DK134160B - Fremgangsmåde til fremstilling af homopyrimidazolderivater eller syreadditionssalte eller kvaternære ammoniumsalte deraf. - Google Patents

Fremgangsmåde til fremstilling af homopyrimidazolderivater eller syreadditionssalte eller kvaternære ammoniumsalte deraf.

Info

Publication number
DK134160B
DK134160B DK545067AA DK545067A DK134160B DK 134160 B DK134160 B DK 134160B DK 545067A A DK545067A A DK 545067AA DK 545067 A DK545067 A DK 545067A DK 134160 B DK134160 B DK 134160B
Authority
DK
Denmark
Prior art keywords
preparation
quaternary ammonium
acid addition
salts
addition salts
Prior art date
Application number
DK545067AA
Other languages
English (en)
Other versions
DK134160C (da
Inventor
Zoltan Meszaros
Jozsef Knoll
Peter Szentmiklosi
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Priority to DK138273A priority Critical patent/DK138949B/da
Priority to DK228474A priority patent/DK136723B/da
Publication of DK134160B publication Critical patent/DK134160B/da
Application granted granted Critical
Publication of DK134160C publication Critical patent/DK134160C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK545067AA 1966-11-02 1967-11-01 Fremgangsmåde til fremstilling af homopyrimidazolderivater eller syreadditionssalte eller kvaternære ammoniumsalte deraf. DK134160B (da)

Priority Applications (2)

Application Number Priority Date Filing Date Title
DK138273A DK138949B (da) 1966-11-02 1973-03-14 Analogifremgangsmåde til fremstilling af homopyrimidazolderivater eller salte deraf.
DK228474A DK136723B (da) 1966-11-02 1974-04-25 Analogifremgangsmåde til fremstilling af homopyrimidazol-derivater eller salte deraf.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HUCI000670 1966-11-02

Publications (2)

Publication Number Publication Date
DK134160B true DK134160B (da) 1976-09-20
DK134160C DK134160C (da) 1977-02-21

Family

ID=10994330

Family Applications (1)

Application Number Title Priority Date Filing Date
DK545067AA DK134160B (da) 1966-11-02 1967-11-01 Fremgangsmåde til fremstilling af homopyrimidazolderivater eller syreadditionssalte eller kvaternære ammoniumsalte deraf.

Country Status (15)

Country Link
US (2) US3585198A (da)
JP (1) JPS4939278B1 (da)
AT (5) AT294107B (da)
BE (1) BE705934A (da)
CH (1) CH538494A (da)
CS (1) CS165991B2 (da)
DE (2) DE1670480C2 (da)
DK (1) DK134160B (da)
FR (1) FR7813M (da)
GB (1) GB1209946A (da)
HK (1) HK27876A (da)
IL (1) IL28863A (da)
NL (1) NL6714810A (da)
SE (3) SE336134B (da)
YU (2) YU35136B (da)

Families Citing this family (42)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3907798A (en) * 1966-06-15 1975-09-23 Sterling Drug Inc Preparation of 4H-pyrido{8 1,2-a{9 pyrimidin-4-ones from cyclic alkylidene 2-pyridylaminomethylenemalonates
BE788601A (fr) * 1971-09-10 1973-03-08 Takeda Chemical Industries Ltd Procede de preparation de derives de pyrimidine
CA1005056A (en) * 1971-09-17 1977-02-08 E.R. Squibb And Sons Manufacture of substituted pyridopyrimidinones
HU169230B (da) * 1972-03-29 1976-10-28
US3960847A (en) * 1972-04-17 1976-06-01 E. R. Squibb & Sons, Inc. 9-Substituted-4-oxopyrido(1,2-α)pyrimidine-3-carboxylic acids and derivatives thereof
US4013656A (en) * 1972-06-07 1977-03-22 Dynamit Nobel Aktiengesellschaft Process for the preparation of pyridylamino-methylenemalonic acid derivatives
HU166378B (da) 1972-12-19 1975-03-28
SE422272B (sv) * 1972-08-03 1982-03-01 Chinoin Gyogyszer Es Vegyeszet Sett att framstella ett for oral administration lempligt farmaceutiskt preparat med synergistisk, analgetisk aktivitet, innehallande bl a azidokodein
US4027024A (en) 1972-12-19 1977-05-31 Chinoin Gyogyszer-Es Vegyeszeti Termekek Gyara Rt Pharmaceutical composition having synergistic analgesic activity
US4209622A (en) * 1973-03-30 1980-06-24 Chinoin Gygyszer es Vegyeszeti Termekek Gyara Rt. 3-(Ethoxycarbonyl-methyl)-6-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine
HU168014B (da) * 1973-03-30 1976-02-28
HU169223B (da) * 1973-12-29 1976-10-28
US4022897A (en) * 1974-03-04 1977-05-10 E. R. Squibb & Sons, Inc. CNS active compounds
US3929787A (en) * 1974-04-22 1975-12-30 Squibb & Sons Inc 6,7,8,9-Tetrahydro-pyrido(1,2-a)pyrimidin-4-ones
US3935197A (en) * 1975-05-16 1976-01-27 E. R. Squibb & Sons, Inc. 2-Styryl-4H-pyrido(1,2-a)pyrimidin-4-ones
HU173823B (hu) * 1975-07-25 1979-08-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija stabil'nogo lechebnogo preparata dlja oral'noj dozirovki, kotoryj soderzhit proizvodnyj gomopirimidazola
JPS5822040B2 (ja) * 1975-10-13 1983-05-06 わかもと製薬 （株） ホモピリイミダゾ−ル誘導体の製造法
HU173438B (hu) * 1975-11-27 1979-05-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija novykh proizvodnykh 4-okso-1,6,7,8-/tetragidro-4h-pirido/1,2/pirimidina s zaderzhivajuhhejj vozgoranie aktivnot'ju i protivosvertivajuhhem effektom
US4495189A (en) * 1975-11-27 1985-01-22 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara R.T. Condensed pyrimidines
HU174693B (hu) * 1976-02-12 1980-03-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija kondensirovannykh proizvodnykh pirimidina
HU174901B (hu) * 1976-06-25 1980-04-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija novykh proizvodnykh pirido/1,2-a/pirimidina
FR2358891A1 (fr) * 1976-07-22 1978-02-17 Yamanouchi Pharma Co Ltd Composes heterocycliques contenant un azote, utilise comme agents analgesiques et anti-inflammatoires
US4122274A (en) * 1977-05-25 1978-10-24 Bristol-Myers Company 3-Tetrazolo-5,6,7,8-substituted-pyrido[1,2-a]pyrimidin-4-ones
HU178910B (en) * 1977-08-19 1982-07-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 2,3-disubstituted-4-oxo-4h-pyrido/1,2-a/-pyrimidines
HU180439B (en) * 1977-12-29 1983-03-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-amino-pyrido-square bracket-1,2-a-square bracket closed-pyrimidine derivatives
HU178496B (en) * 1977-12-29 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyrimidine derivatives with antiallergic activity
US4192944A (en) * 1978-04-03 1980-03-11 Bristol-Myers Company Optionally substituted 4-oxo-4H-pyrido[1,2-a]pyrimidine-3-N-(1H-tetrazol-4-yl)carboxamides and their use as antiallergy agents
FR2449689A1 (fr) * 1979-02-20 1980-09-19 Logeais Labor Jacques Nouveaux derives condenses de pyrrolidine ou de piperidine, leur procede de preparation et leurs applications en therapeutique
HU176942B (hu) * 1979-05-11 1981-06-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija 2,3- i 3,4-dvuzamehhjonnykh tetragidro-pirrolo!1,2-a!-pirimidinov
HU179443B (en) * 1979-05-11 1982-10-28 Chinoin Gyogyszer Es Vegyeszet Process for producing substituted geminal dihalogeno-derivatives of pyrido-square bracket-1,2-a-square closed-pyrimidines,pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines and pyrimido-square bracket-1,2,-a-square bracket closed-asepines
HU178452B (en) * 1979-05-11 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 9-substituted amino-4-oxo-6,7-dihydro-4h-pyrido/1,2-a/pyrimidine derivatives
US4482557A (en) * 1979-05-11 1984-11-13 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. 3-Substituted-2-oxo-tetrahydro-pyrrol[1,2-a]pyrimidines having digitalis-like activity
HU177184B (en) * 1979-05-11 1981-08-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 2,3- and 3,4-disubstituted-hexahydro-pyrimido-square bracket-1,2-a-square bracket closed-asepines
HU186607B (en) * 1982-03-31 1985-08-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing pharmaceutical composition with synergetic antiinflammatory activity
US4474953A (en) * 1982-09-09 1984-10-02 Riker Laboratories, Inc. Process and intermediates for the preparation of 3(1H-tetrazol-5-yl)-4H-pyrido[1,2-a]pyrimidin-4-ones
US4507477A (en) * 1982-09-09 1985-03-26 Riker Laboratories, Inc. Process for tetrazolyl-pyrimidinone derivatives
US4476130A (en) * 1982-09-09 1984-10-09 Riker Laboratories, Inc. 3-(1H-Tetrazol-5-yl)-4H-pyrimido[2,1-b]benzoxazol-4-one compounds exhibiting anti-allergic activity
US4457932A (en) * 1983-07-22 1984-07-03 Bristol-Myers Company Anti-ulcer agents
CA1283411C (en) * 1985-09-25 1991-04-23 Masami Doteuchi 9-(substituted thio)-4h-pyrido[1,2-a]-pyrimidin-4-one derivatives
HU201551B (en) * 1988-02-03 1990-11-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 4-oxo-4h-pyrido(1,2-a)pyrimidine-3-carboxylic acid amide derivatives and pharmaceutical compositions comprising same
CA2205313C (en) 1996-05-28 2005-01-18 Tecton Products Method of manufacture of a plastic component which is insensitive to the elements, and a plastic component so manufactured
BR112012005200A2 (pt) * 2009-09-09 2021-02-02 E.I. Du Pont De Nemours And Company compostos, mistura herbicida, composições herbicidas e método para controlar o crescimento de vegetação indesejada

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3149112A (en) * 1964-09-15 Z-diethylaminoethoxy

Also Published As

Publication number Publication date
US3585198A (en) 1971-06-15
DE1670480C2 (de) 1983-06-01
FR7813M (da) 1970-05-20
HK27876A (en) 1976-05-21
DE1795769A1 (de) 1975-04-10
DK134160C (da) 1977-02-21
YU35142B (en) 1980-09-25
JPS4939278B1 (da) 1974-10-24
YU35136B (en) 1980-09-25
CH538494A (de) 1973-06-30
AT302311B (de) 1972-09-15
YU250373A (en) 1980-03-15
NL6714810A (da) 1968-05-03
US3696197A (en) 1972-10-03
AT296996B (de) 1972-03-10
CS165991B2 (da) 1975-12-22
DE1795769B2 (de) 1978-03-09
AT286990B (de) 1971-01-11
YU209567A (en) 1980-03-15
SE336134B (da) 1971-06-28
DE1795769C3 (de) 1978-11-02
AT294107B (de) 1971-11-10
AT299212B (de) 1972-06-12
GB1209946A (en) 1970-10-21
SE363333B (da) 1974-01-14
SE409327B (sv) 1979-08-13
BE705934A (da) 1968-03-01
IL28863A (en) 1973-07-30
DE1670480A1 (de) 1972-05-10

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