DK114836B - Fremgangsmåde til fremstilling af 3-hydroxy-1,3-dihydro-2H-1,4-benzodiazepin-2-oner eller estere deraf. - Google Patents

Fremgangsmåde til fremstilling af 3-hydroxy-1,3-dihydro-2H-1,4-benzodiazepin-2-oner eller estere deraf.

Info

Publication number
DK114836B
DK114836B DK594863AA DK594863A DK114836B DK 114836 B DK114836 B DK 114836B DK 594863A A DK594863A A DK 594863AA DK 594863 A DK594863 A DK 594863A DK 114836 B DK114836 B DK 114836B
Authority
DK
Denmark
Prior art keywords
benzodiazepin
dihydro
hydroxy
esters
ones
Prior art date
Application number
DK594863AA
Other languages
Danish (da)
English (en)
Inventor
S Bell
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Home Prod filed Critical American Home Prod
Publication of DK114836B publication Critical patent/DK114836B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK594863AA 1962-12-20 1963-12-19 Fremgangsmåde til fremstilling af 3-hydroxy-1,3-dihydro-2H-1,4-benzodiazepin-2-oner eller estere deraf. DK114836B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US247460A US3197467A (en) 1962-12-20 1962-12-20 Process for preparing 1, 3-dihydro-3-hydroxy-2h-1, 4-benzodiazepin-2-ones

Publications (1)

Publication Number Publication Date
DK114836B true DK114836B (da) 1969-08-11

Family

ID=22935024

Family Applications (1)

Application Number Title Priority Date Filing Date
DK594863AA DK114836B (da) 1962-12-20 1963-12-19 Fremgangsmåde til fremstilling af 3-hydroxy-1,3-dihydro-2H-1,4-benzodiazepin-2-oner eller estere deraf.

Country Status (12)

Country Link
US (1) US3197467A (sv)
BE (1) BE641547A (sv)
BR (1) BR6355463D0 (sv)
CH (1) CH438337A (sv)
DE (1) DE1445420A1 (sv)
DK (1) DK114836B (sv)
ES (1) ES294651A1 (sv)
FI (1) FI46385C (sv)
GB (1) GB1035174A (sv)
IT (1) IT1193740B (sv)
NL (1) NL301733A (sv)
SE (2) SE314680B (sv)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3531473A (en) * 1966-12-06 1970-09-29 Hoffmann La Roche Preparation of 3-hydroxy-1,4-benzodiazepines
US3903103A (en) * 1971-09-15 1975-09-02 Upjohn Co 4-Amino-s-triazolo-{8 4,3-a{9 {8 1,4{9 benzodiazepine
ES405260A1 (es) * 1972-07-28 1975-07-01 Stabilimenti Chim Farmac Riuni Procedimiento para la preparacion de 3-hidroxi-5-aril-7- sustituidos-1, 3-dihidro-2h-1, 4-benzodiacepin-2-onas.

Also Published As

Publication number Publication date
DE1445420A1 (de) 1969-05-22
CH438337A (de) 1967-06-30
NL301733A (sv)
SE314680B (sv) 1969-09-15
FI46385C (sv) 1973-03-12
GB1035174A (en) 1966-07-06
BE641547A (sv) 1964-06-19
US3197467A (en) 1965-07-27
IT1193740B (it) 1988-08-24
FI46385B (sv) 1972-11-30
SE343061B (sv) 1972-02-28
BR6355463D0 (pt) 1973-07-17
ES294651A1 (es) 1964-06-01

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