DK0764150T3 - Fremstilling af hydroxythioacetamider og anvendelse deraf ved syntese af benzothiophener - Google Patents
Fremstilling af hydroxythioacetamider og anvendelse deraf ved syntese af benzothiophenerInfo
- Publication number
- DK0764150T3 DK0764150T3 DK95923804T DK95923804T DK0764150T3 DK 0764150 T3 DK0764150 T3 DK 0764150T3 DK 95923804 T DK95923804 T DK 95923804T DK 95923804 T DK95923804 T DK 95923804T DK 0764150 T3 DK0764150 T3 DK 0764150T3
- Authority
- DK
- Denmark
- Prior art keywords
- benzo
- beta
- hydroxy
- thiophene
- alpha
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/56—Radicals substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C327/00—Thiocarboxylic acids
- C07C327/38—Amides of thiocarboxylic acids
- C07C327/40—Amides of thiocarboxylic acids having carbon atoms of thiocarboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C327/44—Amides of thiocarboxylic acids having carbon atoms of thiocarboxamide groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/66—Nitrogen atoms not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Investigating Or Analyzing Non-Biological Materials By The Use Of Chemical Means (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/258,641 US5420349A (en) | 1994-06-10 | 1994-06-10 | 2-amino-3-aroyl-benzo[β]thiophenes and methods for preparing and using same to produce 6-hydroxy-2-(4-hydroxyphenyl)-3-]benzo[4-(2-aminoethoxy)-benzoyl[β]thiophenes |
| PCT/US1995/007399 WO1995034536A1 (en) | 1994-06-10 | 1995-06-07 | Production of hydroxythioacetamides and use thereof in the synthesis of benzothiophenes |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0764150T3 true DK0764150T3 (da) | 1999-11-08 |
Family
ID=22981480
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK95923804T DK0764150T3 (da) | 1994-06-10 | 1995-06-07 | Fremstilling af hydroxythioacetamider og anvendelse deraf ved syntese af benzothiophener |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US5420349A (hu) |
| EP (1) | EP0764150B1 (hu) |
| JP (1) | JPH10503175A (hu) |
| AT (1) | ATE186050T1 (hu) |
| AU (1) | AU2823695A (hu) |
| BR (1) | BR9507968A (hu) |
| CA (1) | CA2192096A1 (hu) |
| DE (1) | DE69513022T2 (hu) |
| DK (1) | DK0764150T3 (hu) |
| ES (1) | ES2139222T3 (hu) |
| FI (1) | FI964854A0 (hu) |
| GR (1) | GR3032409T3 (hu) |
| HU (3) | HU217822B (hu) |
| WO (1) | WO1995034536A1 (hu) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5466810A (en) * | 1994-06-10 | 1995-11-14 | Eli Lilly And Company | 2-amino-3-aroyl-benzo[β]thiophenes and methods for preparing and using same to produce 6-hydroxy-2-(4-hydroxyphenyl)-3-[4-(2-aminoethoxy)-benzoyl]benzo[β]thiophenes |
| CA2214196A1 (en) * | 1996-09-26 | 1998-03-26 | Eli Lilly And Company | Benzo[b]indeno[2,1-d]thiophene compounds, intermediates, processes, compositions and methods |
| JP2001524114A (ja) * | 1997-04-30 | 2001-11-27 | イーライ・リリー・アンド・カンパニー | ベンゾ［ｂ］チオフェン類の製造における中間体および方法 |
| WO2004029046A2 (en) | 2002-09-30 | 2004-04-08 | A/S Gea Farmaceutisk Fabrik | Novel raloxifene acid addition salts and/or solvates thereof, improved method for purification of said raloxifene acid addition salts and/or solvates thereof and pharmaceutical compositions comprising these |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4133814A (en) * | 1975-10-28 | 1979-01-09 | Eli Lilly And Company | 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents |
| US4380635A (en) * | 1981-04-03 | 1983-04-19 | Eli Lilly And Company | Synthesis of acylated benzothiophenes |
| US4418068A (en) * | 1981-04-03 | 1983-11-29 | Eli Lilly And Company | Antiestrogenic and antiandrugenic benzothiophenes |
-
1994
- 1994-06-10 US US08/258,641 patent/US5420349A/en not_active Expired - Lifetime
-
1995
- 1995-06-07 CA CA002192096A patent/CA2192096A1/en not_active Abandoned
- 1995-06-07 DE DE69513022T patent/DE69513022T2/de not_active Expired - Fee Related
- 1995-06-07 DK DK95923804T patent/DK0764150T3/da active
- 1995-06-07 AU AU28236/95A patent/AU2823695A/en not_active Abandoned
- 1995-06-07 JP JP8502366A patent/JPH10503175A/ja not_active Ceased
- 1995-06-07 HU HU9802648A patent/HU217822B/hu not_active IP Right Cessation
- 1995-06-07 WO PCT/US1995/007399 patent/WO1995034536A1/en active IP Right Grant
- 1995-06-07 HU HU9603403A patent/HU216272B/hu not_active IP Right Cessation
- 1995-06-07 AT AT95923804T patent/ATE186050T1/de not_active IP Right Cessation
- 1995-06-07 ES ES95923804T patent/ES2139222T3/es not_active Expired - Lifetime
- 1995-06-07 BR BR9507968A patent/BR9507968A/pt not_active Application Discontinuation
- 1995-06-07 HU HU9603404A patent/HU213834B/hu not_active IP Right Cessation
- 1995-06-07 EP EP95923804A patent/EP0764150B1/en not_active Expired - Lifetime
-
1996
- 1996-12-04 FI FI964854A patent/FI964854A0/fi unknown
-
2000
- 2000-01-19 GR GR20000400106T patent/GR3032409T3/el not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| DE69513022D1 (de) | 1999-12-02 |
| FI964854A (fi) | 1996-12-04 |
| EP0764150B1 (en) | 1999-10-27 |
| HUT76525A (en) | 1997-09-29 |
| US5420349A (en) | 1995-05-30 |
| WO1995034536A1 (en) | 1995-12-21 |
| DE69513022T2 (de) | 2000-03-16 |
| HU9603404D0 (en) | 1997-02-28 |
| ES2139222T3 (es) | 2000-02-01 |
| GR3032409T3 (en) | 2000-05-31 |
| HU217822B (hu) | 2000-04-28 |
| HU9603403D0 (en) | 1997-02-28 |
| JPH10503175A (ja) | 1998-03-24 |
| HU216272B (hu) | 1999-05-28 |
| AU2823695A (en) | 1996-01-05 |
| FI964854A0 (fi) | 1996-12-04 |
| HU213834B (en) | 1997-10-28 |
| EP0764150A1 (en) | 1997-03-26 |
| BR9507968A (pt) | 1997-11-18 |
| ATE186050T1 (de) | 1999-11-15 |
| HUT76000A (en) | 1997-06-30 |
| EP0764150A4 (en) | 1997-09-10 |
| CA2192096A1 (en) | 1995-12-21 |
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