DE60010344D1 - Diketopiperazinderivate als thrombininhibitoren - Google Patents

Diketopiperazinderivate als thrombininhibitoren

Info

Publication number
DE60010344D1
DE60010344D1 DE60010344T DE60010344T DE60010344D1 DE 60010344 D1 DE60010344 D1 DE 60010344D1 DE 60010344 T DE60010344 T DE 60010344T DE 60010344 T DE60010344 T DE 60010344T DE 60010344 D1 DE60010344 D1 DE 60010344D1
Authority
DE
Germany
Prior art keywords
alkyl
moiety
aryl
hydrogen
hydroheteroaryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE60010344T
Other languages
English (en)
Other versions
DE60010344T2 (de
Inventor
Yudu Cheng
Jeffrey Manwell
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BEST EXPRESS WORLDWIDE Ltd TRU
Original Assignee
BEST EXPRESS WORLDWIDE Ltd TRU
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BEST EXPRESS WORLDWIDE Ltd TRU filed Critical BEST EXPRESS WORLDWIDE Ltd TRU
Publication of DE60010344D1 publication Critical patent/DE60010344D1/de
Application granted granted Critical
Publication of DE60010344T2 publication Critical patent/DE60010344T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DE60010344T 1999-11-30 2000-11-29 Diketopiperazinderivate als thrombininhibitoren Expired - Fee Related DE60010344T2 (de)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US16790199P 1999-11-30 1999-11-30
US167901P 1999-11-30
US19436600P 2000-04-04 2000-04-04
US194366P 2000-04-04
PCT/CA2000/001414 WO2001040224A1 (en) 1999-11-30 2000-11-29 Diketopiperazine derivatives to inhibit thrombin

Publications (2)

Publication Number Publication Date
DE60010344D1 true DE60010344D1 (de) 2004-06-03
DE60010344T2 DE60010344T2 (de) 2005-02-17

Family

ID=26863579

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60010344T Expired - Fee Related DE60010344T2 (de) 1999-11-30 2000-11-29 Diketopiperazinderivate als thrombininhibitoren

Country Status (7)

Country Link
EP (1) EP1261608B1 (de)
CN (1) CN1174982C (de)
AT (1) ATE265453T1 (de)
AU (1) AU1847401A (de)
CA (1) CA2392936A1 (de)
DE (1) DE60010344T2 (de)
WO (1) WO2001040224A1 (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN112010930B (zh) * 2019-05-28 2022-08-02 首都医科大学 Rgd修饰的五环哌嗪二酮及其制备和应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL112627A0 (en) * 1994-02-14 1995-05-26 Xenova Ltd Diketopiperazines, their preparation and pharmaceutical or veterinary compositions containing them

Also Published As

Publication number Publication date
CN1174982C (zh) 2004-11-10
ATE265453T1 (de) 2004-05-15
EP1261608A1 (de) 2002-12-04
WO2001040224A1 (en) 2001-06-07
CN1402725A (zh) 2003-03-12
AU1847401A (en) 2001-06-12
CA2392936A1 (en) 2001-06-07
DE60010344T2 (de) 2005-02-17
EP1261608B1 (de) 2004-04-28

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee