BR9507968A - Produção de hidroxitoacetamidas e seu uso na sintese de benzotiofenos - Google Patents
Produção de hidroxitoacetamidas e seu uso na sintese de benzotiofenosInfo
- Publication number
- BR9507968A BR9507968A BR9507968A BR9507968A BR9507968A BR 9507968 A BR9507968 A BR 9507968A BR 9507968 A BR9507968 A BR 9507968A BR 9507968 A BR9507968 A BR 9507968A BR 9507968 A BR9507968 A BR 9507968A
- Authority
- BR
- Brazil
- Prior art keywords
- benzo
- beta
- hydroxy
- thiophene
- alpha
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/56—Radicals substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C327/00—Thiocarboxylic acids
- C07C327/38—Amides of thiocarboxylic acids
- C07C327/40—Amides of thiocarboxylic acids having carbon atoms of thiocarboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C327/44—Amides of thiocarboxylic acids having carbon atoms of thiocarboxamide groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/66—Nitrogen atoms not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Investigating Or Analyzing Non-Biological Materials By The Use Of Chemical Means (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/258,641 US5420349A (en) | 1994-06-10 | 1994-06-10 | 2-amino-3-aroyl-benzo[β]thiophenes and methods for preparing and using same to produce 6-hydroxy-2-(4-hydroxyphenyl)-3-]benzo[4-(2-aminoethoxy)-benzoyl[β]thiophenes |
| PCT/US1995/007399 WO1995034536A1 (en) | 1994-06-10 | 1995-06-07 | Production of hydroxythioacetamides and use thereof in the synthesis of benzothiophenes |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9507968A true BR9507968A (pt) | 1997-11-18 |
Family
ID=22981480
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9507968A BR9507968A (pt) | 1994-06-10 | 1995-06-07 | Produção de hidroxitoacetamidas e seu uso na sintese de benzotiofenos |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US5420349A (pt) |
| EP (1) | EP0764150B1 (pt) |
| JP (1) | JPH10503175A (pt) |
| AT (1) | ATE186050T1 (pt) |
| AU (1) | AU2823695A (pt) |
| BR (1) | BR9507968A (pt) |
| CA (1) | CA2192096A1 (pt) |
| DE (1) | DE69513022T2 (pt) |
| DK (1) | DK0764150T3 (pt) |
| ES (1) | ES2139222T3 (pt) |
| FI (1) | FI964854A (pt) |
| GR (1) | GR3032409T3 (pt) |
| HU (3) | HU213834B (pt) |
| WO (1) | WO1995034536A1 (pt) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5466810A (en) * | 1994-06-10 | 1995-11-14 | Eli Lilly And Company | 2-amino-3-aroyl-benzo[β]thiophenes and methods for preparing and using same to produce 6-hydroxy-2-(4-hydroxyphenyl)-3-[4-(2-aminoethoxy)-benzoyl]benzo[β]thiophenes |
| CA2214196A1 (en) * | 1996-09-26 | 1998-03-26 | Eli Lilly And Company | Benzo[b]indeno[2,1-d]thiophene compounds, intermediates, processes, compositions and methods |
| JP2001524114A (ja) * | 1997-04-30 | 2001-11-27 | イーライ・リリー・アンド・カンパニー | ベンゾ［ｂ］チオフェン類の製造における中間体および方法 |
| AU2003266940B2 (en) | 2002-09-30 | 2007-02-08 | A/S Gea Farmaceutisk Fabrik | Novel raloxifene acid addition salts and/or solvates thereof, improved method for purification of said raloxifene acid addition salts and/or solvates thereof and pharmaceutical compositions comprising these |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4133814A (en) * | 1975-10-28 | 1979-01-09 | Eli Lilly And Company | 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents |
| US4418068A (en) * | 1981-04-03 | 1983-11-29 | Eli Lilly And Company | Antiestrogenic and antiandrugenic benzothiophenes |
| US4380635A (en) * | 1981-04-03 | 1983-04-19 | Eli Lilly And Company | Synthesis of acylated benzothiophenes |
-
1994
- 1994-06-10 US US08/258,641 patent/US5420349A/en not_active Expired - Lifetime
-
1995
- 1995-06-07 JP JP8502366A patent/JPH10503175A/ja not_active Ceased
- 1995-06-07 EP EP95923804A patent/EP0764150B1/en not_active Expired - Lifetime
- 1995-06-07 AU AU28236/95A patent/AU2823695A/en not_active Abandoned
- 1995-06-07 HU HU9603404A patent/HU213834B/hu not_active IP Right Cessation
- 1995-06-07 CA CA002192096A patent/CA2192096A1/en not_active Abandoned
- 1995-06-07 DE DE69513022T patent/DE69513022T2/de not_active Expired - Fee Related
- 1995-06-07 HU HU9802648A patent/HU217822B/hu not_active IP Right Cessation
- 1995-06-07 HU HU9603403A patent/HU216272B/hu not_active IP Right Cessation
- 1995-06-07 ES ES95923804T patent/ES2139222T3/es not_active Expired - Lifetime
- 1995-06-07 WO PCT/US1995/007399 patent/WO1995034536A1/en active IP Right Grant
- 1995-06-07 AT AT95923804T patent/ATE186050T1/de not_active IP Right Cessation
- 1995-06-07 DK DK95923804T patent/DK0764150T3/da active
- 1995-06-07 BR BR9507968A patent/BR9507968A/pt not_active Application Discontinuation
-
1996
- 1996-12-04 FI FI964854A patent/FI964854A/fi unknown
-
2000
- 2000-01-19 GR GR20000400106T patent/GR3032409T3/el not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| FI964854A0 (fi) | 1996-12-04 |
| HU216272B (hu) | 1999-05-28 |
| JPH10503175A (ja) | 1998-03-24 |
| EP0764150A1 (en) | 1997-03-26 |
| AU2823695A (en) | 1996-01-05 |
| HU213834B (en) | 1997-10-28 |
| FI964854A (fi) | 1996-12-04 |
| DE69513022T2 (de) | 2000-03-16 |
| CA2192096A1 (en) | 1995-12-21 |
| DE69513022D1 (de) | 1999-12-02 |
| EP0764150A4 (en) | 1997-09-10 |
| ES2139222T3 (es) | 2000-02-01 |
| GR3032409T3 (en) | 2000-05-31 |
| US5420349A (en) | 1995-05-30 |
| WO1995034536A1 (en) | 1995-12-21 |
| HU217822B (hu) | 2000-04-28 |
| DK0764150T3 (da) | 1999-11-08 |
| HU9603403D0 (en) | 1997-02-28 |
| HUT76000A (en) | 1997-06-30 |
| HUT76525A (en) | 1997-09-29 |
| EP0764150B1 (en) | 1999-10-27 |
| ATE186050T1 (de) | 1999-11-15 |
| HU9603404D0 (en) | 1997-02-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EG | Technical examination (opinion): publication of technical examination (opinion) | ||
| FC | Decision: refusal | ||
| HO | Change of classification |
Free format text: C07C327/44; C07D333/66; C07D401/10; C07D403/10 |