DE60336504D1 - 4-hydroxypiperidin-derivate zur verwendung als antimycobakterielle mittel - Google Patents
4-hydroxypiperidin-derivate zur verwendung als antimycobakterielle mittelInfo
- Publication number
- DE60336504D1 DE60336504D1 DE60336504T DE60336504T DE60336504D1 DE 60336504 D1 DE60336504 D1 DE 60336504D1 DE 60336504 T DE60336504 T DE 60336504T DE 60336504 T DE60336504 T DE 60336504T DE 60336504 D1 DE60336504 D1 DE 60336504D1
- Authority
- DE
- Germany
- Prior art keywords
- hydroxypiperidin
- derivatives
- antimycobacterial agents
- compositions
- methods
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
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- C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
- C07C323/24—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
- C07C323/25—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/132—Amines having two or more amino groups, e.g. spermidine, putrescine
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- A61K31/133—Amines having hydroxy groups, e.g. sphingosine
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
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- C07C211/41—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton containing condensed ring systems
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- C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
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- C07C215/06—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/36—Systems containing two condensed rings the rings having more than two atoms in common
- C07C2602/42—Systems containing two condensed rings the rings having more than two atoms in common the bicyclo ring system containing seven carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2603/00—Systems containing at least three condensed rings
- C07C2603/56—Ring systems containing bridged rings
- C07C2603/58—Ring systems containing bridged rings containing three rings
- C07C2603/70—Ring systems containing bridged rings containing three rings containing only six-membered rings
- C07C2603/74—Adamantanes
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US38124402P | 2002-05-17 | 2002-05-17 | |
US10/147,587 US6951961B2 (en) | 2002-05-17 | 2002-05-17 | Methods of use and compositions for the diagnosis and treatment of infectious disease |
PCT/US2003/015925 WO2003096987A2 (en) | 2002-05-17 | 2003-05-19 | Methods of use and compositions for the diagnosis and treatment of infectious disease |
Publications (1)
Publication Number | Publication Date |
---|---|
DE60336504D1 true DE60336504D1 (de) | 2011-05-05 |
Family
ID=29552724
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE60336504T Expired - Lifetime DE60336504D1 (de) | 2002-05-17 | 2003-05-19 | 4-hydroxypiperidin-derivate zur verwendung als antimycobakterielle mittel |
Country Status (9)
Country | Link |
---|---|
EP (1) | EP1578353B1 (de) |
JP (1) | JP4563797B2 (de) |
AT (1) | ATE502639T1 (de) |
AU (1) | AU2003228240C1 (de) |
CA (1) | CA2485586A1 (de) |
DE (1) | DE60336504D1 (de) |
EA (1) | EA016659B1 (de) |
SG (1) | SG188670A1 (de) |
WO (1) | WO2003096987A2 (de) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20050159625A1 (en) * | 2004-01-19 | 2005-07-21 | Coates John S. | Alkoxylated amine and process therefor |
EP2061780A4 (de) * | 2006-09-14 | 2010-12-22 | Zalicus Pharmaceuticals Ltd | Diarylpiperidinverbindungen als kalziumkanalblocker |
US9572809B2 (en) | 2012-07-18 | 2017-02-21 | Spero Trinem, Inc. | Combination therapy to treat Mycobacterium diseases |
-
2003
- 2003-05-19 AT AT03726938T patent/ATE502639T1/de not_active IP Right Cessation
- 2003-05-19 JP JP2004504986A patent/JP4563797B2/ja not_active Expired - Fee Related
- 2003-05-19 AU AU2003228240A patent/AU2003228240C1/en not_active Ceased
- 2003-05-19 CA CA002485586A patent/CA2485586A1/en not_active Abandoned
- 2003-05-19 DE DE60336504T patent/DE60336504D1/de not_active Expired - Lifetime
- 2003-05-19 EA EA200401523A patent/EA016659B1/ru not_active IP Right Cessation
- 2003-05-19 EP EP03726938A patent/EP1578353B1/de not_active Expired - Lifetime
- 2003-05-19 SG SG2010009181A patent/SG188670A1/en unknown
- 2003-05-19 WO PCT/US2003/015925 patent/WO2003096987A2/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
JP4563797B2 (ja) | 2010-10-13 |
AU2003228240B2 (en) | 2009-07-16 |
CA2485586A1 (en) | 2003-11-27 |
ATE502639T1 (de) | 2011-04-15 |
AU2003228240A1 (en) | 2003-12-02 |
EA200401523A1 (ru) | 2005-06-30 |
WO2003096987A2 (en) | 2003-11-27 |
EP1578353A4 (de) | 2010-04-07 |
EA016659B1 (ru) | 2012-06-29 |
EP1578353A2 (de) | 2005-09-28 |
JP2006504633A (ja) | 2006-02-09 |
EP1578353B1 (de) | 2011-03-23 |
AU2003228240C1 (en) | 2009-10-22 |
WO2003096987A9 (en) | 2009-11-12 |
SG188670A1 (en) | 2013-04-30 |
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