DK1140029T3 - Fremstilling af mikropartikler med en valgt release-profil - Google Patents
Fremstilling af mikropartikler med en valgt release-profilInfo
- Publication number
- DK1140029T3 DK1140029T3 DK99965212T DK99965212T DK1140029T3 DK 1140029 T3 DK1140029 T3 DK 1140029T3 DK 99965212 T DK99965212 T DK 99965212T DK 99965212 T DK99965212 T DK 99965212T DK 1140029 T3 DK1140029 T3 DK 1140029T3
- Authority
- DK
- Denmark
- Prior art keywords
- microparticles
- release profile
- preparation
- release
- active agent
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
- A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1682—Processes
- A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J13/00—Colloid chemistry, e.g. the production of colloidal materials or their solutions, not otherwise provided for; Making microcapsules or microballoons
- B01J13/02—Making microcapsules or microballoons
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10T—TECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
- Y10T428/00—Stock material or miscellaneous articles
- Y10T428/29—Coated or structually defined flake, particle, cell, strand, strand portion, rod, filament, macroscopic fiber or mass thereof
- Y10T428/2982—Particulate matter [e.g., sphere, flake, etc.]
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Chemistry (AREA)
- Dispersion Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Preparation (AREA)
- Manufacturing Of Micro-Capsules (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US09/223,276 US6194006B1 (en) | 1998-12-30 | 1998-12-30 | Preparation of microparticles having a selected release profile |
Publications (1)
Publication Number | Publication Date |
---|---|
DK1140029T3 true DK1140029T3 (da) | 2006-02-13 |
Family
ID=22835812
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK99965212T DK1140029T3 (da) | 1998-12-30 | 1999-12-10 | Fremstilling af mikropartikler med en valgt release-profil |
Country Status (10)
Country | Link |
---|---|
US (4) | US6194006B1 (ja) |
EP (1) | EP1140029B1 (ja) |
JP (1) | JP4694694B2 (ja) |
AT (1) | ATE308977T1 (ja) |
AU (1) | AU759214B2 (ja) |
CA (1) | CA2352818C (ja) |
DE (1) | DE69928283T2 (ja) |
DK (1) | DK1140029T3 (ja) |
ES (1) | ES2251850T3 (ja) |
WO (1) | WO2000040221A1 (ja) |
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NZ276088A (en) | 1993-11-19 | 1999-07-29 | Janssen Pharmaceutica Nv | [(1,2-benzisoxazol-3-yl)-1-piperidinyl-alkyl-6,7,8,9-tetrahydro-4h- pyrido[1,2-a]-pyrimidin-4-one derivatives (ie risperidone) |
EP1649850A1 (en) * | 1993-11-19 | 2006-04-26 | Alkermes Controlled Therapeutics Inc. II | Preparation of biodegradable microparticles containing a biologically active agent |
US5904935A (en) | 1995-06-07 | 1999-05-18 | Alza Corporation | Peptide/protein suspending formulations |
US5851538A (en) * | 1995-12-29 | 1998-12-22 | Advanced Polymer Systems, Inc. | Retinoid formulations in porous microspheres for reduced irritation and enhanced stability |
US5792477A (en) * | 1996-05-07 | 1998-08-11 | Alkermes Controlled Therapeutics, Inc. Ii | Preparation of extended shelf-life biodegradable, biocompatible microparticles containing a biologically active agent |
US5945126A (en) | 1997-02-13 | 1999-08-31 | Oakwood Laboratories L.L.C. | Continuous microsphere process |
GB9718986D0 (en) | 1997-09-09 | 1997-11-12 | Danbiosyst Uk | Controlled release microsphere delivery system |
US6194006B1 (en) * | 1998-12-30 | 2001-02-27 | Alkermes Controlled Therapeutics Inc. Ii | Preparation of microparticles having a selected release profile |
US6306425B1 (en) * | 1999-04-09 | 2001-10-23 | Southern Research Institute | Injectable naltrexone microsphere compositions and their use in reducing consumption of heroin and alcohol |
US6264987B1 (en) * | 2000-05-19 | 2001-07-24 | Alkermes Controlled Therapeutics Inc. Ii | Method for preparing microparticles having a selected polymer molecular weight |
-
1998
- 1998-12-30 US US09/223,276 patent/US6194006B1/en not_active Expired - Lifetime
-
1999
- 1999-12-10 EP EP99965212A patent/EP1140029B1/en not_active Expired - Lifetime
- 1999-12-10 ES ES99965212T patent/ES2251850T3/es not_active Expired - Lifetime
- 1999-12-10 DE DE69928283T patent/DE69928283T2/de not_active Expired - Lifetime
- 1999-12-10 CA CA002352818A patent/CA2352818C/en not_active Expired - Lifetime
- 1999-12-10 AU AU31178/00A patent/AU759214B2/en not_active Expired
- 1999-12-10 DK DK99965212T patent/DK1140029T3/da active
- 1999-12-10 WO PCT/US1999/029349 patent/WO2000040221A1/en active IP Right Grant
- 1999-12-10 JP JP2000591978A patent/JP4694694B2/ja not_active Expired - Lifetime
- 1999-12-10 AT AT99965212T patent/ATE308977T1/de active
-
2000
- 2000-11-28 US US09/722,335 patent/US6379703B1/en not_active Expired - Lifetime
-
2002
- 2002-01-31 US US10/059,115 patent/US6596316B2/en not_active Expired - Lifetime
-
2003
- 2003-05-12 US US10/435,586 patent/US20030203039A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
US6194006B1 (en) | 2001-02-27 |
US20030003156A1 (en) | 2003-01-02 |
US6379703B1 (en) | 2002-04-30 |
JP2002534372A (ja) | 2002-10-15 |
EP1140029A1 (en) | 2001-10-10 |
AU3117800A (en) | 2000-07-24 |
CA2352818A1 (en) | 2000-07-13 |
DE69928283T2 (de) | 2006-08-10 |
DE69928283D1 (de) | 2005-12-15 |
CA2352818C (en) | 2009-04-14 |
ES2251850T3 (es) | 2006-05-01 |
EP1140029B1 (en) | 2005-11-09 |
US20030203039A1 (en) | 2003-10-30 |
JP4694694B2 (ja) | 2011-06-08 |
WO2000040221A1 (en) | 2000-07-13 |
US6596316B2 (en) | 2003-07-22 |
AU759214B2 (en) | 2003-04-10 |
ATE308977T1 (de) | 2005-11-15 |
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