue 4,5,7,8-tetrahydro-6h-thiazolo(5,4,-d)azepine, ihre herstellung und ihre verwendung als arzneimittel
JP3054738B2 (ja) * 1988-07-22 2000-06-19 武田薬品工業株式会社 チアゾロ[5,4―b]アゼピン誘導体
US5424431A (en) * 1990-10-24 1995-06-13 Yamanouchi Pharmaceutical Co., Ltd. Thiazole derivatives
US6369222B1 (en) * 2000-07-18 2002-04-09 Hoffmann-La Roche Inc. mGluR antagonists and a method for their synthesis
BRPI0619159B1 (pt) * 2005-12-08 2016-04-12 Huntsman Int Llc processo para a preparação de diamino difenil metano e poli-(diamino difenil metano), e, processo para a preparação de metileno difenileno diisocianato e poli-(metileno difenileno diisocianato)
EP2236511A4 (en) 2007-12-21 2011-04-13 Alla Chem Llc LIGANDS OF ALPHA ADRENOCEPTORS AND OF DOPAMINE, HISTAMIN, IMIDAZOLIN AND SEROTONIN RECEPTORS AND THEIR APPLICATION THEREOF
RU2374245C1 (ru) 2008-08-22 2009-11-27 Андрей Александрович Иващенко Лиганд с широким спектром одновременной рецепторной активности, фармацевтическая композиция, способ ее получения и лекарственное средство
EP2327704A4 (en) * 2008-08-29 2012-05-09 Shionogi & Co RING-CONDENSED AZOL DERIVATIVE WITH PI3K-INHIBITING EFFECT
TWI537274B (zh) 2011-03-14 2016-06-11 橘生藥品工業股份有限公司 新穎之八氫噻吩并喹啉衍生物、含有其之醫藥組成物及該等之用途
WO2014092006A1 (ja) 2012-12-10 2014-06-19 キッセイ薬品工業株式会社 新規なオクタヒドロピリドキナゾリン誘導体、それを含有する医薬組成物およびそれらの用途
CN104031072A (zh) * 2014-06-24 2014-09-10 重庆植恩药业有限公司 一种盐酸他利克索的制备方法

Also Published As

Publication number Publication date
DK136654C (da) 1978-04-10
BG17786A3 (da) 1973-12-25
YU35027B (en) 1980-06-30
IE35517B1 (en) 1976-03-03
RO59925A (da) 1976-08-15
FR2102192A1 (da) 1972-04-07
FI54925C (fi) 1979-04-10
IL37492A (en) 1974-03-14
BE771330A (da) 1972-02-14
ES396453A1 (es) 1974-05-16
YU288378A (en) 1979-12-31
AT310174B (de) 1973-09-25
YU35029B (en) 1980-06-30
NO131887C (da) 1975-08-20
NL168516B (nl) 1981-11-16
IE35517L (en) 1972-02-14
YU35028B (en) 1980-06-30
FI54925B (fi) 1978-12-29
CH571003A5 (da) 1975-12-31
CS178084B2 (da) 1977-08-31
NO131887B (da) 1975-05-12
ES393881A1 (es) 1973-09-16
RO59127A (da) 1976-02-15
RO60635A (da) 1976-10-15
AU3241171A (en) 1973-02-22
NL7111176A (da) 1972-02-16
PL85080B1 (da) 1976-04-30
ES396454A1 (es) 1974-05-16
BG17968A3 (da) 1974-03-05
SE380529B (sv) 1975-11-10
HU162343B (da) 1973-01-29
FR2102192B1 (da) 1974-11-15
JPS5246236B1 (da) 1977-11-22
YU288478A (en) 1982-06-30
IL37492A0 (en) 1971-11-29
YU42168B (en) 1988-06-30
YU208471A (en) 1979-12-31
GB1321509A (en) 1973-06-27
CA965423A (en) 1975-04-01
BG17785A3 (da) 1973-12-25
US3804849A (en) 1974-04-16
YU288278A (en) 1982-06-30
NL168516C (nl) 1982-04-16
RO59129A (da) 1976-01-15
AU462319B2 (en) 1975-06-19
YU288178A (en) 1979-12-31
YU40542B (en) 1986-02-28

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Legal Events

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PUP Patent expired