DK131036B - Analogifremgangsmåde til fremstilling af 3,16alfa,17xi-trihydroxy-11beta-alkoxyestra-1,3,5(10)-triener. - Google Patents

Analogifremgangsmåde til fremstilling af 3,16alfa,17xi-trihydroxy-11beta-alkoxyestra-1,3,5(10)-triener.

Info

Publication number
DK131036B
DK131036B DK447272AA DK447272A DK131036B DK 131036 B DK131036 B DK 131036B DK 447272A A DK447272A A DK 447272AA DK 447272 A DK447272 A DK 447272A DK 131036 B DK131036 B DK 131036B
Authority
DK
Denmark
Prior art keywords
alkoxyestra
16alpha
11beta
trienes
trihydroxy
Prior art date
Application number
DK447272AA
Other languages
English (en)
Other versions
DK131036C (da
Inventor
J-C Gasc
A Pierdet
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of DK131036B publication Critical patent/DK131036B/da
Application granted granted Critical
Publication of DK131036C publication Critical patent/DK131036C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0081Substituted in position 17 alfa and 17 beta
    • C07J1/0088Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0092Alkenyl derivatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0081Substituted in position 17 alfa and 17 beta
    • C07J1/0088Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0096Alkynyl derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J63/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008Expansion of ring D by one atom, e.g. D homo steroids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J9/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK447272AA 1971-09-10 1972-09-11 Analogifremgangsmåde til fremstilling af 3,16alfa,17xi-trihydroxy-11beta-alkoxyestra-1,3,5(10)-triener. DK131036B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7132703A FR2152392B1 (da) 1971-09-10 1971-09-10

Publications (2)

Publication Number Publication Date
DK131036B true DK131036B (da) 1975-05-20
DK131036C DK131036C (da) 1975-10-20

Family

ID=9082761

Family Applications (1)

Application Number Title Priority Date Filing Date
DK447272AA DK131036B (da) 1971-09-10 1972-09-11 Analogifremgangsmåde til fremstilling af 3,16alfa,17xi-trihydroxy-11beta-alkoxyestra-1,3,5(10)-triener.

Country Status (14)

Country Link
US (1) US3776902A (da)
JP (2) JPS5124511B2 (da)
AU (1) AU462880B2 (da)
BE (1) BE788500A (da)
CA (1) CA974227A (da)
CH (1) CH556832A (da)
DK (1) DK131036B (da)
ES (1) ES406543A1 (da)
FR (1) FR2152392B1 (da)
GB (2) GB1407477A (da)
IL (1) IL40251A (da)
NL (1) NL7212228A (da)
SE (1) SE385903B (da)
ZA (1) ZA726138B (da)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS51107960A (ja) * 1975-03-10 1976-09-24 Hiraoka Kogyo Kk Chojuruikuchikuhatsuonsochi
JPS5854940Y2 (ja) * 1977-04-01 1983-12-15 ニッタン株式会社 鼠追放装置
JPS5442680U (da) * 1977-08-31 1979-03-23
FI83087C (fi) * 1984-05-16 1991-05-27 Schering Ag Foerfarande foer framstaellning av terapeutiskt anvaendbara estriol-3,17-diestrar.
DE10151365A1 (de) * 2001-10-17 2003-04-30 Schering Ag 17-Chlor-D-Homosteroide als selektive Estrogenrezeptorantagonisten
JP4925164B2 (ja) * 2006-01-31 2012-04-25 株式会社吉野工業所 蓋付き高気密容器

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5634321B2 (da) * 1973-11-16 1981-08-10

Also Published As

Publication number Publication date
IL40251A (en) 1976-11-30
US3776902A (en) 1973-12-04
GB1407477A (en) 1975-09-24
FR2152392A1 (da) 1973-04-27
JPS4834868A (da) 1973-05-22
ZA726138B (en) 1973-10-31
IL40251A0 (en) 1972-10-29
ES406543A1 (es) 1975-09-16
DK131036C (da) 1975-10-20
GB1407478A (en) 1975-09-24
AU462880B2 (en) 1975-07-10
DE2244522A1 (de) 1973-03-22
BE788500A (fr) 1973-03-07
NL7212228A (da) 1973-03-13
JPS51101969A (da) 1976-09-08
JPS5619880B2 (da) 1981-05-09
DE2244522B2 (de) 1976-02-12
SE385903B (sv) 1976-07-26
CA974227A (en) 1975-09-09
CH556832A (de) 1974-12-13
FR2152392B1 (da) 1974-10-18
AU4646972A (en) 1974-03-14
JPS5124511B2 (da) 1976-07-24

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Legal Events

Date Code Title Description
PBP Patent lapsed