DD116830A5 - - Google Patents

Info

Publication number
DD116830A5
DD116830A5 DD181858A DD18185874A DD116830A5 DD 116830 A5 DD116830 A5 DD 116830A5 DD 181858 A DD181858 A DD 181858A DD 18185874 A DD18185874 A DD 18185874A DD 116830 A5 DD116830 A5 DD 116830A5
Authority
DD
German Democratic Republic
Application number
DD181858A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of DD116830A5 publication Critical patent/DD116830A5/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D263/57Aryl or substituted aryl radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • C07C45/46Friedel-Crafts reactions
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Rheumatology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DD181858A 1973-10-23 1974-10-23 DD116830A5 (US06168776-20010102-C00041.png)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB49259/73A GB1488003A (en) 1973-10-23 1973-10-23 1,2-benzisoxazole derivatives processes for their preparation and their use as pharmaceuticals

Publications (1)

Publication Number Publication Date
DD116830A5 true DD116830A5 (US06168776-20010102-C00041.png) 1975-12-12

Family

ID=10451720

Family Applications (1)

Application Number Title Priority Date Filing Date
DD181858A DD116830A5 (US06168776-20010102-C00041.png) 1973-10-23 1974-10-23

Country Status (27)

Country Link
US (1) US3951999A (US06168776-20010102-C00041.png)
JP (2) JPS5912671B2 (US06168776-20010102-C00041.png)
AR (3) AR209755A1 (US06168776-20010102-C00041.png)
AT (1) AT341520B (US06168776-20010102-C00041.png)
AU (1) AU510909B2 (US06168776-20010102-C00041.png)
BE (1) BE821406A (US06168776-20010102-C00041.png)
BG (2) BG26531A4 (US06168776-20010102-C00041.png)
CA (1) CA1042005A (US06168776-20010102-C00041.png)
CH (2) CH595360A5 (US06168776-20010102-C00041.png)
CS (1) CS189671B2 (US06168776-20010102-C00041.png)
DD (1) DD116830A5 (US06168776-20010102-C00041.png)
DE (1) DE2450053A1 (US06168776-20010102-C00041.png)
DK (1) DK552674A (US06168776-20010102-C00041.png)
ES (3) ES431247A1 (US06168776-20010102-C00041.png)
FR (3) FR2248041B1 (US06168776-20010102-C00041.png)
GB (1) GB1488003A (US06168776-20010102-C00041.png)
HU (1) HU171613B (US06168776-20010102-C00041.png)
IE (1) IE40078B1 (US06168776-20010102-C00041.png)
IL (3) IL45880A (US06168776-20010102-C00041.png)
NL (1) NL7413848A (US06168776-20010102-C00041.png)
NZ (1) NZ175780A (US06168776-20010102-C00041.png)
PH (1) PH11022A (US06168776-20010102-C00041.png)
RO (2) RO74031A (US06168776-20010102-C00041.png)
SE (3) SE424324B (US06168776-20010102-C00041.png)
SU (3) SU604491A3 (US06168776-20010102-C00041.png)
YU (1) YU282474A (US06168776-20010102-C00041.png)
ZA (1) ZA746594B (US06168776-20010102-C00041.png)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1590587A (en) * 1977-06-28 1981-06-03 Lilly Industries Ltd Benoxaprofen
US4728662A (en) * 1977-11-21 1988-03-01 Hoechst-Roussel Pharmaceuticals Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4673746A (en) * 1978-10-06 1987-06-16 Hoechst-Roussel Pharmaceuticals, Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
NZ189705A (en) * 1978-03-01 1981-07-13 Boots Co Ltd Benzophenone-hydrazone derivatives and pesticidal compositions intermediates
US4337261A (en) * 1980-07-28 1982-06-29 Hoechst-Roussel Pharmaceuticals Inc. (1,2-Benzisoxazol)phenoxyacetic acids as diuretics
US4894461A (en) * 1981-04-27 1990-01-16 Hoechst-Roussel Pharmaceuticals, Inc. 3-(γ-chloropropyl)-6-fluoro-1,2-benzisoxazole
US4396770A (en) * 1982-04-09 1983-08-02 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-hydroxy-4-phenylpiperidines
US4609658A (en) * 1982-04-09 1986-09-02 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted) piperazines useful for reducing blood pressure
US4536578A (en) * 1982-04-09 1985-08-20 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines
US4458075A (en) * 1982-04-09 1984-07-03 Hoechst-Roussel Pharmaceuticals Inc. 6-Fluoro-3-[3-(1-heterocyclo)propyl]-1,2-benzisoxazoles
US4374245A (en) * 1982-04-09 1983-02-15 Hoechst-Roussel Pharmaceuticals Inc. 8-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
US4610988A (en) * 1982-04-09 1986-09-09 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines useful for alleviating pain
US4390544A (en) * 1982-04-09 1983-06-28 Hoechst-Roussel Pharmaceuticals Inc. {1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(2-oxo-1-benzimidazolinyl}p
US4420485A (en) * 1982-09-29 1983-12-13 Hoechst-Roussel Pharmaceuticals Inc. 1'-[3-(1,2-Benzisoxazol-3-yl) proply]spiro[benzofuran-2(3H),3' or 4'-piperidines or 3'-pyrrolidines]
FR2540107B1 (fr) * 1983-01-28 1986-10-17 Inst Rech Chim Biolog Nouveaux derives d'halogenobenzophenone-oxime, utilisation en therapeutique et procede de preparation
FI92189C (fi) * 1986-03-17 1994-10-10 Eisai Co Ltd Menetelmä lääkeaineina käyttökelpoisen difenyylimetaanijohdannaisen valmistamiseksi
US4898874A (en) * 1986-09-15 1990-02-06 A. H. Robins Company, Inc. Acetic acid derivatives of 3-aryl-2,1-benzisoxazole and esters and amides thereof
JPH037961U (US06168776-20010102-C00041.png) * 1989-06-14 1991-01-25
US5114960A (en) * 1989-07-20 1992-05-19 Hoffmann-La Roche Inc. Substituted isoxazole derivatives
BRPI0707719A2 (pt) * 2006-02-10 2011-05-10 Summit Corp Plc uso de um composto ou de um sal farmaceuticamente aceitÁvel do mesmo
RU2586330C2 (ru) * 2011-09-16 2016-06-10 Пфайзер Инк. Твердые формы ингибитора диссоциации транстиретина

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH1093669A4 (US06168776-20010102-C00041.png) * 1969-07-17 1971-02-15
FR2093173A5 (en) * 1970-06-04 1972-01-28 Gen Mills Inc Substituted 2-hydroxybenzophenoximes for - copper extraction

Also Published As

Publication number Publication date
SE7710600L (sv) 1977-09-21
ES431247A1 (es) 1977-02-16
GB1488003A (en) 1977-10-05
DK552674A (US06168776-20010102-C00041.png) 1975-06-16
SE7413237L (US06168776-20010102-C00041.png) 1975-04-24
ZA746594B (en) 1976-06-30
SE7710599L (sv) 1977-09-21
SU608476A3 (ru) 1978-05-25
JPS5077364A (US06168776-20010102-C00041.png) 1975-06-24
SE435713B (sv) 1984-10-15
AR209755A1 (es) 1977-05-31
FR2361359B1 (US06168776-20010102-C00041.png) 1979-07-20
NL7413848A (nl) 1975-04-25
BG25991A3 (bg) 1979-01-12
FR2361328A1 (fr) 1978-03-10
JPS57154174A (en) 1982-09-22
ES449655A1 (es) 1977-07-01
AU510909B2 (en) 1980-07-17
CS189671B2 (en) 1979-04-30
IL52180A0 (en) 1977-07-31
AU2880177A (en) 1979-03-15
CA1042005A (en) 1978-11-07
FR2248041A1 (US06168776-20010102-C00041.png) 1975-05-16
PH11022A (en) 1977-10-25
YU282474A (en) 1982-02-28
FR2248041B1 (US06168776-20010102-C00041.png) 1978-09-08
ES449654A1 (es) 1977-07-01
DE2450053A1 (de) 1975-04-24
IE40078L (en) 1975-04-23
JPS5912671B2 (ja) 1984-03-24
IL45880A (en) 1979-09-30
AU7454774A (en) 1976-04-29
BE821406A (fr) 1975-04-23
FR2361359A1 (fr) 1978-03-10
JPS636066B2 (US06168776-20010102-C00041.png) 1988-02-08
NZ175780A (en) 1978-04-03
IL52179A0 (en) 1977-07-31
FR2361328B1 (US06168776-20010102-C00041.png) 1979-07-13
CH605864A5 (US06168776-20010102-C00041.png) 1978-10-13
US3951999A (en) 1976-04-20
AT341520B (de) 1978-02-10
CH595360A5 (US06168776-20010102-C00041.png) 1978-02-15
AR221321A1 (es) 1981-01-30
IE40078B1 (en) 1979-03-14
AR213086A1 (es) 1978-12-15
IL45880A0 (en) 1974-12-31
RO74031A (ro) 1982-02-01
SE424324B (sv) 1982-07-12
SE424325B (sv) 1982-07-12
BG26531A4 (bg) 1979-04-12
SU795459A3 (ru) 1981-01-07
SU604491A3 (ru) 1978-04-25
HU171613B (hu) 1978-02-28
RO78465A (ro) 1982-02-26
ATA852374A (de) 1977-06-15

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