DK0949250T3 - Fremgangsmåde til fremstilling af alpha1L-adrenoceptorantagonister - Google Patents
Fremgangsmåde til fremstilling af alpha1L-adrenoceptorantagonisterInfo
- Publication number
- DK0949250T3 DK0949250T3 DK99105755T DK99105755T DK0949250T3 DK 0949250 T3 DK0949250 T3 DK 0949250T3 DK 99105755 T DK99105755 T DK 99105755T DK 99105755 T DK99105755 T DK 99105755T DK 0949250 T3 DK0949250 T3 DK 0949250T3
- Authority
- DK
- Denmark
- Prior art keywords
- alpha1l
- preparation
- adrenoceptor antagonists
- fluoro
- chem
- Prior art date
Links
- 108060003345 Adrenergic Receptor Proteins 0.000 title 1
- 102000017910 Adrenergic receptor Human genes 0.000 title 1
- 239000005557 antagonist Substances 0.000 title 1
- 125000001153 fluoro group Chemical group F* 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
- C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
- C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
- C07D239/545—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/553—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms with halogen atoms or nitro radicals directly attached to ring carbon atoms, e.g. fluorouracil
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US7997498P | 1998-03-30 | 1998-03-30 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0949250T3 true DK0949250T3 (da) | 2006-08-28 |
Family
ID=22153993
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK99105755T DK0949250T3 (da) | 1998-03-30 | 1999-03-22 | Fremgangsmåde til fremstilling af alpha1L-adrenoceptorantagonister |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US6156894A (da) |
| EP (1) | EP0949250B1 (da) |
| JP (1) | JP3276342B2 (da) |
| KR (1) | KR100347469B1 (da) |
| CN (1) | CN1136199C (da) |
| AT (1) | ATE325104T1 (da) |
| CA (1) | CA2267510C (da) |
| DE (1) | DE69931100T2 (da) |
| DK (1) | DK0949250T3 (da) |
| ES (1) | ES2263238T3 (da) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5127366B2 (ja) | 2007-08-29 | 2013-01-23 | 富士通コンポーネント株式会社 | 情報処理装置、ｋｖｍスイッチ、サーバ及び制御プログラム |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3867456A (en) * | 1965-07-30 | 1975-02-18 | Oreal | Mono-omega-haloalkyl amines |
| JPS5324952B2 (da) * | 1973-11-28 | 1978-07-24 | ||
| US5859014A (en) * | 1995-06-09 | 1999-01-12 | Syntex (U.S.A.) Inc. | Pyrimidinedione, pyrimidinetrione, triazinedione and tetrahydroquinazolinedione derivatives as α1 -adrenergic receptor antagonists |
| EP0748800B1 (en) * | 1995-06-09 | 2001-05-09 | F. Hoffmann-La Roche Ag | Pyrimidinedione, pyrimidinetrione, triazinedione derivatives as alpha-1-adrenergic receptor antagonists |
| HRP970239B1 (en) * | 1997-05-09 | 2004-04-30 | Inst Ru Er Bouekovic | Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity |
-
1999
- 1999-03-22 ES ES99105755T patent/ES2263238T3/es not_active Expired - Lifetime
- 1999-03-22 EP EP99105755A patent/EP0949250B1/en not_active Expired - Lifetime
- 1999-03-22 DK DK99105755T patent/DK0949250T3/da active
- 1999-03-22 DE DE69931100T patent/DE69931100T2/de not_active Expired - Fee Related
- 1999-03-22 AT AT99105755T patent/ATE325104T1/de not_active IP Right Cessation
- 1999-03-24 US US09/275,333 patent/US6156894A/en not_active Expired - Fee Related
- 1999-03-29 CA CA002267510A patent/CA2267510C/en not_active Expired - Fee Related
- 1999-03-29 KR KR1019990010780A patent/KR100347469B1/ko not_active IP Right Cessation
- 1999-03-29 JP JP08508899A patent/JP3276342B2/ja not_active Expired - Fee Related
- 1999-03-30 CN CNB991045041A patent/CN1136199C/zh not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CN1234398A (zh) | 1999-11-10 |
| CA2267510C (en) | 2005-05-17 |
| JPH11322724A (ja) | 1999-11-24 |
| KR19990078360A (ko) | 1999-10-25 |
| DE69931100T2 (de) | 2007-04-19 |
| EP0949250A1 (en) | 1999-10-13 |
| ATE325104T1 (de) | 2006-06-15 |
| JP3276342B2 (ja) | 2002-04-22 |
| CA2267510A1 (en) | 1999-09-30 |
| US6156894A (en) | 2000-12-05 |
| KR100347469B1 (ko) | 2002-08-07 |
| ES2263238T3 (es) | 2006-12-01 |
| EP0949250B1 (en) | 2006-05-03 |
| CN1136199C (zh) | 2004-01-28 |
| DE69931100D1 (de) | 2006-06-08 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NO932870L (no) | Ny fremgangsmaate for fremstilling av 9-amino-6-demetyl-6-deoksyetracykliner | |
| MXPA04001323A (es) | Dihidro-3-halo-1h-pirazol-5-carboxilatos sustituidos, su preparacion y uso. | |
| ES2188661T3 (es) | Preparacion de un derivado de camptothecin por ciclacion intramolecular. | |
| EA200200481A1 (ru) | Способ получения производных 4-трифторметилсульфинилпиразола | |
| ATE442363T1 (de) | Verfahren zur herstellung von pyridinverbindungen | |
| DK0503453T3 (da) | Fremgangsmåde til fremstilling af cephalosporiner og mellemprodukter i denne fremgangsmåde | |
| DE60228724D1 (de) | Verfahren zur herstellung von beraprost und dessen salzen | |
| DE60235365D1 (de) | Verfahren zur herstellung von 7-amino-syn-3,5-dihydroxyheptansäurederivaten und zwischenverbindungen diesesverfahrens und deren herestellung | |
| TR200302288T2 (tr) | Terapi için yeni bileşikler ve metotlar. | |
| DE59910677D1 (de) | Verfahren sowie neue zwischenprodukte zur herstellung von isoxazolin-3-yl-acylbenzolen | |
| ATE255103T1 (de) | Verfahren zur herstellung von pyridinmethanol- verbindungen | |
| ES2158425T3 (es) | Procedimiento para la preparacion de derivados de pirimidina. | |
| DK0781764T3 (da) | Fremgangsmåde til fremstilling af alkoxyiminoacetamid-derivater | |
| ATE266618T1 (de) | Verfahren zur herstellung von zwischenprodukten für pestizide | |
| DE60224884D1 (de) | Verfahren zur herstellung von 3, 3', 6, 6'-tetraalkylen-2, 2'-biphenolen und 3, 3', 6, 6'-tetraalkylen-5, 5'-dihalo-2, 2' biphenolen | |
| DK0949250T3 (da) | Fremgangsmåde til fremstilling af alpha1L-adrenoceptorantagonister | |
| BR9503845A (pt) | Processo para a preparação de um composto e composto obtido | |
| NZ333229A (da) | ||
| DK1105392T3 (da) | Fremgangsmåde til fremstilling af mellemprodukter for imidazodiazepin | |
| MY130817A (en) | Herbicides | |
| EE200300090A (et) | Asendatud imidasopüridiinühendite valmistamise meetod | |
| DK0979822T3 (da) | Fremgangsmåde til fremstilling af 2-carbamoyl-pyridiner | |
| DK0662475T3 (da) | Fremgangsmåde til fremstilling af 2-perfluoralkyl-3-oxazolin-5-on. | |
| ATE286058T1 (de) | Thiazolpyrimidin-verbindungen, verfahren zu ihrer herstellung und ihre anwendung | |
| DK0492350T3 (da) | Fremgangsmåde til fremstilling af (S)-vinyl- og (S)-allenyl-GABA |