CY1124177T1 - Ενωσεις χρησιμες για την αναστολη του ror-γαμμα-τ - Google Patents

Ενωσεις χρησιμες για την αναστολη του ror-γαμμα-τ

Info

Publication number
CY1124177T1
CY1124177T1 CY20211100455T CY211100455T CY1124177T1 CY 1124177 T1 CY1124177 T1 CY 1124177T1 CY 20211100455 T CY20211100455 T CY 20211100455T CY 211100455 T CY211100455 T CY 211100455T CY 1124177 T1 CY1124177 T1 CY 1124177T1
Authority
CY
Cyprus
Prior art keywords
gamma
compounds useful
ror
inhibiting ror
inhibiting
Prior art date
Application number
CY20211100455T
Other languages
English (en)
Inventor
Christian Alexander Clarke
Charles Willis Lugar Iii
John Richard Morphy
Timothy Ivo Richardson
Helene Rudyk
Selma Sapmaz
Ryan Edward Stites
Grant Mathews Vaught
Original Assignee
Eli Lilly And Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly And Company filed Critical Eli Lilly And Company
Publication of CY1124177T1 publication Critical patent/CY1124177T1/el

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/20Spiro-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Η παρούσα εφεύρεση παρέχει νέους αναστολείς του ROR γάμμα-t και φαρμακευτικές συνθέσεις αυτών, τύπος (Α).
CY20211100455T 2017-03-02 2021-05-26 Ενωσεις χρησιμες για την αναστολη του ror-γαμμα-τ CY1124177T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201762466117P 2017-03-02 2017-03-02
PCT/US2018/019920 WO2018160550A1 (en) 2017-03-02 2018-02-27 Compounds useful for inhibiting ror-gamma-t

Publications (1)

Publication Number Publication Date
CY1124177T1 true CY1124177T1 (el) 2022-05-27

Family

ID=61622740

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20211100455T CY1124177T1 (el) 2017-03-02 2021-05-26 Ενωσεις χρησιμες για την αναστολη του ror-γαμμα-τ

Country Status (15)

Country Link
US (1) US11008336B2 (el)
EP (1) EP3589638B1 (el)
JP (1) JP6766273B2 (el)
CN (1) CN110337440B (el)
CY (1) CY1124177T1 (el)
DK (1) DK3589638T3 (el)
ES (1) ES2871911T3 (el)
HR (1) HRP20210898T1 (el)
HU (1) HUE054483T2 (el)
LT (1) LT3589638T (el)
PL (1) PL3589638T3 (el)
PT (1) PT3589638T (el)
RS (1) RS61788B1 (el)
SI (1) SI3589638T1 (el)
WO (1) WO2018160550A1 (el)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022122740A1 (en) 2020-12-07 2022-06-16 Diaccurate Ror-gamma inhibitors for the treatment of ror-gamma-dependent cancer

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA05000729A (es) * 2002-07-17 2005-04-08 Warner Lambert Co Combinacion de un inhibidor alosterico de metaloproteinasa-13 de matriz con celecoxib o valdecoxib.
UA107943C2 (en) 2009-11-16 2015-03-10 Lilly Co Eli Compounds of spiropiperidines as antagonists of the orl-1 receptors
SI2501704T1 (sl) 2009-11-16 2013-11-29 Eli Lilly Company Spojine spiropiperidina kot antagonisti oral-1 receptorja
TWI582096B (zh) 2011-12-06 2017-05-11 美國禮來大藥廠 用於酒精依賴及濫用處理之4',5'-二氫螺[哌啶-4,7'-噻吩并[2,3-c]哌喃]化合物
WO2014179564A1 (en) 2013-05-01 2014-11-06 Vitae Pharmaceuticals, Inc. Thiazalopyrrolidine inhibitors of ror-gamma
JP6192836B2 (ja) * 2013-07-30 2017-09-06 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Rorcモジュレーターとしてのアザインドール化合物
WO2015101928A1 (en) * 2013-12-31 2015-07-09 Aurigene Discovery Technologies Limited Fused thiophene and thiazole derivatives as ror gamma modulators
MX2016009621A (es) * 2014-01-24 2016-11-17 Abbvie Inc Derivados de fur0-3-carboxamida y metodos de uso.
AR105821A1 (es) 2015-09-09 2017-11-15 Lilly Co Eli COMPUESTOS ÚTILES PARA INHIBIR ROR-g-T
PT3589637T (pt) * 2017-03-02 2021-06-02 Lilly Co Eli Compostos úteis para inibir ror-gamma-t

Also Published As

Publication number Publication date
HUE054483T2 (hu) 2021-09-28
US11008336B2 (en) 2021-05-18
SI3589638T1 (sl) 2021-08-31
ES2871911T3 (es) 2021-11-02
US20200048279A1 (en) 2020-02-13
HRP20210898T1 (hr) 2021-08-20
JP2020509049A (ja) 2020-03-26
CN110337440B (zh) 2021-08-03
PT3589638T (pt) 2021-05-27
RS61788B1 (sr) 2021-06-30
CN110337440A (zh) 2019-10-15
EP3589638A1 (en) 2020-01-08
JP6766273B2 (ja) 2020-10-07
PL3589638T3 (pl) 2021-09-27
DK3589638T3 (da) 2021-06-07
LT3589638T (lt) 2021-06-10
WO2018160550A1 (en) 2018-09-07
EP3589638B1 (en) 2021-04-07

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