DE10360745A1 - Neue Amid-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel - Google Patents

Neue Amid-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel Download PDF

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Publication number
DE10360745A1
DE10360745A1 DE10360745A DE10360745A DE10360745A1 DE 10360745 A1 DE10360745 A1 DE 10360745A1 DE 10360745 A DE10360745 A DE 10360745A DE 10360745 A DE10360745 A DE 10360745A DE 10360745 A1 DE10360745 A1 DE 10360745A1
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Germany
Prior art keywords
alkyl
phenyl
group
amino
chloro
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DE10360745A
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German (de)
English (en)
Inventor
Thorsten Dr. Lehmann-Lintz
Gerald Jürgen Dr. Roth
Philipp Dr. Lustenberger
Dirk Dr. Stenkamp
Stephan Georg Dr. Mueller
Klaus Dr. Rudolf
Marcus Dr. Schindler
Leo Dr. Thomas
Ralf R. H. Dr. Lotz
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
Boehringer Ingelheim Pharmaceuticals Inc
Original Assignee
Boehringer Ingelheim Pharma GmbH and Co KG
Boehringer Ingelheim Pharmaceuticals Inc
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34706476&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE10360745(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority to DE10360745A priority Critical patent/DE10360745A1/de
Application filed by Boehringer Ingelheim Pharma GmbH and Co KG, Boehringer Ingelheim Pharmaceuticals Inc filed Critical Boehringer Ingelheim Pharma GmbH and Co KG
Priority to EP04803987A priority patent/EP1708698A1/de
Priority to JP2006546009A priority patent/JP2007520466A/ja
Priority to PCT/EP2004/014378 priority patent/WO2005063239A1/de
Priority to CA002550649A priority patent/CA2550649A1/en
Priority to UY28689A priority patent/UY28689A1/es
Priority to TW093140144A priority patent/TW200530180A/zh
Priority to ARP040104840A priority patent/AR048019A1/es
Priority to US11/021,897 priority patent/US7592373B2/en
Priority to PE2005000007A priority patent/PE20050678A1/es
Publication of DE10360745A1 publication Critical patent/DE10360745A1/de
Withdrawn legal-status Critical Current

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DE10360745A 2003-12-23 2003-12-23 Neue Amid-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel Withdrawn DE10360745A1 (de)

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DE10360745A DE10360745A1 (de) 2003-12-23 2003-12-23 Neue Amid-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel
EP04803987A EP1708698A1 (de) 2003-12-23 2004-12-17 3-(4-piperidin-1ylmethyl-phenyl)-propionsäure-phenylamid-derivate und verwandte verbindungen als mch (melanine concentrating hormone) antagonsiten zur behandlung von essstörungen
JP2006546009A JP2007520466A (ja) 2003-12-23 2004-12-17 摂食障害を治療するためのｍｃｈアンタゴニスト（メラニン含有ホルモン）の形態で使用される３−（４−ピペリジン−１−イルメチル−フェニル）−プロピオン酸−フェニルアミド誘導体及び関連化合物
PCT/EP2004/014378 WO2005063239A1 (de) 2003-12-23 2004-12-17 3-(4-piperidin-1ylmethyl-phenyl) -propionsäure-phrnylamid-derivate und verwandte verbindungen als mch (melanine concentrating hormone) antagonisten zur behandlung von essstörungen
CA002550649A CA2550649A1 (en) 2003-12-23 2004-12-17 3-(4-piperidine-1ylmethyl-phenyl)-propion acid-phenylamide-derivatives and related compounds used in the form of mch antagonists (melanine concentrating hormone) for treating eating disorders
UY28689A UY28689A1 (es) 2003-12-23 2004-12-20 Nuevos compuestos amida con actividad antagonista de mch y medicamentos que contienen estos compuestos.
ARP040104840A AR048019A1 (es) 2003-12-23 2004-12-22 Derivados de amida con actividad antagonista de mch y composiciones farmaceuticas que los contienen
TW093140144A TW200530180A (en) 2003-12-23 2004-12-22 New amide compounds with MCH antagonistic activity and medicaments comprising these compounds
US11/021,897 US7592373B2 (en) 2003-12-23 2004-12-23 Amide compounds with MCH antagonistic activity and medicaments comprising these compounds
PE2005000007A PE20050678A1 (es) 2003-12-23 2005-01-03 Nuevos compuestos amida con actividad antagonista de mch y medicamentos que contiene estos compuestos

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US7351719B2 (en) 2002-10-31 2008-04-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg Amide compounds having MCH-antagonistic activity and medicaments comprising these compounds
US7605176B2 (en) 2004-03-06 2009-10-20 Boehringer Ingelheim International Gmbh β-ketoamide compounds with MCH antagonistic activity
EP1863756A1 (en) * 2005-03-24 2007-12-12 Janssen Pharmaceutica N.V. Biaryl derived amide modulators of vanilloid vr1 receptor
CN101296906A (zh) * 2005-10-26 2008-10-29 贝林格尔·英格海姆国际有限公司 具有mch拮抗活性的(杂)芳基化合物及包含这些化合物的药物
US7977346B2 (en) * 2006-01-17 2011-07-12 Guoqing Paul Chen Spiro compounds and methods of use
NZ575520A (en) 2006-08-25 2012-03-30 Boehringer Ingelheim Int New pyridone derivatives with mch antagonistic activity and medicaments comprising these compounds
TW200831485A (en) 2006-12-11 2008-08-01 Boehringer Ingelheim Int New pyridazine derivatives with MCH antagonistic activity and medicaments comprising these compounds
JP5722892B2 (ja) 2010-07-15 2015-05-27 武田薬品工業株式会社 複素環化合物
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AR048019A1 (es) 2006-03-22
WO2005063239A1 (de) 2005-07-14
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