CS187388B2 - Method of producing n-acyl derivatives of ampicillin and p-hydroxyampicillin - Google Patents

Method of producing n-acyl derivatives of ampicillin and p-hydroxyampicillin

Info

Publication number
CS187388B2
CS187388B2 CS738474A CS847473A CS187388B2 CS 187388 B2 CS187388 B2 CS 187388B2 CS 738474 A CS738474 A CS 738474A CS 847473 A CS847473 A CS 847473A CS 187388 B2 CS187388 B2 CS 187388B2
Authority
CS
Czechoslovakia
Prior art keywords
hydroxyampicillin
ampicillin
producing
acyl derivatives
acyl
Prior art date
Application number
CS738474A
Other languages
Czech (cs)
English (en)
Inventor
Gunter Schmidt
Karl G Metzger
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of CS187388B2 publication Critical patent/CS187388B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/16—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • C07D249/18—Benzotriazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Cephalosporin Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Fodder In General (AREA)
CS738474A 1972-12-08 1973-12-07 Method of producing n-acyl derivatives of ampicillin and p-hydroxyampicillin CS187388B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2260118A DE2260118C2 (de) 1972-12-08 1972-12-08 Penicilline sowie ihre Verwendung als Arzneimittel

Publications (1)

Publication Number Publication Date
CS187388B2 true CS187388B2 (en) 1979-01-31

Family

ID=5863890

Family Applications (1)

Application Number Title Priority Date Filing Date
CS738474A CS187388B2 (en) 1972-12-08 1973-12-07 Method of producing n-acyl derivatives of ampicillin and p-hydroxyampicillin

Country Status (27)

Country Link
US (1) US3931153A (fr)
JP (2) JPS5747679B2 (fr)
AR (1) AR207749A1 (fr)
AT (1) AT326268B (fr)
AU (1) AU476464B2 (fr)
BE (1) BE808374A (fr)
BG (1) BG21860A3 (fr)
CA (1) CA1026748A (fr)
CH (1) CH593983A5 (fr)
CS (1) CS187388B2 (fr)
DD (1) DD112652A5 (fr)
DE (1) DE2260118C2 (fr)
DK (1) DK141728C (fr)
EG (1) EG11021A (fr)
ES (1) ES421281A1 (fr)
FR (1) FR2209548B1 (fr)
GB (1) GB1409689A (fr)
HU (1) HU167710B (fr)
IE (1) IE38615B1 (fr)
IL (1) IL43757A (fr)
LU (1) LU68952A1 (fr)
NL (1) NL7316679A (fr)
PH (1) PH10602A (fr)
PL (1) PL91236B1 (fr)
RO (1) RO65788A (fr)
SU (1) SU515458A3 (fr)
ZA (1) ZA739331B (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU626881B2 (en) * 1988-07-14 1992-08-13 F. Hoffmann-La Roche Ag Benzofused heterocyclics used as pharmaceuticals
HU229049B1 (en) * 1995-03-31 2013-07-29 Emisphere Tech Inc Compound and compositions for delivering active ingredients
US6001347A (en) * 1995-03-31 1999-12-14 Emisphere Technologies, Inc. Compounds and compositions for delivering active agents
DE60133555T2 (de) * 2000-06-29 2008-09-18 Emisphere Technologies, Inc. Verbindungen und gemische zur verabreichung eines aktiven agens
KR100463418B1 (ko) * 2002-11-11 2004-12-23 한국전자통신연구원 Ｃｅｌｐ 음성 부호화기에서 사용되는 가변적인 고정코드북 검색방법 및 장치
KR100786300B1 (ko) * 2006-09-19 2007-12-18 (주)아모레퍼시픽 3,4-메틸렌디옥시벤젠 또는 3,4-에틸렌디옥시벤젠 모핵을가지는 4-치환된 벤조산 유도체 화합물을 함유하는항노화용 화장료 조성물
GB0915196D0 (en) 2009-09-01 2009-10-07 King S College London Therapeutic compounds and their use

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3268513A (en) * 1964-03-20 1966-08-23 American Home Prod Process for producing 6-(alpha-amino-acylamino-acylamino)-penicillanic acids
US3340252A (en) * 1964-04-07 1967-09-05 American Home Prod Amino-acylamino-acylamino-penicillanic acids
DE1545615A1 (de) * 1964-09-03 1969-08-07 Beecham Group Ltd Verfahren zur Herstellung von Penicillinen
GB1130445A (en) * 1966-04-26 1968-10-16 Beecham Group Ltd Penicillins
CH571524A5 (fr) * 1970-05-25 1976-01-15 Bayer Ag

Also Published As

Publication number Publication date
RO65788A (fr) 1980-06-15
CA1026748A (fr) 1978-02-21
DK141728B (da) 1980-06-02
AU6337573A (en) 1975-06-12
PL91236B1 (fr) 1977-02-28
AT326268B (de) 1975-12-10
DD112652A5 (fr) 1975-04-20
DE2260118A1 (de) 1974-06-12
NL7316679A (fr) 1974-06-11
HU167710B (fr) 1975-12-25
AR207749A1 (es) 1976-10-29
DE2260118C2 (de) 1982-06-03
IL43757A (en) 1976-09-30
GB1409689A (en) 1975-10-15
AU476464B2 (en) 1976-09-23
DK141728C (da) 1980-12-08
ATA1020373A (de) 1975-02-15
US3931153A (en) 1976-01-06
IE38615B1 (en) 1978-04-26
ZA739331B (en) 1974-10-30
FR2209548A1 (fr) 1974-07-05
FR2209548B1 (fr) 1977-09-02
LU68952A1 (fr) 1974-02-12
JPS4987692A (fr) 1974-08-22
BE808374A (fr) 1974-06-07
CH593983A5 (fr) 1977-12-30
IE38615L (en) 1974-06-08
JPS4986521A (fr) 1974-08-19
PH10602A (en) 1977-07-15
BG21860A3 (fr) 1976-09-20
ES421281A1 (es) 1976-04-16
SU515458A3 (ru) 1976-05-25
JPS5747679B2 (fr) 1982-10-12
EG11021A (en) 1977-12-31
IL43757A0 (en) 1974-03-14

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