DK0780375T3 - 3-((5-substitueret benzyl)amino)-2-phenylpiperidiner som substans P-antagonister - Google Patents
3-((5-substitueret benzyl)amino)-2-phenylpiperidiner som substans P-antagonisterInfo
- Publication number
- DK0780375T3 DK0780375T3 DK96203560T DK96203560T DK0780375T3 DK 0780375 T3 DK0780375 T3 DK 0780375T3 DK 96203560 T DK96203560 T DK 96203560T DK 96203560 T DK96203560 T DK 96203560T DK 0780375 T3 DK0780375 T3 DK 0780375T3
- Authority
- DK
- Denmark
- Prior art keywords
- alkyl
- halo
- disorders
- cycloalkyl
- hydrogen
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IB9501148 | 1995-12-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
DK0780375T3 true DK0780375T3 (da) | 2002-10-07 |
Family
ID=11004393
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK96203560T DK0780375T3 (da) | 1995-12-21 | 1996-12-16 | 3-((5-substitueret benzyl)amino)-2-phenylpiperidiner som substans P-antagonister |
Country Status (8)
Country | Link |
---|---|
US (1) | US5789423A (da) |
EP (1) | EP0780375B1 (da) |
AT (1) | ATE223896T1 (da) |
CA (1) | CA2193468C (da) |
DE (1) | DE69623580T2 (da) |
DK (1) | DK0780375T3 (da) |
ES (1) | ES2180693T3 (da) |
PT (1) | PT780375E (da) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW340842B (en) * | 1995-08-24 | 1998-09-21 | Pfizer | Substituted benzylaminopiperidine compounds |
JP2002506459A (ja) * | 1997-06-27 | 2002-02-26 | メルク シヤープ エンド ドーム リミテツド | 置換された3−(ベンジルアミノ)ピペリジン誘導体およびその治療薬としての使用 |
OA11864A (en) * | 1999-05-06 | 2006-03-03 | Pfizer Prod Inc | Substituted benzolactam compounds. |
KR20030036834A (ko) * | 2000-09-26 | 2003-05-09 | 다나베 세이야꾸 가부시키가이샤 | 5-페닐벤질아민 화합물, 그의 제법 및 그의 합성 중간체 |
US10154988B2 (en) | 2012-11-14 | 2018-12-18 | The Johns Hopkins University | Methods and compositions for treating schizophrenia |
AU2015220427B2 (en) | 2014-02-19 | 2017-09-21 | Piramal Enterprises Limited | Compounds for use as GPR120 agonists |
EP3172185B1 (en) | 2014-07-25 | 2020-03-04 | Piramal Enterprises Limited | Substituted phenyl alkanoic acid compounds as gpr120 agonists and uses thereof |
AU2015313829B2 (en) | 2014-09-11 | 2020-07-23 | Piramal Enterprises Limited | Fused heterocyclic compounds as GPR120 agonists |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4680283A (en) | 1984-09-26 | 1987-07-14 | Merck & Co., Inc. | Analogs of substance P and eledoisin |
DE3602169A1 (de) | 1986-01-22 | 1987-07-23 | Schering Ag | Neue alkan- und alkoxyalkanderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende insektizide und akarizide mittel |
WO1991009844A1 (en) | 1990-01-04 | 1991-07-11 | Pfizer Inc. | Substance p antagonists |
US5232929A (en) * | 1990-11-28 | 1993-08-03 | Pfizer Inc. | 3-aminopiperidine derivatives and related nitrogen containing heterocycles and pharmaceutical compositions and use |
US5364943A (en) | 1991-11-27 | 1994-11-15 | Pfizer Inc. | Preparation of substituted piperidines |
RU2105001C1 (ru) * | 1991-03-26 | 1998-02-20 | Пфайзер Инк. | Способ получения замещенных 3-аминопиперидинов |
RU2114848C1 (ru) | 1991-06-20 | 1998-07-10 | Пфайзер Инк. | Фторалкоксибензиламинные производные азотсодержащих гетероциклов, фармацевтическая композиция, способ ингибирования действия вещества р у млекопитающих |
EP0655996B1 (en) * | 1992-08-19 | 2001-11-07 | Pfizer Inc. | Substituted benzylamino nitrogen containing non-aromatic heterocycles |
GB9305718D0 (en) * | 1993-03-19 | 1993-05-05 | Glaxo Group Ltd | Medicaments |
IL109646A0 (en) | 1993-05-19 | 1994-08-26 | Pfizer | Heteroatom substituted alkyl benzylamino-quinuclidines |
-
1996
- 1996-12-16 PT PT96203560T patent/PT780375E/pt unknown
- 1996-12-16 DE DE69623580T patent/DE69623580T2/de not_active Expired - Fee Related
- 1996-12-16 ES ES96203560T patent/ES2180693T3/es not_active Expired - Lifetime
- 1996-12-16 AT AT96203560T patent/ATE223896T1/de not_active IP Right Cessation
- 1996-12-16 DK DK96203560T patent/DK0780375T3/da active
- 1996-12-16 EP EP96203560A patent/EP0780375B1/en not_active Expired - Lifetime
- 1996-12-17 US US08/767,985 patent/US5789423A/en not_active Expired - Fee Related
- 1996-12-19 CA CA002193468A patent/CA2193468C/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
DE69623580D1 (de) | 2002-10-17 |
ATE223896T1 (de) | 2002-09-15 |
CA2193468C (en) | 2001-04-24 |
US5789423A (en) | 1998-08-04 |
DE69623580T2 (de) | 2003-01-09 |
EP0780375B1 (en) | 2002-09-11 |
ES2180693T3 (es) | 2003-02-16 |
EP0780375A1 (en) | 1997-06-25 |
PT780375E (pt) | 2002-12-31 |
CA2193468A1 (en) | 1997-06-22 |
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