DK135895B - Analogifremgangsmåde til fremstilling af derivater af 4'-fluor-4-(4-(alfa-hydroxybenzyl)piperidino)butyrophenoner. - Google Patents
Analogifremgangsmåde til fremstilling af derivater af 4'-fluor-4-(4-(alfa-hydroxybenzyl)piperidino)butyrophenoner.Info
- Publication number
- DK135895B DK135895B DK582171AA DK582171A DK135895B DK 135895 B DK135895 B DK 135895B DK 582171A A DK582171A A DK 582171AA DK 582171 A DK582171 A DK 582171A DK 135895 B DK135895 B DK 135895B
- Authority
- DK
- Denmark
- Prior art keywords
- butyrophenones
- hydroxybenzyl
- piperidino
- fluoro
- alpha
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US9349570A | 1970-11-27 | 1970-11-27 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK135895B true DK135895B (da) | 1977-07-11 |
| DK135895C DK135895C (da) | 1977-12-12 |
Family
ID=22239276
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK582171AA DK135895B (da) | 1970-11-27 | 1971-11-26 | Analogifremgangsmåde til fremstilling af derivater af 4'-fluor-4-(4-(alfa-hydroxybenzyl)piperidino)butyrophenoner. |
Country Status (16)
| Country | Link |
|---|---|
| JP (1) | JPS5623985B2 (da) |
| BE (1) | BE775593A (da) |
| CA (1) | CA957376A (da) |
| CH (1) | CH562215A5 (da) |
| DE (1) | DE2158136C2 (da) |
| DK (1) | DK135895B (da) |
| ES (1) | ES397370A1 (da) |
| FR (1) | FR2115451B1 (da) |
| GB (1) | GB1314955A (da) |
| IE (1) | IE35778B1 (da) |
| IL (1) | IL38079A (da) |
| NL (1) | NL175411C (da) |
| NO (1) | NO135248C (da) |
| PH (1) | PH9306A (da) |
| SE (1) | SE369900B (da) |
| ZA (1) | ZA717147B (da) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK152669B (da) * | 1979-02-09 | 1988-04-11 | Richardson Merrell Inc | Analogifremgangsmaade til fremstilling af 4-(naphthyl-methyl)-piperidin-derivater eller farmaceutisk acceptable syreadditionssalte deraf samt forbindelser til anvendelse som udgangsmaterialer ved fremgangsmaaden |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE7409245L (da) * | 1973-07-19 | 1975-01-20 | Robins Co Inc A H | |
| IE49998B1 (en) * | 1979-08-06 | 1986-01-22 | Merrell Dow Pharma | 4-(naphthalenyloxy)piperidine derivatives |
| US4283404A (en) * | 1979-09-04 | 1981-08-11 | Richardson-Merrell Inc. | Aroylethenylpiperidinobutyrophenone antipsychotic agents |
| US4284636A (en) * | 1979-09-04 | 1981-08-18 | Richardson-Merrell Inc. | Cinnamoylpiperidinobutyrophenone antipsychotic agents |
| ZA806501B (en) * | 1979-10-27 | 1981-10-28 | Richardson Merrell Inc | 4-(4-alkyl-aroyl-1-piperidino)butyrophenone antipsychotic agents |
| CA1280421C (en) * | 1985-07-02 | 1991-02-19 | Albert A. Carr | 1,4-disubstituted piperidinyl derivatives |
| US4783471A (en) * | 1985-07-02 | 1988-11-08 | Merrell Dow Pharmaceuticals Inc. | N-aralkyl piperidine methanol derivatives and the uses thereof |
| IL117149A0 (en) * | 1995-02-23 | 1996-06-18 | Schering Corp | Muscarinic antagonists |
| WO2006031764A2 (en) * | 2004-09-13 | 2006-03-23 | Bayer Cropscience Ag | Processes for prepating n-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and intermediates |
-
1971
- 1971-10-26 ZA ZA717147A patent/ZA717147B/xx unknown
- 1971-10-27 IE IE1361/71A patent/IE35778B1/xx unknown
- 1971-10-27 GB GB4994271A patent/GB1314955A/en not_active Expired
- 1971-10-29 CA CA126,448A patent/CA957376A/en not_active Expired
- 1971-11-04 IL IL38079A patent/IL38079A/xx unknown
- 1971-11-16 PH PH13014*UA patent/PH9306A/en unknown
- 1971-11-17 CH CH1670071A patent/CH562215A5/xx not_active IP Right Cessation
- 1971-11-18 JP JP9200371A patent/JPS5623985B2/ja not_active Expired
- 1971-11-19 BE BE775593A patent/BE775593A/xx not_active IP Right Cessation
- 1971-11-24 DE DE2158136A patent/DE2158136C2/de not_active Expired
- 1971-11-24 NO NO4318/71A patent/NO135248C/no unknown
- 1971-11-24 SE SE15032/71A patent/SE369900B/xx unknown
- 1971-11-25 NL NLAANVRAGE7116194,A patent/NL175411C/xx not_active IP Right Cessation
- 1971-11-26 DK DK582171AA patent/DK135895B/da not_active IP Right Cessation
- 1971-11-26 FR FR7142529A patent/FR2115451B1/fr not_active Expired
- 1971-11-26 ES ES397370A patent/ES397370A1/es not_active Expired
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK152669B (da) * | 1979-02-09 | 1988-04-11 | Richardson Merrell Inc | Analogifremgangsmaade til fremstilling af 4-(naphthyl-methyl)-piperidin-derivater eller farmaceutisk acceptable syreadditionssalte deraf samt forbindelser til anvendelse som udgangsmaterialer ved fremgangsmaaden |
Also Published As
| Publication number | Publication date |
|---|---|
| CA957376A (en) | 1974-11-05 |
| FR2115451B1 (da) | 1975-02-07 |
| BE775593A (fr) | 1972-03-16 |
| IL38079A0 (en) | 1972-01-27 |
| NO135248B (da) | 1976-11-29 |
| GB1314955A (en) | 1973-04-26 |
| JPS5623985B2 (da) | 1981-06-03 |
| DE2158136A1 (de) | 1972-05-31 |
| FR2115451A1 (da) | 1972-07-07 |
| NL175411C (nl) | 1984-11-01 |
| NL175411B (nl) | 1984-06-01 |
| IL38079A (en) | 1974-10-22 |
| IE35778L (en) | 1972-05-27 |
| CH562215A5 (da) | 1975-05-30 |
| SE369900B (da) | 1974-09-23 |
| DE2158136C2 (de) | 1982-11-18 |
| DK135895C (da) | 1977-12-12 |
| NO135248C (da) | 1977-03-09 |
| ES397370A1 (es) | 1974-05-16 |
| ZA717147B (en) | 1972-07-26 |
| NL7116194A (da) | 1972-05-30 |
| PH9306A (en) | 1975-08-18 |
| IE35778B1 (en) | 1976-05-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PUP | Patent expired |