DK0877738T3 - Fremgangsmåde til fremstilling af phenylimidazolidinderivater - Google Patents

Fremgangsmåde til fremstilling af phenylimidazolidinderivater

Info

Publication number
DK0877738T3
DK0877738T3 DK96938306T DK96938306T DK0877738T3 DK 0877738 T3 DK0877738 T3 DK 0877738T3 DK 96938306 T DK96938306 T DK 96938306T DK 96938306 T DK96938306 T DK 96938306T DK 0877738 T3 DK0877738 T3 DK 0877738T3
Authority
DK
Denmark
Prior art keywords
preparation
phenylimidazolidine
derivatives
phenylimidazolidine derivatives
Prior art date
Application number
DK96938306T
Other languages
Danish (da)
English (en)
Inventor
Raphaoel Bouchet
Michel Delthil
Daniel Guilmard
Philippe Mackiewicz
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Application granted granted Critical
Publication of DK0877738T3 publication Critical patent/DK0877738T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/72—Two oxygen atoms, e.g. hydantoin
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK96938306T 1995-11-16 1996-11-14 Fremgangsmåde til fremstilling af phenylimidazolidinderivater DK0877738T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9513589A FR2741346B1 (fr) 1995-11-16 1995-11-16 Nouveau procede de preparation de derives phenylimidazolidine
PCT/FR1996/001794 WO1997018197A1 (fr) 1995-11-16 1996-11-14 Nouveau procede de preparation de derives phenylimidazolidine

Publications (1)

Publication Number Publication Date
DK0877738T3 true DK0877738T3 (da) 2003-09-08

Family

ID=9484624

Family Applications (1)

Application Number Title Priority Date Filing Date
DK96938306T DK0877738T3 (da) 1995-11-16 1996-11-14 Fremgangsmåde til fremstilling af phenylimidazolidinderivater

Country Status (29)

Country Link
US (1) US6107488A (no)
EP (1) EP0877738B1 (no)
JP (1) JP2000500150A (no)
KR (1) KR100466991B1 (no)
CN (1) CN1131219C (no)
AR (1) AR004965A1 (no)
AT (1) ATE240300T1 (no)
AU (1) AU718832B2 (no)
BR (1) BR9611573A (no)
CA (1) CA2235335A1 (no)
CU (1) CU22890A3 (no)
CZ (1) CZ144498A3 (no)
DE (1) DE69628203T2 (no)
DK (1) DK0877738T3 (no)
EA (1) EA002658B1 (no)
ES (1) ES2193271T3 (no)
FR (1) FR2741346B1 (no)
HU (1) HUP9904034A3 (no)
IL (1) IL124382A0 (no)
MX (1) MX9803730A (no)
NO (1) NO316514B1 (no)
PL (1) PL189697B1 (no)
PT (1) PT877738E (no)
SI (1) SI0877738T1 (no)
TR (1) TR199800865T2 (no)
TW (1) TW404942B (no)
UA (1) UA67720C2 (no)
WO (1) WO1997018197A1 (no)
ZA (1) ZA969442B (no)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007514442A (ja) * 2003-12-19 2007-06-07 ザ リージェンツ オブ ザ ユニバーシティ オブ カリフォルニア 前立腺癌治療を評価するための方法および物質
NZ550102A (en) * 2004-02-24 2010-10-29 Univ California Methods and materials for assessing prostate cancer therapies and compounds (thiohydantoine derivatives)
US7709517B2 (en) 2005-05-13 2010-05-04 The Regents Of The University Of California Diarylhydantoin compounds
HUE053877T2 (hu) 2006-03-27 2021-07-28 Univ California Androgén receptormodulátor a prosztatarák és az androgén receptorral összefüggõ betegségek kezeléséhez
NZ572374A (en) 2006-03-29 2011-12-22 Univ California Diarylthiohydantoin compounds
CA2703635C (en) 2007-10-26 2017-06-27 Michael E. Jung Diarylhydantoin compounds as androgen receptor modulators
CN102481294A (zh) 2009-09-11 2012-05-30 拜耳医药股份有限公司 作为抗癌药物的取代(杂芳基甲基)乙内酰硫脲
EP2478020A4 (en) 2009-09-15 2015-04-15 Mylan Group COPOLYMERS, POLYMER PARTICLES WITH THESE COPOLYMERS AND COPOLYMER BINDER FOR RADIATION-SENSITIVE COATING COMPOSITIONS FOR NEGATIVELY WORKING RADIATION-SENSITIVE LITHOGRAPHIC PLASTERS
CN106983749A (zh) 2010-02-16 2017-07-28 亚拉冈制药公司 雄激素受体调节剂及其用途
UA106533C2 (uk) 2010-09-14 2014-09-10 Майлен Груп Співполімери для чутливих у близькій інфрачервоній області випромінювання композицій для покриття позитивних термічних літографічних друкарських форм
BR112015006705A8 (pt) 2012-09-26 2019-08-27 Aragon Pharmaceuticals Inc antiandrogênios para o tratamento de câncer de próstata resistente à castração não metastático e usos destes
JOP20200097A1 (ar) 2013-01-15 2017-06-16 Aragon Pharmaceuticals Inc معدل مستقبل أندروجين واستخداماته
TWI726969B (zh) 2016-01-11 2021-05-11 比利時商健生藥品公司 用作雄性激素受體拮抗劑之經取代之硫尿囊素衍生物
CA3079135A1 (en) 2017-10-16 2019-04-25 Arturo Molina Anti-androgens for the treatment of non-metastatic castration-resistant prostate cancer
CN108218784A (zh) * 2018-01-16 2018-06-29 吴江信凯医药科技有限公司 一种尼鲁米特的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS4916937B1 (no) * 1970-01-21 1974-04-25
JPS5136332B1 (no) * 1970-12-09 1976-10-07
CH544491A (de) * 1971-03-16 1973-11-30 Ciba Geigy Ag Herbizides Mittel
MC1220A1 (fr) * 1977-10-28 1979-07-20 Hoffmann La Roche Nouveaux derives d'imidazolidine
JPS57197268A (en) * 1981-05-29 1982-12-03 Sumitomo Chem Co Ltd Substituted phenylhydantoin derivative, its preparation, and herbicide containing the same as active ingredient
JPS62298562A (ja) * 1986-06-17 1987-12-25 Nippon Kayaku Co Ltd ブロモアニリン類の製造法
FR2656302B1 (fr) * 1989-12-22 1992-05-07 Roussel Uclaf Nouveau procede de preparation de l'anandron et derives de l'anandron.
US5411981A (en) * 1991-01-09 1995-05-02 Roussel Uclaf Phenylimidazolidines having antiandrogenic activity
FR2694290B1 (fr) * 1992-07-08 1994-09-02 Roussel Uclaf Nouvelles phénylimidazolidines éventuellement substituées, leur procédé de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant.

Also Published As

Publication number Publication date
TR199800865T2 (xx) 1998-08-21
EP0877738B1 (fr) 2003-05-14
DE69628203D1 (de) 2003-06-18
AU7577396A (en) 1997-06-05
HUP9904034A3 (en) 2001-08-28
HUP9904034A2 (hu) 2000-05-28
CA2235335A1 (fr) 1997-05-22
PT877738E (pt) 2003-09-30
EA002658B1 (ru) 2002-08-29
AU718832B2 (en) 2000-04-20
BR9611573A (pt) 1999-05-11
IL124382A0 (en) 1998-12-06
CN1131219C (zh) 2003-12-17
FR2741346A1 (fr) 1997-05-23
ZA969442B (en) 1997-11-11
CN1207732A (zh) 1999-02-10
CU22890A3 (es) 2004-01-23
UA67720C2 (en) 2004-07-15
FR2741346B1 (fr) 1997-12-19
ES2193271T3 (es) 2003-11-01
EA199800378A1 (ru) 1998-10-29
NO316514B1 (no) 2004-02-02
US6107488A (en) 2000-08-22
NO982237L (no) 1998-07-10
EP0877738A1 (fr) 1998-11-18
SI0877738T1 (en) 2003-10-31
WO1997018197A1 (fr) 1997-05-22
DE69628203T2 (de) 2004-02-05
PL189697B1 (pl) 2005-09-30
KR19990067639A (ko) 1999-08-25
TW404942B (en) 2000-09-11
NO982237D0 (no) 1998-05-15
PL326491A1 (en) 1998-09-28
MX9803730A (es) 1998-11-30
ATE240300T1 (de) 2003-05-15
JP2000500150A (ja) 2000-01-11
KR100466991B1 (ko) 2005-04-06
CZ144498A3 (cs) 1998-09-16
AR004965A1 (es) 1999-04-07

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