CY1113982T1 - Μεθοδος διεργασιων για την παρασκευη βενζοφουραν-2-καρβοξαμιδιων - Google Patents

Μεθοδος διεργασιων για την παρασκευη βενζοφουραν-2-καρβοξαμιδιων

Info

Publication number
CY1113982T1
CY1113982T1 CY20131100370T CY131100370T CY1113982T1 CY 1113982 T1 CY1113982 T1 CY 1113982T1 CY 20131100370 T CY20131100370 T CY 20131100370T CY 131100370 T CY131100370 T CY 131100370T CY 1113982 T1 CY1113982 T1 CY 1113982T1
Authority
CY
Cyprus
Prior art keywords
benzofuran
preparation
carboxamide
processing
carboxamides
Prior art date
Application number
CY20131100370T
Other languages
English (en)
Inventor
Andreas Bathe
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of CY1113982T1 publication Critical patent/CY1113982T1/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/84—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D307/85—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Furan Compounds (AREA)

Abstract

Η εφεύρεση αφορά μία μέθοδο διεργασιών για την παρασκευή βενζοφουραν-2-καρβοξαμιδίων του τύπου (I), στον οποίον R1, R2, R3, R4, R5, και R6 έχουν τις σημασίες που δίδονται στην αξίωση 1.
CY20131100370T 2006-12-21 2013-05-07 Μεθοδος διεργασιων για την παρασκευη βενζοφουραν-2-καρβοξαμιδιων CY1113982T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102006060597A DE102006060597A1 (de) 2006-12-21 2006-12-21 Verfahren zur Herstellung von Benzofuran-2-carboxamiden
EP07856224A EP2121649B1 (de) 2006-12-21 2007-11-22 Verfahren zur Herstellung von Benzofuran-2-carboxamiden

Publications (1)

Publication Number Publication Date
CY1113982T1 true CY1113982T1 (el) 2016-07-27

Family

ID=39246392

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20131100370T CY1113982T1 (el) 2006-12-21 2013-05-07 Μεθοδος διεργασιων για την παρασκευη βενζοφουραν-2-καρβοξαμιδιων

Country Status (20)

Country Link
US (1) US20100036139A1 (el)
EP (1) EP2121649B1 (el)
JP (1) JP5319547B2 (el)
KR (1) KR20090092334A (el)
CN (1) CN101573347B (el)
AR (1) AR064441A1 (el)
AU (1) AU2007341750B2 (el)
BR (1) BRPI0720450A2 (el)
CA (1) CA2673429A1 (el)
CY (1) CY1113982T1 (el)
DE (1) DE102006060597A1 (el)
DK (1) DK2121649T3 (el)
ES (1) ES2404804T3 (el)
HK (1) HK1134925A1 (el)
MX (1) MX2009006402A (el)
PL (1) PL2121649T3 (el)
PT (1) PT2121649E (el)
SI (1) SI2121649T1 (el)
WO (1) WO2008080456A1 (el)
ZA (1) ZA200905055B (el)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101361145B1 (ko) * 2011-03-10 2014-02-12 한국화학연구원 신규한 벤조퓨란-2-카르복사미드 유도체 및 그의 ｍｃｈ 수용체-1 관련 질환에 대한 치료학적 용도

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU6004073A (en) * 1972-09-09 1975-03-06 Basf Ag Fluorescent benzofuran compounds
IT1115926B (it) * 1977-03-30 1986-02-10 Minnesota Mining & Mfg Copulanti magenta 5-pirazolonici per uso fotografico elementi fotografici che li contengono e procedimento per la loro produzione
US4229467A (en) * 1979-08-16 1980-10-21 Richardson-Merrell Inc. Alkoxy benzofuran carboxylic acids and salts and esters thereof as hypolipidemic agents
US4495357A (en) * 1981-07-01 1985-01-22 The Upjohn Company Pyridyl-substituted-benzofurans
DE19932314A1 (de) * 1999-07-10 2001-01-11 Merck Patent Gmbh Benzofuranderivate
DE19958496A1 (de) * 1999-12-04 2001-06-07 Merck Patent Gmbh Verfahren zur Herstellung von 5-(1-Piperazinyl)-benzofuran-2-carboxamid durch Übergangsmetallkatalysierte Aminierung
DE10112151A1 (de) * 2001-03-14 2002-09-19 Merck Patent Gmbh Substituierte Benzofuran-2-carbonsäureamide
SE0400441D0 (sv) * 2004-02-25 2004-02-25 Active Biotech Ab Novel Benzofurans and Indols

Also Published As

Publication number Publication date
AU2007341750A1 (en) 2008-07-10
PL2121649T3 (pl) 2013-06-28
ES2404804T3 (es) 2013-05-29
US20100036139A1 (en) 2010-02-11
CN101573347A (zh) 2009-11-04
JP2010513336A (ja) 2010-04-30
EP2121649A1 (de) 2009-11-25
BRPI0720450A2 (pt) 2014-01-14
CN101573347B (zh) 2012-10-10
PT2121649E (pt) 2013-05-21
HK1134925A1 (en) 2010-05-20
DE102006060597A1 (de) 2008-06-26
EP2121649B1 (de) 2013-02-27
JP5319547B2 (ja) 2013-10-16
SI2121649T1 (sl) 2013-06-28
ZA200905055B (en) 2010-04-28
KR20090092334A (ko) 2009-08-31
CA2673429A1 (en) 2008-07-10
MX2009006402A (es) 2009-06-23
AU2007341750B2 (en) 2013-04-18
WO2008080456A1 (de) 2008-07-10
DK2121649T3 (da) 2013-05-06
AR064441A1 (es) 2009-04-01

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