DK0771217T3 - Faste lægemiddelformer, som indeholder clathrater af det steroide könshormon ethinylestadiol - Google Patents

Faste lægemiddelformer, som indeholder clathrater af det steroide könshormon ethinylestadiol

Info

Publication number
DK0771217T3
DK0771217T3 DK95943492T DK95943492T DK0771217T3 DK 0771217 T3 DK0771217 T3 DK 0771217T3 DK 95943492 T DK95943492 T DK 95943492T DK 95943492 T DK95943492 T DK 95943492T DK 0771217 T3 DK0771217 T3 DK 0771217T3
Authority
DK
Denmark
Prior art keywords
estadiol
solid pharmaceutical
pharmaceutical forms
forms containing
sex hormone
Prior art date
Application number
DK95943492T
Other languages
Danish (da)
English (en)
Inventor
Johannes Tack
Thomas Backensfeld
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=6524338&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK0771217(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Ag filed Critical Schering Ag
Application granted granted Critical
Publication of DK0771217T3 publication Critical patent/DK0771217T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/69—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit
    • A61K47/6949—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes
    • A61K47/6951—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes using cyclodextrin
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B82—NANOTECHNOLOGY
    • B82Y—SPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00—Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Nanotechnology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • General Engineering & Computer Science (AREA)
  • Medical Informatics (AREA)
  • Biotechnology (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Biophysics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Steroid Compounds (AREA)
DK95943492T 1994-07-20 1995-07-10 Faste lægemiddelformer, som indeholder clathrater af det steroide könshormon ethinylestadiol DK0771217T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4426709A DE4426709A1 (de) 1994-07-20 1994-07-20 Steroidale Sexualhormone enthaltende feste Arzneiformen
PCT/EP1995/002656 WO1996002277A1 (de) 1994-07-20 1995-07-10 Feste arzneiformen, enthaltend clathrate von steroidalen sexualhormonen

Publications (1)

Publication Number Publication Date
DK0771217T3 true DK0771217T3 (da) 2004-08-02

Family

ID=6524338

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95943492T DK0771217T3 (da) 1994-07-20 1995-07-10 Faste lægemiddelformer, som indeholder clathrater af det steroide könshormon ethinylestadiol

Country Status (11)

Country Link
US (1) US5798338A (enEXAMPLES)
EP (1) EP0771217B1 (enEXAMPLES)
JP (1) JPH10502912A (enEXAMPLES)
AT (1) ATE263578T1 (enEXAMPLES)
CA (1) CA2194979C (enEXAMPLES)
DE (4) DE4426709A1 (enEXAMPLES)
DK (1) DK0771217T3 (enEXAMPLES)
ES (1) ES2218561T3 (enEXAMPLES)
FR (1) FR07C0001I2 (enEXAMPLES)
PT (1) PT771217E (enEXAMPLES)
WO (1) WO1996002277A1 (enEXAMPLES)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19652196A1 (de) * 1996-12-16 1998-06-18 Jenapharm Gmbh Homogene steroidhaltige Präformulierungen zur Herstellung niedrigdosierter fester und halbfester pharmazeutischer Zubereitungen
DE19848303A1 (de) * 1998-10-14 2000-04-20 Schering Ag Kombination aus Gestagenen und Zuckern
EP1216712A1 (en) * 2000-12-20 2002-06-26 Schering Aktiengesellschaft Cyclodextrin-drospirenone inclusion complexes
EP1353699B1 (en) * 2000-12-20 2012-02-01 Bayer Pharma Aktiengesellschaft Beta-cyclodextrin-drospirenone inclusion complexes
EP1216713A1 (en) * 2000-12-20 2002-06-26 Schering Aktiengesellschaft Compositions of estrogen-cyclodextrin complexes
US20050020554A1 (en) * 2003-06-06 2005-01-27 Ahmed Salah U. Stability of hormone formulations
WO2005117899A1 (en) * 2004-06-02 2005-12-15 Cipla Limited Pharmaceutical composition comprising tibolone and process for procuding the same
US20070287684A1 (en) * 2006-05-22 2007-12-13 Irshad Chaudry Methods and compositions for treating trauma-hemorrhage using estrogen and derivatives thereof
CN101489563A (zh) 2006-07-06 2009-07-22 拜耳先灵医药股份有限公司 用于避孕和预防先天性畸形风险的药物制剂
US8617597B2 (en) * 2006-07-06 2013-12-31 Bayer Intellectual Property Gmbh Pharmaceutical composition containing a tetrahydrofolic acid
AU2009214193A1 (en) * 2008-02-13 2009-08-20 Bayer Intellectual Property Gmbh Estradiol-containing drug delivery system
EP2252261A2 (en) * 2008-02-13 2010-11-24 Bayer Schering Pharma Aktiengesellschaft Drug delivery system with stabilising effect
CA2725578A1 (en) * 2008-04-24 2009-10-29 Evestra, Inc. Oral contraceptive dosage forms comprising a progestogen dispersed in an enteric polymer and further comprising an estrogen
EP2143432A1 (en) 2008-07-11 2010-01-13 Bayer Schering Pharma AG 9-alpha estratriene derivatives as ER-beta selective ligands for the prevention and treatment of intestinal cancer
UY32836A (es) 2009-08-12 2011-03-31 Bayer Schering Pharma Ag Partículas estabilizadas que comprenden 5-metil-(6s)-tetrahidrofolato
EP2558063B1 (en) 2010-04-15 2021-09-29 Bayer Intellectual Property GmbH Very low-dosed solid oral dosage forms for hrt
CA2796139A1 (en) 2010-04-15 2011-10-20 Bayer Intellectual Property Gmbh Low-dosed solid oral dosage forms for hrt
CN101869113B (zh) * 2010-06-17 2013-09-04 中国农业科学院植物保护研究所 一种鼠类不育剂的环糊精包合物及其制备方法
JP2013537219A (ja) 2010-09-16 2013-09-30 シモダ・バイオテック・（ピーティーワイ）・リミテッド フルベストラント組成物および使用方法
WO2012120365A1 (en) 2011-03-07 2012-09-13 Aurobindo Pharma Limited Stable pharmaceutical composition comprising ethinyl estradiol
US9359451B2 (en) 2012-05-15 2016-06-07 The Uab Research Foundation Methods and compositions for treating trauma-hemorrhage using estrogen and derivatives thereof
ES2858573T3 (es) 2017-10-16 2021-09-30 Faes Farma Sa Composiciones acuosas que comprenden bilastina y mometasona
EP3666260A1 (en) 2018-12-13 2020-06-17 Laboratorios Leon Farma SA Ethinyl estradiol-beta-cyclodextrin complex and process for preparing thereof
CN114225050B (zh) * 2022-01-29 2022-12-13 国家卫生健康委科学技术研究所 炔雌醇环糊精复合物的制备及应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57106698A (en) * 1980-12-22 1982-07-02 Kyowa Hakko Kogyo Co Ltd Easily absorbable map composition and preparation containing the same
US4596795A (en) * 1984-04-25 1986-06-24 The United States Of America As Represented By The Secretary, Dept. Of Health & Human Services Administration of sex hormones in the form of hydrophilic cyclodextrin derivatives
JPH0764884B2 (ja) * 1986-11-27 1995-07-12 株式会社トクヤマ シクロデキストリン組成物
US4877774A (en) * 1987-09-09 1989-10-31 The United States Of America As Represented By The Department Of Health And Human Services Administration of steroid hormones

Also Published As

Publication number Publication date
CA2194979C (en) 2009-01-06
FR07C0001I1 (enEXAMPLES) 2007-03-09
CA2194979A1 (en) 1996-02-01
FR07C0001I2 (enEXAMPLES) 2009-01-02
US5798338A (en) 1998-08-25
DE4426709A1 (de) 1996-01-25
WO1996002277A1 (de) 1996-02-01
PT771217E (pt) 2004-08-31
EP0771217B1 (de) 2004-04-07
DE122007000013I1 (enEXAMPLES) 2007-04-26
DE59510887D1 (de) 2004-05-13
DE122007000011I1 (de) 2007-05-10
JPH10502912A (ja) 1998-03-17
ATE263578T1 (de) 2004-04-15
ES2218561T3 (es) 2004-11-16
EP0771217A1 (de) 1997-05-07

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