CS801886A2 - Method of substituted imidazopyrrole,-pyridine and-azepine derivatives production - Google Patents
Method of substituted imidazopyrrole,-pyridine and-azepine derivatives productionInfo
- Publication number
- CS801886A2 CS801886A2 CS868018A CS801886A CS801886A2 CS 801886 A2 CS801886 A2 CS 801886A2 CS 868018 A CS868018 A CS 868018A CS 801886 A CS801886 A CS 801886A CS 801886 A2 CS801886 A2 CS 801886A2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- opt
- alkyl
- substd
- alkoxy
- etherified
- Prior art date
Links
- JUJWROOIHBZHMG-UHFFFAOYSA-N pyridine Substances C1=CC=NC=C1 JUJWROOIHBZHMG-UHFFFAOYSA-N 0.000 title 1
- MHOZZUICEDXVGD-UHFFFAOYSA-N pyrrolo[2,3-d]imidazole Chemical class C1=NC2=CC=NC2=N1 MHOZZUICEDXVGD-UHFFFAOYSA-N 0.000 title 1
- -1 alkanoyl alkanoyloxy Chemical group 0.000 abstract 10
- 125000000217 alkyl group Chemical group 0.000 abstract 9
- 125000003545 alkoxy group Chemical group 0.000 abstract 6
- 229910052736 halogen Inorganic materials 0.000 abstract 6
- 150000002367 halogens Chemical class 0.000 abstract 6
- 125000001589 carboacyl group Chemical group 0.000 abstract 5
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 5
- 125000004423 acyloxy group Chemical group 0.000 abstract 4
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 4
- 125000004414 alkyl thio group Chemical group 0.000 abstract 3
- RAXXELZNTBOGNW-UHFFFAOYSA-N imidazole Natural products C1=CNC=N1 RAXXELZNTBOGNW-UHFFFAOYSA-N 0.000 abstract 3
- 125000000020 sulfo group Chemical group O=S(=O)([*])O[H] 0.000 abstract 3
- JCXJVPUVTGWSNB-UHFFFAOYSA-N Nitrogen dioxide Chemical compound O=[N]=O JCXJVPUVTGWSNB-UHFFFAOYSA-N 0.000 abstract 2
- 229910006069 SO3H Inorganic materials 0.000 abstract 2
- 125000005078 alkoxycarbonylalkyl group Chemical group 0.000 abstract 2
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 2
- 125000004181 carboxyalkyl group Chemical group 0.000 abstract 2
- 125000004663 dialkyl amino group Chemical group 0.000 abstract 2
- 125000002485 formyl group Chemical group [H]C(*)=O 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 125000003884 phenylalkyl group Chemical group 0.000 abstract 2
- 125000004660 phenylalkylthio group Chemical group 0.000 abstract 2
- 125000003356 phenylsulfanyl group Chemical group [*]SC1=C([H])C([H])=C([H])C([H])=C1[H] 0.000 abstract 2
- 102000014654 Aromatase Human genes 0.000 abstract 1
- 108010078554 Aromatase Proteins 0.000 abstract 1
- 229910006074 SO2NH2 Inorganic materials 0.000 abstract 1
- 125000005042 acyloxymethyl group Chemical group 0.000 abstract 1
- 125000004849 alkoxymethyl group Chemical group 0.000 abstract 1
- 125000004644 alkyl sulfinyl group Chemical group 0.000 abstract 1
- 125000004390 alkyl sulfonyl group Chemical group 0.000 abstract 1
- 125000005278 alkyl sulfonyloxy group Chemical group 0.000 abstract 1
- 125000004397 aminosulfonyl group Chemical group NS(=O)(=O)* 0.000 abstract 1
- MDFFNEOEWAXZRQ-UHFFFAOYSA-N aminyl Chemical compound [NH2] MDFFNEOEWAXZRQ-UHFFFAOYSA-N 0.000 abstract 1
- 125000003236 benzoyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C(*)=O 0.000 abstract 1
- 125000002619 bicyclic group Chemical group 0.000 abstract 1
- 125000005117 dialkylcarbamoyl group Chemical group 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 125000004005 formimidoyl group Chemical group [H]\N=C(/[H])* 0.000 abstract 1
- 125000004970 halomethyl group Chemical group 0.000 abstract 1
- CBOIHMRHGLHBPB-UHFFFAOYSA-N hydroxymethyl Chemical compound O[CH2] CBOIHMRHGLHBPB-UHFFFAOYSA-N 0.000 abstract 1
- 230000005764 inhibitory process Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CS868018A CS268684B2 (en) | 1984-06-20 | 1986-11-05 | Method of substituted imidazopyrrole,-pyridine and-azepine derivatives production |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/622,421 US4617307A (en) | 1984-06-20 | 1984-06-20 | Substituted imidazo[1,5-A]pyridine derivatives as aromatase inhibitors |
| CS854449A CS268672B2 (en) | 1984-06-20 | 1985-06-18 | Method of substituted imidazo-(1,5-a)pyridine derivatives production |
| CS868018A CS268684B2 (en) | 1984-06-20 | 1986-11-05 | Method of substituted imidazopyrrole,-pyridine and-azepine derivatives production |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CS801886A2 true CS801886A2 (en) | 1989-07-12 |
| CS268684B2 CS268684B2 (en) | 1990-04-11 |
Family
ID=25745999
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS868018A CS268684B2 (en) | 1984-06-20 | 1986-11-05 | Method of substituted imidazopyrrole,-pyridine and-azepine derivatives production |
| CS868021A CS268687B2 (en) | 1984-06-20 | 1986-11-05 | Method of substituted imidazopyridine derivatives production |
| CS868019A CS268685B2 (en) | 1984-06-20 | 1986-11-05 | Method of substituted imidazopyrrole,-pyridine and-azepine derivatives production |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS868021A CS268687B2 (en) | 1984-06-20 | 1986-11-05 | Method of substituted imidazopyridine derivatives production |
| CS868019A CS268685B2 (en) | 1984-06-20 | 1986-11-05 | Method of substituted imidazopyrrole,-pyridine and-azepine derivatives production |
Country Status (1)
| Country | Link |
|---|---|
| CS (3) | CS268684B2 (cs) |
-
1986
- 1986-11-05 CS CS868018A patent/CS268684B2/cs not_active IP Right Cessation
- 1986-11-05 CS CS868021A patent/CS268687B2/cs not_active IP Right Cessation
- 1986-11-05 CS CS868019A patent/CS268685B2/cs not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| CS268684B2 (en) | 1990-04-11 |
| CS268687B2 (en) | 1990-04-11 |
| CS268685B2 (en) | 1990-04-11 |
| CS801986A2 (en) | 1989-07-12 |
| CS802186A2 (en) | 1989-07-12 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK4A | Patent expired |
Effective date: 20000618 |