BR9507968A - Produção de hidroxitoacetamidas e seu uso na sintese de benzotiofenos - Google Patents
Produção de hidroxitoacetamidas e seu uso na sintese de benzotiofenosInfo
- Publication number
- BR9507968A BR9507968A BR9507968A BR9507968A BR9507968A BR 9507968 A BR9507968 A BR 9507968A BR 9507968 A BR9507968 A BR 9507968A BR 9507968 A BR9507968 A BR 9507968A BR 9507968 A BR9507968 A BR 9507968A
- Authority
- BR
- Brazil
- Prior art keywords
- benzo
- beta
- hydroxy
- thiophene
- alpha
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/56—Radicals substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C327/00—Thiocarboxylic acids
- C07C327/38—Amides of thiocarboxylic acids
- C07C327/40—Amides of thiocarboxylic acids having carbon atoms of thiocarboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C327/44—Amides of thiocarboxylic acids having carbon atoms of thiocarboxamide groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/66—Nitrogen atoms not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Investigating Or Analyzing Non-Biological Materials By The Use Of Chemical Means (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/258,641 US5420349A (en) | 1994-06-10 | 1994-06-10 | 2-amino-3-aroyl-benzo[β]thiophenes and methods for preparing and using same to produce 6-hydroxy-2-(4-hydroxyphenyl)-3-]benzo[4-(2-aminoethoxy)-benzoyl[β]thiophenes |
| PCT/US1995/007399 WO1995034536A1 (en) | 1994-06-10 | 1995-06-07 | Production of hydroxythioacetamides and use thereof in the synthesis of benzothiophenes |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9507968A true BR9507968A (pt) | 1997-11-18 |
Family
ID=22981480
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9507968A BR9507968A (pt) | 1994-06-10 | 1995-06-07 | Produção de hidroxitoacetamidas e seu uso na sintese de benzotiofenos |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US5420349A (pt) |
| EP (1) | EP0764150B1 (pt) |
| JP (1) | JPH10503175A (pt) |
| AT (1) | ATE186050T1 (pt) |
| AU (1) | AU2823695A (pt) |
| BR (1) | BR9507968A (pt) |
| CA (1) | CA2192096A1 (pt) |
| DE (1) | DE69513022T2 (pt) |
| DK (1) | DK0764150T3 (pt) |
| ES (1) | ES2139222T3 (pt) |
| FI (1) | FI964854A (pt) |
| GR (1) | GR3032409T3 (pt) |
| HU (3) | HU216272B (pt) |
| WO (1) | WO1995034536A1 (pt) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5466810A (en) * | 1994-06-10 | 1995-11-14 | Eli Lilly And Company | 2-amino-3-aroyl-benzo[β]thiophenes and methods for preparing and using same to produce 6-hydroxy-2-(4-hydroxyphenyl)-3-[4-(2-aminoethoxy)-benzoyl]benzo[β]thiophenes |
| CA2214196A1 (en) * | 1996-09-26 | 1998-03-26 | Eli Lilly And Company | Benzo[b]indeno[2,1-d]thiophene compounds, intermediates, processes, compositions and methods |
| CN1252717A (zh) * | 1997-04-30 | 2000-05-10 | 伊莱利利公司 | 制备苯并[b]噻吩的中间体和方法 |
| EP1832582A1 (en) | 2002-09-30 | 2007-09-12 | A/S GEA Farmaceutisk Fabrik | Novel raloxifene malonic acid addition salts and/or solvates thereof, and pharmaceutical compositions comprising these |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4133814A (en) * | 1975-10-28 | 1979-01-09 | Eli Lilly And Company | 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents |
| US4380635A (en) * | 1981-04-03 | 1983-04-19 | Eli Lilly And Company | Synthesis of acylated benzothiophenes |
| US4418068A (en) * | 1981-04-03 | 1983-11-29 | Eli Lilly And Company | Antiestrogenic and antiandrugenic benzothiophenes |
-
1994
- 1994-06-10 US US08/258,641 patent/US5420349A/en not_active Expired - Lifetime
-
1995
- 1995-06-07 HU HU9603403A patent/HU216272B/hu not_active IP Right Cessation
- 1995-06-07 ES ES95923804T patent/ES2139222T3/es not_active Expired - Lifetime
- 1995-06-07 JP JP8502366A patent/JPH10503175A/ja not_active Ceased
- 1995-06-07 BR BR9507968A patent/BR9507968A/pt not_active Application Discontinuation
- 1995-06-07 DE DE69513022T patent/DE69513022T2/de not_active Expired - Fee Related
- 1995-06-07 WO PCT/US1995/007399 patent/WO1995034536A1/en active IP Right Grant
- 1995-06-07 CA CA002192096A patent/CA2192096A1/en not_active Abandoned
- 1995-06-07 AT AT95923804T patent/ATE186050T1/de not_active IP Right Cessation
- 1995-06-07 HU HU9603404A patent/HU213834B/hu not_active IP Right Cessation
- 1995-06-07 AU AU28236/95A patent/AU2823695A/en not_active Abandoned
- 1995-06-07 HU HU9802648A patent/HU217822B/hu not_active IP Right Cessation
- 1995-06-07 EP EP95923804A patent/EP0764150B1/en not_active Expired - Lifetime
- 1995-06-07 DK DK95923804T patent/DK0764150T3/da active
-
1996
- 1996-12-04 FI FI964854A patent/FI964854A/fi unknown
-
2000
- 2000-01-19 GR GR20000400106T patent/GR3032409T3/el not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| US5420349A (en) | 1995-05-30 |
| JPH10503175A (ja) | 1998-03-24 |
| EP0764150A1 (en) | 1997-03-26 |
| DE69513022D1 (de) | 1999-12-02 |
| DE69513022T2 (de) | 2000-03-16 |
| GR3032409T3 (en) | 2000-05-31 |
| HU216272B (hu) | 1999-05-28 |
| WO1995034536A1 (en) | 1995-12-21 |
| DK0764150T3 (da) | 1999-11-08 |
| ATE186050T1 (de) | 1999-11-15 |
| HU9603403D0 (en) | 1997-02-28 |
| HUT76525A (en) | 1997-09-29 |
| HU9603404D0 (en) | 1997-02-28 |
| HU217822B (hu) | 2000-04-28 |
| EP0764150A4 (en) | 1997-09-10 |
| CA2192096A1 (en) | 1995-12-21 |
| AU2823695A (en) | 1996-01-05 |
| FI964854A0 (fi) | 1996-12-04 |
| FI964854A (fi) | 1996-12-04 |
| HUT76000A (en) | 1997-06-30 |
| HU213834B (en) | 1997-10-28 |
| ES2139222T3 (es) | 2000-02-01 |
| EP0764150B1 (en) | 1999-10-27 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| FI964914A (fi) | 2-amino-3-aroyylibentso/beta/tiofeenejä ja menetelmä niiden valmistamiseksi | |
| SE9503213L (sv) | Syntes av 3-4-(2-aminoetoxi)bensoyl -2aryl-4-hydroxi-benso(b)tiofener | |
| RO81451A (ro) | Procedeu de preparare a unor derivati de benzo(d)-izotiazol-1,1-dioxid | |
| BR9507968A (pt) | Produção de hidroxitoacetamidas e seu uso na sintese de benzotiofenos | |
| GB2211407B (en) | 4h-benz[4,5]cyclohepta[1,2-b]thiophene derivatives as il-1 inhibitors | |
| NO174345C (no) | Analogifremgangsmåte for fremstilling av terapeutisk aktive indol-, benzofuran- og benzotiofenderivater | |
| MX9606177A (es) | 2-AMINO-3-AROIL-BENZO[ beta]TIOFENOS Y METODOS PARA PREPARAR Y USAR LOS MISMOS PARA PRODUCIR 6-HIDROXI-2-(4-HIDROXIFENIL)3-[4-(2-AMINOETOXI)-BENZOIL]BENZO[ beta]TIOFENOS | |
| MXPA99010090A (es) | Procedimiento mejorado para preparar 3(4-aminoetoxibenzoil) benzo[b]tiofenos. | |
| MX9606140A (es) | 2-AMINO-3-AROIL-BENZO[ beta]TIOFENOS Y METODO PARA LA ELABORACION DE LOS MISMOS. | |
| FI20001722A0 (fi) | 6-hydroksi-3-(4-/2-(piperidin-1-yyli)etoksi/fenoksi)-2-(4-metoksifenyyli)bentso/b/tiofeenihydrokloridin uusi kiteinen muoto | |
| WO1995034536B1 (en) | Production of hydroxythioacetamides and use thereof in the synthesis of benzothiophenes | |
| NO822225L (no) | Fremgangsmaate ved fremstilling av 2-(2-thienyl)- og 2-(3-thienyl)-ethylaminderivater | |
| PT81721A (en) | Process for preparing 2-azolylmethyl-3-difluorobenzyloxy-2,3-dihydrofluorobenzo<b>thiophenes and pharmaceutical compositions containing them | |
| EP0878474A3 (en) | Intermediates and a process for preparing benzo[b]thiophenes | |
| ZA867610B (en) | Thiophene ring-substituted alpha-(alkylaminopropionyl)-thiophene derivatives,a process for preparing them and pharmaceutical composition containing them |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EG | Technical examination (opinion): publication of technical examination (opinion) | ||
| FC | Decision: refusal | ||
| HO | Change of classification |
Free format text: C07C327/44; C07D333/66; C07D401/10; C07D403/10 |