DK0948525T3 - Cyclopeptidderivater - Google Patents

Cyclopeptidderivater

Info

Publication number
DK0948525T3
DK0948525T3 DK97953826T DK97953826T DK0948525T3 DK 0948525 T3 DK0948525 T3 DK 0948525T3 DK 97953826 T DK97953826 T DK 97953826T DK 97953826 T DK97953826 T DK 97953826T DK 0948525 T3 DK0948525 T3 DK 0948525T3
Authority
DK
Denmark
Prior art keywords
cyclopeptide derivatives
cyclopeptide
derivatives
Prior art date
Application number
DK97953826T
Other languages
Danish (da)
English (en)
Inventor
Guenter Hoelzemann
Claus Fittschen
Simon Goodman
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Application granted granted Critical
Publication of DK0948525T3 publication Critical patent/DK0948525T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK97953826T 1996-12-19 1997-12-15 Cyclopeptidderivater DK0948525T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19653036A DE19653036A1 (de) 1996-12-19 1996-12-19 Cyclopeptidderivate
PCT/EP1997/007048 WO1998027112A1 (de) 1996-12-19 1997-12-15 Cyclopeptidderivate

Publications (1)

Publication Number Publication Date
DK0948525T3 true DK0948525T3 (da) 2001-06-11

Family

ID=7815374

Family Applications (1)

Application Number Title Priority Date Filing Date
DK97953826T DK0948525T3 (da) 1996-12-19 1997-12-15 Cyclopeptidderivater

Country Status (22)

Country Link
US (1) US6333308B1 (ru)
EP (1) EP0948525B1 (ru)
CN (1) CN1247543A (ru)
AR (1) AR008717A1 (ru)
AT (1) ATE199256T1 (ru)
AU (1) AU722817B2 (ru)
CA (1) CA2280233A1 (ru)
CZ (1) CZ223299A3 (ru)
DE (2) DE19653036A1 (ru)
DK (1) DK0948525T3 (ru)
ES (1) ES2156011T3 (ru)
GR (1) GR3035848T3 (ru)
HU (1) HUP0000490A3 (ru)
NO (1) NO993010L (ru)
PL (1) PL334186A1 (ru)
PT (1) PT948525E (ru)
RU (1) RU2202557C2 (ru)
SK (1) SK82099A3 (ru)
TW (1) TW494105B (ru)
UA (1) UA55439C2 (ru)
WO (1) WO1998027112A1 (ru)
ZA (1) ZA9711392B (ru)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19728524A1 (de) 1997-07-04 1999-01-07 Merck Patent Gmbh Cyclische Azapeptide
US6235877B1 (en) * 1999-08-04 2001-05-22 Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. Peptido-mimetic compounds containing RGD sequence useful as integrin inhibitors
DE10041402A1 (de) * 2000-08-23 2002-03-14 Morphochem Ag Neue Verbindungen, die Faktor Xa-Aktivität inhibieren
US7087768B2 (en) * 2001-09-27 2006-08-08 Equispharm Co., Ltd. Fumagillol derivatives and preparing method thereof
ITMI20031476A1 (it) * 2003-07-18 2005-01-19 Univ Degli Studi Milano Composti peptido-mimetici a struttura azabicicloalcanica comprendenti la sequenza rgd
ES2413056T3 (es) * 2005-10-12 2013-07-15 Advanced Accelerator Applications Antagonista del péptido receptor Alfavbeta3 selectivo para aplicaciones terapéuticas y de diagnóstico

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0648224B1 (en) * 1992-06-04 1998-07-15 Merrell Pharmaceuticals Inc. Conformationally restrained peptide analogs as antiplatelet agents
GB9524630D0 (en) * 1994-12-24 1996-01-31 Zeneca Ltd Chemical compounds
JPH09278669A (ja) * 1996-04-17 1997-10-28 Asahi Glass Co Ltd 腎炎治療薬

Also Published As

Publication number Publication date
TW494105B (en) 2002-07-11
UA55439C2 (ru) 2003-04-15
RU2202557C2 (ru) 2003-04-20
NO993010D0 (no) 1999-06-18
PT948525E (pt) 2001-07-31
US6333308B1 (en) 2001-12-25
AU5758498A (en) 1998-07-15
GR3035848T3 (en) 2001-08-31
ZA9711392B (en) 1999-06-18
CN1247543A (zh) 2000-03-15
PL334186A1 (en) 2000-02-14
NO993010L (no) 1999-08-18
ES2156011T3 (es) 2001-06-01
DE59703023D1 (en) 2001-03-29
CA2280233A1 (en) 1998-06-25
WO1998027112A1 (de) 1998-06-25
DE19653036A1 (de) 1998-06-25
CZ223299A3 (cs) 1999-09-15
SK82099A3 (en) 2000-06-12
EP0948525A1 (de) 1999-10-13
AU722817B2 (en) 2000-08-10
EP0948525B1 (de) 2001-02-21
HUP0000490A2 (hu) 2000-08-28
HUP0000490A3 (en) 2000-10-30
ATE199256T1 (de) 2001-03-15
AR008717A1 (es) 2000-02-09

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