DK0937100T3 - En ny polymorfisk krystallinsk form af fluticasonpropionat, fremgangsmåder til fremstilling deraf og farmaceutiske præparater deraf - Google Patents

En ny polymorfisk krystallinsk form af fluticasonpropionat, fremgangsmåder til fremstilling deraf og farmaceutiske præparater deraf

Info

Publication number
DK0937100T3
DK0937100T3 DK97909496T DK97909496T DK0937100T3 DK 0937100 T3 DK0937100 T3 DK 0937100T3 DK 97909496 T DK97909496 T DK 97909496T DK 97909496 T DK97909496 T DK 97909496T DK 0937100 T3 DK0937100 T3 DK 0937100T3
Authority
DK
Denmark
Prior art keywords
crystalline form
polymorphic crystalline
fluticasone propionate
new polymorphic
preparation
Prior art date
Application number
DK97909496T
Other languages
Danish (da)
English (en)
Inventor
Simon Murray Cooper
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of DK0937100T3 publication Critical patent/DK0937100T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Disintegrating Or Milling (AREA)
  • Formation And Processing Of Food Products (AREA)
DK97909496T 1996-10-24 1997-10-23 En ny polymorfisk krystallinsk form af fluticasonpropionat, fremgangsmåder til fremstilling deraf og farmaceutiske præparater deraf DK0937100T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9622173.4A GB9622173D0 (en) 1996-10-24 1996-10-24 Particulate Products
PCT/GB1997/002929 WO1998017676A1 (fr) 1996-10-24 1997-10-23 Nouvelle forme cristalline polymorphe de propionate de fluticasone, son procede de production et des compositions pharmaceutiques la renfermant

Publications (1)

Publication Number Publication Date
DK0937100T3 true DK0937100T3 (da) 2003-09-01

Family

ID=10801903

Family Applications (1)

Application Number Title Priority Date Filing Date
DK97909496T DK0937100T3 (da) 1996-10-24 1997-10-23 En ny polymorfisk krystallinsk form af fluticasonpropionat, fremgangsmåder til fremstilling deraf og farmaceutiske præparater deraf

Country Status (13)

Country Link
US (1) US6406718B1 (fr)
EP (1) EP0937100B1 (fr)
JP (1) JP2001502350A (fr)
AT (1) ATE240345T1 (fr)
AU (1) AU4717197A (fr)
CA (1) CA2269134C (fr)
DE (1) DE69722023T2 (fr)
DK (1) DK0937100T3 (fr)
ES (1) ES2198555T3 (fr)
GB (1) GB9622173D0 (fr)
PE (1) PE68099A1 (fr)
PT (1) PT937100E (fr)
WO (1) WO1998017676A1 (fr)

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US9339459B2 (en) 2003-04-24 2016-05-17 Nektar Therapeutics Particulate materials
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US20040208833A1 (en) * 2003-02-04 2004-10-21 Elan Pharma International Ltd. Novel fluticasone formulations
CA2524773C (fr) 2003-05-08 2014-04-08 Nektar Therapeutics Uk Ltd Coformulations particulaires de substances actives comprenant des excipients
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US20060009435A1 (en) * 2004-06-23 2006-01-12 Joseph Kaspi Synthesis and powder preparation of fluticasone propionate
EP1904219A4 (fr) 2005-07-15 2011-07-27 Map Pharmaceuticals Inc Procede de formation de particules
US11311477B2 (en) 2006-03-07 2022-04-26 Sgn Nanopharma Inc. Ophthalmic preparations
WO2007103294A2 (fr) * 2006-03-07 2007-09-13 Novavax, Inc. Compositions nano-structurees et leurs procedes de fabrication et d'utilisation
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EP3167875A1 (fr) 2009-05-27 2017-05-17 Alkermes Pharma Ireland Limited Réduction d'agrégation de type paillettes dans des compositions de meloxicam nanoparticulaire
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IL293779B2 (en) * 2012-01-13 2023-09-01 Xspray Microparticles Ab A pharmaceutical preparation containing stable amorphous hybrid nanoparticles of at least one protein kinase inhibitor and at least one polymeric stabilizing and matrix-forming component
US8765725B2 (en) 2012-05-08 2014-07-01 Aciex Therapeutics, Inc. Preparations of hydrophobic therapeutic agents, methods of manufacture and use thereof
BR112014027681B8 (pt) 2012-05-08 2023-10-31 Aciex Therapeutics Inc Nanocristais de propionato de fluticasona, composição tópica farmacêutica compreendendo os mesmos, seu uso e método de fabricação
US9815865B2 (en) 2013-01-07 2017-11-14 Nicox Ophthalmics, Inc. Preparations of hydrophobic therapeutic agents, methods of manufacture and use thereof
US9452173B2 (en) 2013-01-31 2016-09-27 Merz Pharmaceuticals, Llc Topical compositions and methods for making and using same
US8778365B1 (en) 2013-01-31 2014-07-15 Merz Pharmaceuticals, Llc Topical compositions and methods for making and using same
US9433680B2 (en) 2013-01-31 2016-09-06 Merz Pharmaceuticals, Llc Topical compositions and methods for making and using same
US9446131B2 (en) 2013-01-31 2016-09-20 Merz Pharmaceuticals, Llc Topical compositions and methods for making and using same
CN104004044A (zh) * 2013-02-25 2014-08-27 武汉诺安药业有限公司 高纯度丙酸氟替卡松制备方法
CN112494492B (zh) 2014-08-18 2023-08-25 阿尔科姆斯制药爱尔兰有限公司 阿立哌唑前体药物组合物
US10016415B2 (en) 2014-08-18 2018-07-10 Alkermes Pharma Ireland Limited Aripiprazole prodrug compositions
CN108066329B (zh) * 2016-11-11 2021-11-16 江苏恒瑞医药股份有限公司 一种吸入用氟替卡松或其衍生物的微粒的制备方法
WO2021219230A1 (fr) 2020-04-30 2021-11-04 Paolo Fiorina Traitement antiviral

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Also Published As

Publication number Publication date
US6406718B1 (en) 2002-06-18
GB9622173D0 (en) 1996-12-18
DE69722023T2 (de) 2004-04-08
AU4717197A (en) 1998-05-15
JP2001502350A (ja) 2001-02-20
PE68099A1 (es) 1999-07-19
DE69722023D1 (de) 2003-06-18
ES2198555T3 (es) 2004-02-01
WO1998017676A1 (fr) 1998-04-30
EP0937100A1 (fr) 1999-08-25
PT937100E (pt) 2003-09-30
ATE240345T1 (de) 2003-05-15
CA2269134A1 (fr) 1998-04-30
CA2269134C (fr) 2007-01-09
EP0937100B1 (fr) 2003-05-14

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