DK131036B - Analogifremgangsmåde til fremstilling af 3,16alfa,17xi-trihydroxy-11beta-alkoxyestra-1,3,5(10)-triener. - Google Patents

Analogifremgangsmåde til fremstilling af 3,16alfa,17xi-trihydroxy-11beta-alkoxyestra-1,3,5(10)-triener.

Info

Publication number
DK131036B
DK131036B DK447272AA DK447272A DK131036B DK 131036 B DK131036 B DK 131036B DK 447272A A DK447272A A DK 447272AA DK 447272 A DK447272 A DK 447272A DK 131036 B DK131036 B DK 131036B
Authority
DK
Denmark
Prior art keywords
alkoxyestra
16alpha
11beta
trienes
trihydroxy
Prior art date
Application number
DK447272AA
Other languages
Danish (da)
English (en)
Other versions
DK131036C (en:Method
Inventor
J-C Gasc
A Pierdet
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of DK131036B publication Critical patent/DK131036B/da
Application granted granted Critical
Publication of DK131036C publication Critical patent/DK131036C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0092—Alkenyl derivatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0096—Alkynyl derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008—Expansion of ring D by one atom, e.g. D homo steroids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK447272AA 1971-09-10 1972-09-11 Analogifremgangsmåde til fremstilling af 3,16alfa,17xi-trihydroxy-11beta-alkoxyestra-1,3,5(10)-triener. DK131036B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7132703A FR2152392B1 (en:Method) 1971-09-10 1971-09-10

Publications (2)

Publication Number Publication Date
DK131036B true DK131036B (da) 1975-05-20
DK131036C DK131036C (en:Method) 1975-10-20

Family

ID=9082761

Family Applications (1)

Application Number Title Priority Date Filing Date
DK447272AA DK131036B (da) 1971-09-10 1972-09-11 Analogifremgangsmåde til fremstilling af 3,16alfa,17xi-trihydroxy-11beta-alkoxyestra-1,3,5(10)-triener.

Country Status (14)

Country Link
US (1) US3776902A (en:Method)
JP (2) JPS5124511B2 (en:Method)
AU (1) AU462880B2 (en:Method)
BE (1) BE788500A (en:Method)
CA (1) CA974227A (en:Method)
CH (1) CH556832A (en:Method)
DK (1) DK131036B (en:Method)
ES (1) ES406543A1 (en:Method)
FR (1) FR2152392B1 (en:Method)
GB (2) GB1407477A (en:Method)
IL (1) IL40251A (en:Method)
NL (1) NL7212228A (en:Method)
SE (1) SE385903B (en:Method)
ZA (1) ZA726138B (en:Method)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS51107960A (ja) * 1975-03-10 1976-09-24 Hiraoka Kogyo Kk Chojuruikuchikuhatsuonsochi
JPS5854940Y2 (ja) * 1977-04-01 1983-12-15 ニッタン株式会社 鼠追放装置
JPS5442680U (en:Method) * 1977-08-31 1979-03-23
FI83087C (fi) * 1984-05-16 1991-05-27 Schering Ag Foerfarande foer framstaellning av terapeutiskt anvaendbara estriol-3,17-diestrar.
DE10151365A1 (de) * 2001-10-17 2003-04-30 Schering Ag 17-Chlor-D-Homosteroide als selektive Estrogenrezeptorantagonisten
JP4925164B2 (ja) * 2006-01-31 2012-04-25 株式会社吉野工業所 蓋付き高気密容器

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5634321B2 (en:Method) * 1973-11-16 1981-08-10

Also Published As

Publication number Publication date
NL7212228A (en:Method) 1973-03-13
DE2244522B2 (de) 1976-02-12
IL40251A0 (en) 1972-10-29
AU462880B2 (en) 1975-07-10
ES406543A1 (es) 1975-09-16
JPS5124511B2 (en:Method) 1976-07-24
CH556832A (de) 1974-12-13
JPS5619880B2 (en:Method) 1981-05-09
GB1407478A (en) 1975-09-24
AU4646972A (en) 1974-03-14
CA974227A (en) 1975-09-09
DK131036C (en:Method) 1975-10-20
US3776902A (en) 1973-12-04
BE788500A (fr) 1973-03-07
IL40251A (en) 1976-11-30
FR2152392A1 (en:Method) 1973-04-27
ZA726138B (en) 1973-10-31
DE2244522A1 (de) 1973-03-22
SE385903B (sv) 1976-07-26
JPS4834868A (en:Method) 1973-05-22
JPS51101969A (en:Method) 1976-09-08
GB1407477A (en) 1975-09-24
FR2152392B1 (en:Method) 1974-10-18

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Legal Events

Date Code Title Description
PBP Patent lapsed