DK120234B - Fremgangsmåde til fremstilling af 17α-monocarboxylsyreestere af 11β, 17α, 21-trihydroxysteroider af pregnanrækken. - Google Patents

Fremgangsmåde til fremstilling af 17α-monocarboxylsyreestere af 11β, 17α, 21-trihydroxysteroider af pregnanrækken.

Info

Publication number
DK120234B
DK120234B DK36169AA DK36169A DK120234B DK 120234 B DK120234 B DK 120234B DK 36169A A DK36169A A DK 36169AA DK 36169 A DK36169 A DK 36169A DK 120234 B DK120234 B DK 120234B
Authority
DK
Denmark
Prior art keywords
trihydroxysteroids
preparation
acid esters
monocarboxylic acid
pregnane series
Prior art date
Application number
DK36169AA
Other languages
Danish (da)
English (en)
Inventor
J Lens
A Marx
Original Assignee
Koninklijke Gist Spiritus
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Koninklijke Gist Spiritus filed Critical Koninklijke Gist Spiritus
Publication of DK120234B publication Critical patent/DK120234B/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • FMECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
    • F21LIGHTING
    • F21VFUNCTIONAL FEATURES OR DETAILS OF LIGHTING DEVICES OR SYSTEMS THEREOF; STRUCTURAL COMBINATIONS OF LIGHTING DEVICES WITH OTHER ARTICLES, NOT OTHERWISE PROVIDED FOR
    • F21V17/00Fastening of component parts of lighting devices, e.g. shades, globes, refractors, reflectors, filters, screens, grids or protective cages
    • F21V17/10Fastening of component parts of lighting devices, e.g. shades, globes, refractors, reflectors, filters, screens, grids or protective cages characterised by specific fastening means or way of fastening
    • F21V17/20Fastening of component parts of lighting devices, e.g. shades, globes, refractors, reflectors, filters, screens, grids or protective cages characterised by specific fastening means or way of fastening by toggle-action levers

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Engineering & Computer Science (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK36169AA 1968-01-23 1969-01-22 Fremgangsmåde til fremstilling af 17α-monocarboxylsyreestere af 11β, 17α, 21-trihydroxysteroider af pregnanrækken. DK120234B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB358768 1968-01-23

Publications (1)

Publication Number Publication Date
DK120234B true DK120234B (da) 1971-05-03

Family

ID=9761163

Family Applications (1)

Application Number Title Priority Date Filing Date
DK36169AA DK120234B (da) 1968-01-23 1969-01-22 Fremgangsmåde til fremstilling af 17α-monocarboxylsyreestere af 11β, 17α, 21-trihydroxysteroider af pregnanrækken.

Country Status (12)

Country Link
US (1) US3557162A (US06534493-20030318-C00166.png)
AT (1) AT292929B (US06534493-20030318-C00166.png)
BE (1) BE726981A (US06534493-20030318-C00166.png)
CH (1) CH511822A (US06534493-20030318-C00166.png)
DE (1) DE1903118A1 (US06534493-20030318-C00166.png)
DK (1) DK120234B (US06534493-20030318-C00166.png)
ES (1) ES362475A1 (US06534493-20030318-C00166.png)
FR (2) FR8225M (US06534493-20030318-C00166.png)
GB (1) GB1227992A (US06534493-20030318-C00166.png)
IT (1) IT1036015B (US06534493-20030318-C00166.png)
NL (1) NL162083C (US06534493-20030318-C00166.png)
SE (1) SE339828B (US06534493-20030318-C00166.png)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1033042B (it) * 1970-03-14 1979-07-10 Luso Farmaco Inst Desametazone 17 valerato e processi per la sua preparazione
SE418294B (sv) * 1974-03-27 1981-05-18 Plurichemie Anstalt Sett att framstella en 16alfa- eller 16beta-9alfa-klor eller -fluorsteroidester
US4036831A (en) * 1975-10-28 1977-07-19 Steroid Development Company Establishment Trimethyl siloxane steroid intermediates
DE3442527A1 (de) * 1983-11-23 1985-05-30 Bösha GmbH & Co KG, 4780 Lippstadt Langfeldleuchte fuer den einsatz in schlagwetter- und explosionsgeschuetzten bereichen
US6759398B2 (en) * 2000-08-05 2004-07-06 Smithkline Beecham Corporation Anti-inflammatory androstane derivative
US6777399B2 (en) * 2000-08-05 2004-08-17 Smithkline Beecham Corporation Anti-inflammatory androstane derivative compositions
BRPI0113042B8 (pt) * 2000-08-05 2021-05-25 Glaxo Group Ltd composto da fórmula ou um seu solvato fisiologicamente aceitável, uso do mesmo, composição farmacêutica, formulação farmacêutica, método para o tratamento de um indivíduo humano ou animal com uma condição inflamatória e/ou alérgica, e, processo para preparar um composto ou um seu solvato
GB0019172D0 (en) * 2000-08-05 2000-09-27 Glaxo Group Ltd Novel compounds
US6858596B2 (en) * 2000-08-05 2005-02-22 Smithkline Beecham Corporation Formulation containing anti-inflammatory androstane derivative
CZ20032958A3 (en) * 2001-04-30 2004-03-17 Glaxo Group Limited Anti-inflammatory 17.beta.-carbothioate ester derivatives of androstane with a cyclic ester group in position 17.alpha
JP2005500290A (ja) * 2001-06-12 2005-01-06 グラクソ グループ リミテッド 抗炎症性の、17β−カルボチオアートアンドロスタン誘導体である17α複素環エステル
US20050175545A1 (en) * 2002-02-04 2005-08-11 Keith Biggadike Formulation for inhalation comprising a glucocorticoid and a beta 2-adrenoreceptor agonist
GB0202635D0 (en) * 2002-02-05 2002-03-20 Glaxo Wellcome Mfg Pte Ltd Formulation containing novel anti-inflammatory androstane derivative
GB2389530B (en) 2002-06-14 2007-01-10 Cipla Ltd Pharmaceutical compositions
GB0507165D0 (en) * 2005-04-08 2005-05-18 Glaxo Group Ltd Novel crystalline pharmaceutical product
GB0615108D0 (en) * 2006-07-28 2006-09-06 Glaxo Group Ltd Novel formulations
NO331891B1 (no) * 2007-03-20 2012-04-30 Clavis Pharma Asa Kjemiske forbindelser, et farmasoytisk preparat inneholdende slike forbindelser, samt anvendelse derav for behandling av kreft, inflammasjon og KOLS
UA116622C2 (uk) * 2011-11-11 2018-04-25 Аллерган, Інк. Похідні 4-прегенен-11ss-17-21-тріол-3,20-діону для лікування хвороб очей

Also Published As

Publication number Publication date
CH511822A (de) 1971-08-31
GB1227992A (US06534493-20030318-C00166.png) 1971-04-15
NL162083B (nl) 1979-11-15
ES362475A1 (es) 1970-12-01
NL6901024A (US06534493-20030318-C00166.png) 1969-07-25
IT1036015B (it) 1979-10-30
BE726981A (US06534493-20030318-C00166.png) 1969-07-16
DE1903118A1 (de) 1969-08-07
NL162083C (nl) 1980-04-15
AT292929B (de) 1971-09-10
FR2000571A1 (US06534493-20030318-C00166.png) 1969-09-12
SE339828B (US06534493-20030318-C00166.png) 1971-10-25
US3557162A (en) 1971-01-19
FR8225M (US06534493-20030318-C00166.png) 1970-09-28

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