BG17968A3 - Метод за получаване на производни на азепина - Google Patents

Метод за получаване на производни на азепина

Info

Publication number
BG17968A3
BG17968A3 BG018197A BG1819771A BG17968A3 BG 17968 A3 BG17968 A3 BG 17968A3 BG 018197 A BG018197 A BG 018197A BG 1819771 A BG1819771 A BG 1819771A BG 17968 A3 BG17968 A3 BG 17968A3
Authority
BG
Bulgaria
Prior art keywords
obtaining
azepine derivatives
azepine
derivatives
obtaining azepine
Prior art date
Application number
BG018197A
Other languages
English (en)
Inventor
Gerhard Griss
Manfred Kleemann
Wolfgang Grell
Helmut Ballhause
Original Assignee
Dr. Karl Thomae Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE2040510A external-priority patent/DE2040510C3/de
Priority claimed from DE19712127267 external-priority patent/DE2127267A1/de
Application filed by Dr. Karl Thomae Gmbh filed Critical Dr. Karl Thomae Gmbh
Publication of BG17968A3 publication Critical patent/BG17968A3/bg

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BG018197A 1970-08-14 1971-07-30 Метод за получаване на производни на азепина BG17968A3 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE2040510A DE2040510C3 (de) 1970-08-14 1970-08-14 Oxazole- und Thiazole eckige Klammer auf 5,4-d] azepin- Derivate
DE19712127267 DE2127267A1 (en) 1971-06-02 1971-06-02 2-amino-4,5,7,8-tetrahydro-6h-thiazolo-or oxazolo(5,4-d) - azepines - as hypotensive, antiphlogistic, sedative and bechic agents

Publications (1)

Publication Number Publication Date
BG17968A3 true BG17968A3 (bg) 1974-03-05

Family

ID=25759588

Family Applications (3)

Application Number Title Priority Date Filing Date
BG018197A BG17968A3 (bg) 1970-08-14 1971-07-30 Метод за получаване на производни на азепина
BG019141A BG17785A3 (bg) 1970-08-14 1971-07-30 Метод за получаване на нови азетинови производни
BG019142A BG17786A3 (bg) 1970-08-14 1971-07-30 Метод за получаване на нови производни на азепина

Family Applications After (2)

Application Number Title Priority Date Filing Date
BG019141A BG17785A3 (bg) 1970-08-14 1971-07-30 Метод за получаване на нови азетинови производни
BG019142A BG17786A3 (bg) 1970-08-14 1971-07-30 Метод за получаване на нови производни на азепина

Country Status (23)

Country Link
US (1) US3804849A (bg)
JP (1) JPS5246236B1 (bg)
AT (1) AT310174B (bg)
AU (1) AU462319B2 (bg)
BE (1) BE771330A (bg)
BG (3) BG17968A3 (bg)
CA (1) CA965423A (bg)
CH (1) CH571003A5 (bg)
CS (1) CS178084B2 (bg)
DK (1) DK136654C (bg)
ES (3) ES393881A1 (bg)
FI (1) FI54925C (bg)
FR (1) FR2102192B1 (bg)
GB (1) GB1321509A (bg)
HU (1) HU162343B (bg)
IE (1) IE35517B1 (bg)
IL (1) IL37492A (bg)
NL (1) NL168516C (bg)
NO (1) NO131887C (bg)
PL (1) PL85080B1 (bg)
RO (4) RO59925A (bg)
SE (1) SE380529B (bg)
YU (5) YU35027B (bg)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3907996A (en) * 1970-08-14 1975-09-23 Boehringer Sohn Ingelheim Pharmaceutical composition containing a 2-amino-4,5,7,8-tetrahydro-6H-thiazolo or -oxazolo 5,4-D azepine and method of use
BE795257A (fr) * 1972-02-10 1973-08-09 Thomae Gmbh Dr K Nouveaux oxazols
DE2820808A1 (de) * 1978-05-12 1979-11-22 Thomae Gmbh Dr K Arzneimittel mit einer antanginoesen wirksamkeit
US4400378A (en) * 1981-11-02 1983-08-23 Karl Thomae Gesellschaft Mit Beschrankter Haftung Pharmaceutical composition for the treatment of glaucoma
EP0192098B1 (de) 1985-02-06 1991-08-21 Boehringer Ingelheim Kg Verwendung des 2-Amino-6-allyl-5,6,7,8-tetrahydro-4H-thiazolo[4,5-d]azepins zur Herstellung eines zur Behandlung der Parkinsonschen Erkrankung bzw. des Parkinsonismus geeigneten Arzneimittels
US4826686A (en) * 1985-12-14 1989-05-02 Boehringer Ingelheim Kg Therapeutic system
DE3820775A1 (de) * 1988-06-20 1989-12-21 Thomae Gmbh Dr K Neue 4,5,7,8-tetrahydro-6h-thiazolo(5,4,-d)azepine, ihre herstellung und ihre verwendung als arzneimittel
JP3054738B2 (ja) * 1988-07-22 2000-06-19 武田薬品工業株式会社 チアゾロ[5,4―b]アゼピン誘導体
US5424431A (en) * 1990-10-24 1995-06-13 Yamanouchi Pharmaceutical Co., Ltd. Thiazole derivatives
US6369222B1 (en) * 2000-07-18 2002-04-09 Hoffmann-La Roche Inc. mGluR antagonists and a method for their synthesis
EP1960346B2 (en) * 2005-12-08 2019-03-27 Huntsman International Llc Process for preparing diaminodiphenylmethanes
WO2009082268A2 (ru) 2007-12-21 2009-07-02 Alla Chem, Llc ЛИГАНДЫ α-АДРЕНОЦЕПТОРОВ, ДОПАМИНОВЫХ, ГИСТАМИНОВЫХ, ИМИДАЗОЛИНОВЫХ И СЕРОТОНИНОВЫХ РЕЦЕПТОРОВ И ИХ ПРИМЕНЕНИЕ
RU2374245C1 (ru) 2008-08-22 2009-11-27 Андрей Александрович Иващенко Лиганд с широким спектром одновременной рецепторной активности, фармацевтическая композиция, способ ее получения и лекарственное средство
JPWO2010024258A1 (ja) * 2008-08-29 2012-01-26 塩野義製薬株式会社 Pi3k阻害活性を有する縮環アゾール誘導体
TWI537274B (zh) 2011-03-14 2016-06-11 橘生藥品工業股份有限公司 新穎之八氫噻吩并喹啉衍生物、含有其之醫藥組成物及該等之用途
EP2930175A4 (en) 2012-12-10 2016-12-21 Kissei Pharmaceutical NOVEL OCTAHYDROPYRIDOQUINAZOLINE DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USES THEREFOR, AND THE DERIVATIVE THEREOF
CN104031072A (zh) * 2014-06-24 2014-09-10 重庆植恩药业有限公司 一种盐酸他利克索的制备方法

Also Published As

Publication number Publication date
CA965423A (en) 1975-04-01
HU162343B (bg) 1973-01-29
IE35517B1 (en) 1976-03-03
RO60635A (bg) 1976-10-15
NO131887B (bg) 1975-05-12
RO59127A (bg) 1976-02-15
YU35028B (en) 1980-06-30
RO59925A (bg) 1976-08-15
NL168516B (nl) 1981-11-16
DK136654B (da) 1977-11-07
GB1321509A (en) 1973-06-27
FR2102192B1 (bg) 1974-11-15
YU35029B (en) 1980-06-30
YU288378A (en) 1979-12-31
BG17785A3 (bg) 1973-12-25
JPS5246236B1 (bg) 1977-11-22
AU3241171A (en) 1973-02-22
YU35027B (en) 1980-06-30
ES396453A1 (es) 1974-05-16
US3804849A (en) 1974-04-16
IE35517L (en) 1972-02-14
YU208471A (en) 1979-12-31
FI54925C (fi) 1979-04-10
YU42168B (en) 1988-06-30
FI54925B (fi) 1978-12-29
AU462319B2 (en) 1975-06-19
AT310174B (de) 1973-09-25
NL168516C (nl) 1982-04-16
ES393881A1 (es) 1973-09-16
DK136654C (da) 1978-04-10
NO131887C (bg) 1975-08-20
ES396454A1 (es) 1974-05-16
YU40542B (en) 1986-02-28
FR2102192A1 (bg) 1972-04-07
BE771330A (bg) 1972-02-14
YU288478A (en) 1982-06-30
SE380529B (sv) 1975-11-10
YU288178A (en) 1979-12-31
IL37492A (en) 1974-03-14
CS178084B2 (bg) 1977-08-31
PL85080B1 (bg) 1976-04-30
CH571003A5 (bg) 1975-12-31
IL37492A0 (en) 1971-11-29
BG17786A3 (bg) 1973-12-25
YU288278A (en) 1982-06-30
RO59129A (bg) 1976-01-15
NL7111176A (bg) 1972-02-16

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