DK0574312T3 - Diacylglycerolnicotinater, fremgangsmåde til fremstilling heraf og farmaceutiske midler, som indeholder dem - Google Patents

Diacylglycerolnicotinater, fremgangsmåde til fremstilling heraf og farmaceutiske midler, som indeholder dem

Info

Publication number
DK0574312T3
DK0574312T3 DK93401475.4T DK93401475T DK0574312T3 DK 0574312 T3 DK0574312 T3 DK 0574312T3 DK 93401475 T DK93401475 T DK 93401475T DK 0574312 T3 DK0574312 T3 DK 0574312T3
Authority
DK
Denmark
Prior art keywords
nicotinates
diacylglycerol
processes
preparation
pharmaceutical agents
Prior art date
Application number
DK93401475.4T
Other languages
Danish (da)
English (en)
Inventor
Jean-Michel Lacoste
Jacques Duhault
Alex Cordi
Joseph Espinal
Michelle Boulanger
Original Assignee
Adir
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adir filed Critical Adir
Application granted granted Critical
Publication of DK0574312T3 publication Critical patent/DK0574312T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79Acids; Esters
    • C07D213/80Acids; Esters in position 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Vascular Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
DK93401475.4T 1992-06-10 1993-06-10 Diacylglycerolnicotinater, fremgangsmåde til fremstilling heraf og farmaceutiske midler, som indeholder dem DK0574312T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR929206951A FR2692262B1 (fr) 1992-06-10 1992-06-10 Nouveaux nicotinates de diacylglycerols, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.

Publications (1)

Publication Number Publication Date
DK0574312T3 true DK0574312T3 (da) 1995-04-10

Family

ID=9430554

Family Applications (1)

Application Number Title Priority Date Filing Date
DK93401475.4T DK0574312T3 (da) 1992-06-10 1993-06-10 Diacylglycerolnicotinater, fremgangsmåde til fremstilling heraf og farmaceutiske midler, som indeholder dem

Country Status (12)

Country Link
US (1) US5385920A (fr)
EP (1) EP0574312B1 (fr)
JP (1) JPH07103106B2 (fr)
AT (1) ATE112267T1 (fr)
AU (1) AU657222B2 (fr)
CA (1) CA2098069A1 (fr)
DE (1) DE69300011T2 (fr)
DK (1) DK0574312T3 (fr)
ES (1) ES2065192T3 (fr)
FR (1) FR2692262B1 (fr)
NZ (1) NZ247820A (fr)
ZA (1) ZA934110B (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2220091C (fr) * 1995-05-01 2011-01-04 Scotia Holdings Plc Esters d'acide nicotinique et compositions pharmaceutiques contenant de tels esters
USRE40546E1 (en) * 1996-05-01 2008-10-21 Scarista, Ltd. 1,3-Propane diol esters and ethers and methods for their use in drug delivery
MY118354A (en) * 1995-05-01 2004-10-30 Scarista Ltd 1,3-propane diol derivatives as bioactive compounds
WO2004101524A1 (fr) * 2003-05-19 2004-11-25 Lonza Ag Esters polyglyceroliques d'acides pyridinecarboxyliques
CN112955115B (zh) * 2018-11-02 2023-06-30 联合利华知识产权控股有限公司 生物能烟酸甘油酯、组合物和使用其的方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES8101585A1 (es) * 1980-02-15 1980-12-16 Especialidades Farmaco Terape Procedimiento de obtencion de un nuevo compuesto antiateros-clerotico

Also Published As

Publication number Publication date
AU657222B2 (en) 1995-03-02
DE69300011D1 (de) 1994-11-03
AU4012393A (en) 1993-12-16
CA2098069A1 (fr) 1993-12-10
EP0574312B1 (fr) 1994-09-28
DE69300011T2 (de) 1995-05-11
FR2692262A1 (fr) 1993-12-17
NZ247820A (en) 1994-10-26
ZA934110B (en) 1994-01-07
ATE112267T1 (de) 1994-10-15
FR2692262B1 (fr) 1994-08-05
EP0574312A1 (fr) 1993-12-15
JPH07103106B2 (ja) 1995-11-08
ES2065192T3 (es) 1995-02-01
JPH0656786A (ja) 1994-03-01
US5385920A (en) 1995-01-31

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