CU24304B1 - Formulación de fármaco de liberación retardada - Google Patents

Formulación de fármaco de liberación retardada

Info

Publication number
CU24304B1
CU24304B1 CUP2014000123A CU20140123A CU24304B1 CU 24304 B1 CU24304 B1 CU 24304B1 CU P2014000123 A CUP2014000123 A CU P2014000123A CU 20140123 A CU20140123 A CU 20140123A CU 24304 B1 CU24304 B1 CU 24304B1
Authority
CU
Cuba
Prior art keywords
outer layer
core
polymeric material
layer
drug
Prior art date
Application number
CUP2014000123A
Other languages
English (en)
Spanish (es)
Other versions
CU20140123A7 (es
Inventor
Abdul Waseh Basit
González Roberto Carlos Bravo
Thomas Buser
Ana Cristina Freire
Frédéric Jean-Claude Goutte
Felipe José Oliveria Varum
Original Assignee
Tillotts Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46025554&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CU24304(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Tillotts Pharma Ag filed Critical Tillotts Pharma Ag
Publication of CU20140123A7 publication Critical patent/CU20140123A7/es
Publication of CU24304B1 publication Critical patent/CU24304B1/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
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    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/60—Salicylic acid; Derivatives thereof
    • A61K31/606—Salicylic acid; Derivatives thereof having amino groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/60—Salicylic acid; Derivatives thereof
    • A61K31/612—Salicylic acid; Derivatives thereof having the hydroxy group in position 2 esterified, e.g. salicylsulfuric acid
    • A61K31/616—Salicylic acid; Derivatives thereof having the hydroxy group in position 2 esterified, e.g. salicylsulfuric acid by carboxylic acids, e.g. acetylsalicylic acid
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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    • A61K9/2022—Organic macromolecular compounds
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    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
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    • A61K9/2833—Organic macromolecular compounds
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    • A—HUMAN NECESSITIES
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    • A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Inorganic Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Botany (AREA)
  • Zoology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Preparation (AREA)
  • Laminated Bodies (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • General Preparation And Processing Of Foods (AREA)
  • Grain Derivatives (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CUP2014000123A 2012-04-30 2013-04-29 Formulación de fármaco de liberación retardada CU24304B1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261640217P 2012-04-30 2012-04-30
EP12166110.2A EP2659881B1 (de) 2012-04-30 2012-04-30 Arzneimittelformulierung mit verzögerter Freisetzung
PCT/EP2013/058923 WO2013164316A1 (en) 2012-04-30 2013-04-29 A delayed release drug formulation

Publications (2)

Publication Number Publication Date
CU20140123A7 CU20140123A7 (es) 2015-02-26
CU24304B1 true CU24304B1 (es) 2018-01-10

Family

ID=46025554

Family Applications (1)

Application Number Title Priority Date Filing Date
CUP2014000123A CU24304B1 (es) 2012-04-30 2013-04-29 Formulación de fármaco de liberación retardada

Country Status (41)

Country Link
US (6) US9364440B2 (de)
EP (6) EP3187171B1 (de)
JP (2) JP6621662B2 (de)
KR (6) KR102177773B1 (de)
CN (5) CN110237056B (de)
AR (1) AR090898A1 (de)
AU (4) AU2013255913B2 (de)
BR (3) BR112014026935A2 (de)
CA (4) CA2871017A1 (de)
CL (2) CL2014002796A1 (de)
CO (2) CO7151506A2 (de)
CR (4) CR20190245A (de)
CU (1) CU24304B1 (de)
CY (4) CY1120215T1 (de)
DK (5) DK2659881T3 (de)
EA (2) EA032514B1 (de)
ES (6) ES2655622T3 (de)
GE (4) GEP201706736B (de)
HR (2) HRP20180068T1 (de)
HU (5) HUE036187T2 (de)
JO (6) JOP20200144A1 (de)
LT (5) LT2659881T (de)
ME (2) ME03641B (de)
MX (4) MX366677B (de)
MY (3) MY190392A (de)
NO (1) NO2659881T3 (de)
NZ (3) NZ725409A (de)
PE (3) PE20142442A1 (de)
PH (2) PH12014502339A1 (de)
PL (5) PL2659881T3 (de)
PT (5) PT2659881T (de)
RS (5) RS56839B1 (de)
SA (2) SA115370043B1 (de)
SG (2) SG11201406798WA (de)
SI (5) SI2659881T1 (de)
SM (5) SMT201800095T1 (de)
TN (2) TN2014000442A1 (de)
TR (3) TR201809416T4 (de)
TW (3) TWI700102B (de)
UY (1) UY34772A (de)
WO (2) WO2013164316A1 (de)

Families Citing this family (38)

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Publication number Priority date Publication date Assignee Title
SI2659881T1 (en) 2012-04-30 2018-03-30 Tillotts Pharma Ag Formulation of the delayed release medicinal product
CU24343B1 (es) * 2012-04-30 2018-05-08 Tillotts Pharma Ag Formulación de fármaco de liberación retardada
US20140141075A1 (en) 2012-11-21 2014-05-22 Warner Chilcott Company, Llc 5-aminosalicylic acid capsule formulation
TWI688411B (zh) * 2013-02-22 2020-03-21 日商志瑞亞新藥工業股份有限公司 腸溶錠
EA032504B1 (ru) 2013-10-29 2019-06-28 Тиллоттс Фарма АГ Лекарственный препарат с отсроченным высвобождением и его применение для доставки лекарственного средства
EP3086776B1 (de) 2013-12-24 2020-06-17 Sentiss Pharma Private Limited Topische brimonidintartrat-lösung für die augen
AU2016271303C1 (en) 2015-06-01 2022-04-14 Xeno Biosciences Inc. Methods and compositions to modulate the gut microbiota and to manage weight
CN108283000B (zh) 2015-09-23 2021-04-13 凯瑞康宁生物工程（武汉）有限公司 γ-羟基丁酸的前药及其组合物和用途
CN105816883B (zh) * 2016-02-03 2018-12-14 华南师范大学 一种负载抗癌药物姜黄素的益生菌叶酸靶向载体及其制备方法
EP3257501A1 (de) 2016-06-14 2017-12-20 Tillotts Pharma AG Aus mehreren einzeleinheiten zusammengesetzte dosierungsform mit einem kern aus individuellen kerneinheiten, die mit mukoadhäsivem material bedeckt sind, sowie einer enterischen kernbeschichtung
WO2018102469A1 (en) * 2016-11-30 2018-06-07 Xeno Biosciences Inc. Pharmaceutical preparations and methods to manage weight and to modulate the gut microbiota
EP3768302B1 (de) 2018-03-20 2025-05-07 Theriva Biologics, Inc. Intestinale alkalische phosphataseformulierungen
EA202092275A1 (ru) * 2018-03-23 2021-02-09 Палатин Текнолоджиз, Инк. Составы пептидов, специфичных к рецептору меланокортина, и способы доставки в желудочно-кишечный тракт
CN113348011B (zh) 2018-11-19 2023-04-18 比奥拉治疗股份有限公司 用生物治疗剂治疗疾病的方法和装置
EP3662898A1 (de) 2018-12-07 2020-06-10 Tillotts Pharma AG Feste formulierung enthaltend mesalazin
ES3002632T3 (en) 2018-12-07 2025-03-07 Tillotts Pharma Ag Delayed release drug formulation comprising an outerlayer with an enzymatically degradable polymer, its composition and its method of manufacturing
EP3662895A1 (de) 2018-12-07 2020-06-10 Tillotts Pharma AG Verfahren zur herstellung von reduzierenden zuckerfreien 5-asa-tablettenkernen
EP3662902B1 (de) * 2018-12-07 2024-07-31 Tillotts Pharma AG Formulierung mit freisetzung eines wirkstoffs im kolon
EP3662900A1 (de) * 2018-12-07 2020-06-10 Tillotts Pharma AG Kolonwirkstoffverabreichungsformulierung
ES2906316T3 (es) * 2018-12-10 2022-04-18 Aphaia Ip Ag Formas farmacéuticas de dosificación oral para el tratamiento de trastornos metabólicos y enfermedades relacionadas mediante la liberación orquestada de enterocinas
CN111617047B (zh) * 2019-02-27 2021-06-22 广州喜鹊医药有限公司 一种含tbn或其盐或其水合物的药物组合物及其制备方法
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