DE69106323T2 - Imidazol-Derivate, Verfahren zu deren Herstellung und diese enthaltende Zusammenstellungen. - Google Patents
Imidazol-Derivate, Verfahren zu deren Herstellung und diese enthaltende Zusammenstellungen.Info
- Publication number
- DE69106323T2 DE69106323T2 DE69106323T DE69106323T DE69106323T2 DE 69106323 T2 DE69106323 T2 DE 69106323T2 DE 69106323 T DE69106323 T DE 69106323T DE 69106323 T DE69106323 T DE 69106323T DE 69106323 T2 DE69106323 T2 DE 69106323T2
- Authority
- DE
- Germany
- Prior art keywords
- group
- branched
- linear
- processes
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/004—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reaction with organometalhalides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/45—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/04—Saturated compounds containing keto groups bound to acyclic carbon atoms
- C07C49/16—Saturated compounds containing keto groups bound to acyclic carbon atoms containing halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/04—Saturated compounds containing keto groups bound to acyclic carbon atoms
- C07C49/16—Saturated compounds containing keto groups bound to acyclic carbon atoms containing halogen
- C07C49/163—Saturated compounds containing keto groups bound to acyclic carbon atoms containing halogen containing rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/20—Unsaturated compounds containing keto groups bound to acyclic carbon atoms
- C07C49/213—Unsaturated compounds containing keto groups bound to acyclic carbon atoms containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/20—Unsaturated compounds containing keto groups bound to acyclic carbon atoms
- C07C49/213—Unsaturated compounds containing keto groups bound to acyclic carbon atoms containing six-membered aromatic rings
- C07C49/215—Unsaturated compounds containing keto groups bound to acyclic carbon atoms containing six-membered aromatic rings polycyclic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/29—Saturated compounds containing keto groups bound to rings
- C07C49/327—Saturated compounds containing keto groups bound to rings containing halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C53/00—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
- C07C53/38—Acyl halides
- C07C53/46—Acyl halides containing halogen outside the carbonyl halide group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
- C07C57/64—Acyl halides
- C07C57/76—Acyl halides containing halogen outside the carbonyl halide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9014086A FR2669030B1 (fr) | 1990-11-14 | 1990-11-14 | Nouveaux derives d'imidazole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
Publications (2)
Publication Number | Publication Date |
---|---|
DE69106323D1 DE69106323D1 (de) | 1995-02-09 |
DE69106323T2 true DE69106323T2 (de) | 1995-06-22 |
Family
ID=9402134
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69106323T Expired - Fee Related DE69106323T2 (de) | 1990-11-14 | 1991-11-14 | Imidazol-Derivate, Verfahren zu deren Herstellung und diese enthaltende Zusammenstellungen. |
Country Status (15)
Country | Link |
---|---|
US (1) | US5173502A (de) |
EP (1) | EP0486385B1 (de) |
JP (1) | JPH0710851B2 (de) |
AT (1) | ATE116304T1 (de) |
AU (1) | AU639154B2 (de) |
CA (1) | CA2055325A1 (de) |
DE (1) | DE69106323T2 (de) |
DK (1) | DK0486385T3 (de) |
ES (1) | ES2069249T3 (de) |
FR (1) | FR2669030B1 (de) |
GR (1) | GR3015209T3 (de) |
IE (1) | IE66161B1 (de) |
NZ (1) | NZ240578A (de) |
PT (1) | PT99502B (de) |
ZA (1) | ZA918991B (de) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2698789B1 (fr) * | 1992-12-07 | 1995-03-03 | Pf Medicament | Utilisation de l'idazoxan et ses dérivés pour la préparation d'un médicament destiné au traitement de la maladie de Parkinson et de son évolution. |
FR2706303B1 (fr) * | 1993-06-18 | 1995-09-08 | Pf Medicament | Utilisation de l'Efaroxan et de ses dérivés pour la préparation d'un médicament destiné au traitement de la maladie de Parkinson. |
FR2707166B1 (fr) * | 1993-07-09 | 1995-09-29 | Pf Medicament | Utilisation de l'efaroxan et de ses dérivés pour la fabrication de médicaments destinés au traitement de maladies neurodégénératives et leur progression . |
US6448282B1 (en) | 1995-05-30 | 2002-09-10 | Gliatech, Inc. | 1H-4(5)-substituted imidazole derivatives |
ES2170859T3 (es) * | 1995-05-30 | 2002-08-16 | Gliatech Inc | Derivados de imidazol 1h-4(5)-sustituidos. |
KR100432577B1 (ko) * | 2002-02-08 | 2004-05-24 | 주식회사유한양행 | 이미다졸 유도체의 제조방법 |
US8188126B2 (en) * | 2002-05-16 | 2012-05-29 | Pierre Fabre Medicament | Imidazolic compounds and use thereof as alpha-2 adrenergic receptors |
US20080146523A1 (en) * | 2006-12-18 | 2008-06-19 | Guido Galley | Imidazole derivatives |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4497818A (en) * | 1980-09-10 | 1985-02-05 | Syntex (U.S.A.) Inc. | 2-(1,4-Benzodioxan-2-ylalkyl)imidazoles useful as antihypertensives and platelet aggregation inhibitors |
US4576958A (en) * | 1984-01-23 | 1986-03-18 | E. I. Du Pont De Nemours And Company | Antihypertensive 4,5-diaryl-1H-imidazole-2-methanol derivatives |
FI81092C (fi) * | 1986-05-15 | 1990-09-10 | Farmos Oy | Foerfarande foer framstaellning av terapeutiskt aktiva 4(5)-(2,3-dihydro-1h-inden-2-yl)-imidazolderivat. |
JPH02115145A (ja) * | 1988-10-26 | 1990-04-27 | Canon Inc | 液晶性化合物、それを含有する液晶組成物および液晶素子 |
-
1990
- 1990-11-14 FR FR9014086A patent/FR2669030B1/fr not_active Expired - Lifetime
-
1991
- 1991-11-01 US US07/786,280 patent/US5173502A/en not_active Expired - Fee Related
- 1991-11-13 NZ NZ240578A patent/NZ240578A/en unknown
- 1991-11-13 CA CA002055325A patent/CA2055325A1/fr not_active Abandoned
- 1991-11-13 AU AU87779/91A patent/AU639154B2/en not_active Ceased
- 1991-11-13 PT PT99502A patent/PT99502B/pt not_active IP Right Cessation
- 1991-11-13 ZA ZA918991A patent/ZA918991B/xx unknown
- 1991-11-14 IE IE396491A patent/IE66161B1/en not_active IP Right Cessation
- 1991-11-14 JP JP3299225A patent/JPH0710851B2/ja not_active Expired - Lifetime
- 1991-11-14 AT AT91403043T patent/ATE116304T1/de not_active IP Right Cessation
- 1991-11-14 DK DK91403043.2T patent/DK0486385T3/da active
- 1991-11-14 DE DE69106323T patent/DE69106323T2/de not_active Expired - Fee Related
- 1991-11-14 ES ES91403043T patent/ES2069249T3/es not_active Expired - Lifetime
- 1991-11-14 EP EP91403043A patent/EP0486385B1/de not_active Expired - Lifetime
-
1995
- 1995-02-28 GR GR950400413T patent/GR3015209T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
PT99502A (pt) | 1992-09-30 |
EP0486385B1 (de) | 1994-12-28 |
IE66161B1 (en) | 1995-12-13 |
JPH04266875A (ja) | 1992-09-22 |
ES2069249T3 (es) | 1995-05-01 |
PT99502B (pt) | 1999-04-30 |
EP0486385A1 (de) | 1992-05-20 |
ZA918991B (en) | 1992-08-26 |
DK0486385T3 (da) | 1995-06-12 |
DE69106323D1 (de) | 1995-02-09 |
CA2055325A1 (fr) | 1992-05-15 |
FR2669030B1 (fr) | 1992-12-31 |
IE913964A1 (en) | 1992-05-20 |
ATE116304T1 (de) | 1995-01-15 |
JPH0710851B2 (ja) | 1995-02-08 |
NZ240578A (en) | 1992-12-23 |
GR3015209T3 (en) | 1995-05-31 |
FR2669030A1 (fr) | 1992-05-15 |
AU8777991A (en) | 1992-05-21 |
AU639154B2 (en) | 1993-07-15 |
US5173502A (en) | 1992-12-22 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee | ||
8370 | Indication related to discontinuation of the patent is to be deleted | ||
8339 | Ceased/non-payment of the annual fee |