DE3362266D1 - Penicillanic acid dioxide prodrug - Google Patents

Penicillanic acid dioxide prodrug

Info

Publication number
DE3362266D1
DE3362266D1 DE8383302891T DE3362266T DE3362266D1 DE 3362266 D1 DE3362266 D1 DE 3362266D1 DE 8383302891 T DE8383302891 T DE 8383302891T DE 3362266 T DE3362266 T DE 3362266T DE 3362266 D1 DE3362266 D1 DE 3362266D1
Authority
DE
Germany
Prior art keywords
prodrug
penicillanic acid
acid dioxide
dioxide
penicillanic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE8383302891T
Other languages
German (de)
English (en)
Inventor
Robert Fischer Myers
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp Belgium
Pfizer Corp SRL
Original Assignee
Pfizer Corp Belgium
Pfizer Corp SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium, Pfizer Corp SRL filed Critical Pfizer Corp Belgium
Application granted granted Critical
Publication of DE3362266D1 publication Critical patent/DE3362266D1/de
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE8383302891T 1982-05-24 1983-05-20 Penicillanic acid dioxide prodrug Expired DE3362266D1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/381,104 US4428935A (en) 1982-05-24 1982-05-24 Penicillanic acid dioxide prodrug

Publications (1)

Publication Number Publication Date
DE3362266D1 true DE3362266D1 (de) 1986-04-03

Family

ID=23503664

Family Applications (1)

Application Number Title Priority Date Filing Date
DE8383302891T Expired DE3362266D1 (de) 1982-05-24 1983-05-20 Penicillanic acid dioxide prodrug

Country Status (7)

Country Link
US (1) US4428935A (OSRAM)
EP (1) EP0095341B1 (OSRAM)
JP (1) JPS58216191A (OSRAM)
DE (1) DE3362266D1 (OSRAM)
DK (1) DK226983A (OSRAM)
GR (1) GR79260B (OSRAM)
IE (1) IE55577B1 (OSRAM)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4946959A (en) * 1984-11-30 1990-08-07 The Dow Chemical Company Method of preparing 5-alkyl-1-(2-pyridinyl)-1H-1,2,4-triazol-3-ols
US4681943A (en) * 1984-11-30 1987-07-21 The Dow Chemical Company 1-acyl-1-(2-pyridinyl)semicarbazides
US5399678A (en) * 1990-04-13 1995-03-21 Pfizer Inc. Process for sultamicillin intermediate
US7189351B2 (en) * 2001-10-25 2007-03-13 Spherix Incorporated D-tagatose as an anti-biofilm agent
PA8579701A1 (es) * 2002-08-23 2005-05-24 Pfizer Prod Inc Profarmaco inhibidor de beta-lactamasa
EP1636240A1 (en) * 2003-06-05 2006-03-22 Pfizer Products Inc. Beta-lactamase inhibitor prodrug
JP2007534771A (ja) 2004-04-27 2007-11-29 メディシノバ，インコーポレーテッド 炎症性疾患の治療におけるフェノキシアルキルカルボン酸誘導体
JP5324463B2 (ja) 2006-12-10 2013-10-23 チョンシー ユー β−ラクタム抗生物質の経皮送達システム
US9969751B2 (en) 2009-06-10 2018-05-15 Techfields Pharma Co., Ltd. High penetration prodrug compositions of antimicrobials and antimicrobial-related compounds
EP2440523A4 (en) * 2009-06-10 2014-03-19 Chongxi Yu COMPOSITION WITH STRONG PENETRATION OR PRODRUGS FROM ANTIMICROBIA AND COMPOUNDS IN ANTIMICROBIA
PT2445502T (pt) * 2009-06-25 2017-09-22 Alkermes Pharma Ireland Ltd Compostos heterocíclicos para o tratamento de distúrbios neurológicos e psicológicos
WO2010151711A1 (en) 2009-06-25 2010-12-29 Alkermes, Inc. Prodrugs of nh-acidic compounds
US8592427B2 (en) 2010-06-24 2013-11-26 Alkermes Pharma Ireland Limited Prodrugs of NH-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives
HRP20240285T1 (hr) 2011-03-18 2024-05-24 Alkermes Pharma Ireland Limited Farmaceutski pripravci koji sadrže sorbitan estere
CN107261148B (zh) * 2011-07-28 2021-07-13 凯姆制药公司 哌甲酯前药、其制备和使用方法
WO2013088255A1 (en) 2011-12-15 2013-06-20 Alkermes Pharma Ireland Limited Prodrugs of secondary amine compounds
EP2827866B1 (en) 2012-03-19 2023-05-03 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising benzyl alcohol
AU2013235519C1 (en) 2012-03-19 2018-04-26 Alkermes Pharma Ireland Limited Pharmaaceutical compositions comprising fatty acid esters
ES2764383T3 (es) 2012-03-19 2020-06-03 Alkermes Pharma Ireland Ltd Composiciones farmacéuticas que comprenden ésteres de glicerol
ES2792149T3 (es) 2012-09-19 2020-11-10 Alkermes Pharma Ireland Ltd Composiciones farmacéuticas que tienen estabilidad de almacenamiento mejorada
JP6621329B2 (ja) * 2012-10-05 2019-12-18 スファエラ ファーマ ピーティーイー リミテッド 新規化合物、それらの合成及びそれらの使用
MX376057B (es) 2014-03-20 2025-03-07 Alkermes Pharma Ireland Ltd Formulaciones de aripiprazol que tienen mayores velocidades de inyeccion.
AU2019230014B2 (en) 2018-03-05 2024-11-28 Alkermes Pharma Ireland Limited Aripiprazole dosing strategy
EP4578850A3 (en) * 2019-04-17 2025-10-15 Myto Therapeutics, Inc. Prodrugs of monomethyl fumarate

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1255034A (en) * 1968-09-06 1971-11-24 Beecham Group Ltd Penicillin esters
NL7401782A (OSRAM) * 1973-02-14 1974-08-16
JPS6056160B2 (ja) * 1977-06-07 1985-12-09 フアイザ−・インコ−ポレ−テツド β−ラクタマ−ゼ阻害剤としてのペニシラン酸１，１−ジオキシド
US4234579A (en) 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
US4244951A (en) 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
US4376767A (en) * 1981-01-02 1983-03-15 Merck & Co., Inc. Pyridylmethyl esters of selected bio-affecting carboxylic acids
US4323499A (en) 1981-01-05 1982-04-06 Pfizer Inc. 6-(2-Aryl-2-(1,1-dioxopenicillanoyloxy-methoxycarbonyl)acetamido penicillanic acids

Also Published As

Publication number Publication date
DK226983A (da) 1983-11-25
IE831203L (en) 1983-11-24
IE55577B1 (en) 1990-11-07
JPS58216191A (ja) 1983-12-15
EP0095341B1 (en) 1986-02-26
EP0095341A1 (en) 1983-11-30
DK226983D0 (da) 1983-05-20
US4428935A (en) 1984-01-31
GR79260B (OSRAM) 1984-10-22

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8328 Change in the person/name/address of the agent

Free format text: LEDERER, F., DIPL.-CHEM. DR., PAT.-ANW., 8000 MUENCHEN

8339 Ceased/non-payment of the annual fee