CS181221B2 - Method of producing 2,4-diamino-5-/3,4,5-triethoxybenzyl/-pyrimidine - Google Patents

Method of producing 2,4-diamino-5-/3,4,5-triethoxybenzyl/-pyrimidine

Info

Publication number
CS181221B2
CS181221B2 CS7200002539A CS253972A CS181221B2 CS 181221 B2 CS181221 B2 CS 181221B2 CS 7200002539 A CS7200002539 A CS 7200002539A CS 253972 A CS253972 A CS 253972A CS 181221 B2 CS181221 B2 CS 181221B2
Authority
CS
Czechoslovakia
Prior art keywords
triethoxybenzyl
diamino
pyrimidine
producing
Prior art date
Application number
CS7200002539A
Other languages
Czech (cs)
Inventor
Barbara Roth
Original Assignee
Barbara Roth
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Barbara Roth filed Critical Barbara Roth
Publication of CS181221B2 publication Critical patent/CS181221B2/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/41—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by hydrogenolysis or reduction of carboxylic groups or functional derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
CS7200002539A 1971-04-16 1972-04-14 Method of producing 2,4-diamino-5-/3,4,5-triethoxybenzyl/-pyrimidine CS181221B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB963971A GB1407971A (en) 1971-04-16 1971-04-16 2,4-diamino -4-3,4,5-triethoxybenzyl pyrimidine and methods of preparation therefor

Publications (1)

Publication Number Publication Date
CS181221B2 true CS181221B2 (en) 1978-03-31

Family

ID=9875880

Family Applications (1)

Application Number Title Priority Date Filing Date
CS7200002539A CS181221B2 (en) 1971-04-16 1972-04-14 Method of producing 2,4-diamino-5-/3,4,5-triethoxybenzyl/-pyrimidine

Country Status (13)

Country Link
JP (3) JPS5320511B1 (en)
AU (1) AU468447B2 (en)
BE (1) BE782153A (en)
CA (1) CA967964A (en)
CH (1) CH565160A5 (en)
CS (1) CS181221B2 (en)
DE (1) DE2218220A1 (en)
DK (1) DK131466B (en)
FR (1) FR2133752B1 (en)
GB (1) GB1407971A (en)
IL (3) IL47921A (en)
NL (1) NL7205043A (en)
SE (1) SE391180B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA738760B (en) * 1972-12-21 1974-08-28 Hoffmann La Roche Process for the manufacture of benzyl pyrimidines
GB1469521A (en) * 1973-01-05 1977-04-06 Wellcome Found Antimicrobial preparations
FR2502152A1 (en) * 1981-03-20 1982-09-24 Panmedica Laboratoires NOVEL SUBSTITUTED DIAMINO-2,4-BENZYL-5-PYRIMIDINE N2-SOLUBLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING SAME

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1090394A (en) * 1953-03-11 1955-03-30 Wellcome Found Pyrimidine derivatives and their manufacture
FR1459417A (en) * 1964-11-12 1966-04-29 Hoffmann La Roche Process for the preparation of pyrimidine derivatives
FR1518635A (en) * 1965-07-08 1968-03-29 Wellcome Found Process for the preparation of pyrimidine derivatives
GB1261455A (en) * 1969-03-06 1972-01-26 Burroughs Wellcome Co Improvements in or relating to substituted acrylonitriles

Also Published As

Publication number Publication date
NL7205043A (en) 1972-10-18
JPS5430189A (en) 1979-03-06
JPS5422994B2 (en) 1979-08-10
FR2133752B1 (en) 1975-04-25
CA967964A (en) 1975-05-20
DK131466B (en) 1975-07-21
JPS5320511B1 (en) 1978-06-27
DK131466C (en) 1975-12-08
IL47921A0 (en) 1975-11-25
BE782153A (en) 1972-10-16
JPS53111083A (en) 1978-09-28
CH565160A5 (en) 1975-08-15
DE2218220A1 (en) 1972-11-02
IL39218A (en) 1976-10-31
AU468447B2 (en) 1976-01-15
IL39218A0 (en) 1972-06-28
FR2133752A1 (en) 1972-12-01
GB1407971A (en) 1975-10-01
AU4117472A (en) 1973-10-18
SE391180B (en) 1977-02-07
IL47921A (en) 1976-10-31

Similar Documents

Publication Publication Date Title
CS179404B2 (en) Method for production of 1,1,2,3,-tetrachlorpropene
SU721000A3 (en) Method of producing acylaniline
CS183654B2 (en) Method of producing 3-methylencephalosporines
CS182260B2 (en) Method of producing 1,3-oxidated 8alfa-estratrienes
CS171232B2 (en) Method of 2,2-diaryl-4-(4'-aryl-4'-hydroxypiperidino) butyramides production
GB1320984A (en) Method of producing 1,3-bis-hydroxyaryl tetraorganodisolaxanes
CS183671B2 (en) Method of producing pure e-caprolactame
CS180585B2 (en) Method of producing derivatives of 2-nitro-5-vinylimidazole
JPS5387342A (en) Method for production of new 44*44biphenyl**11butanol
CS180588B2 (en) Method od producing 4-hydroxymethyl-1-keto-1,2-dihydrophthalazine
JPS5718699A (en) Manufacture of 17,21-dihydroxy-20-ketopregnanes
CS182781B2 (en) Method of producing 2,6-diaminodihydropyridines
GB1319746A (en) Method of producing linear polyalkylalumoxanes
CS180580B2 (en) Method of producing new derivatives of 2-formyl-3-carboxamidochinoxalin-di-n-oxides
CS181221B2 (en) Method of producing 2,4-diamino-5-/3,4,5-triethoxybenzyl/-pyrimidine
YU36963B (en) Process for producing hetacillin derivatives
CS184313B2 (en) Method of producing alkyl-7-deoxy-7-rs-alpha-thiolincosaminides
CA964283A (en) Method of producing 3-phenyl-1-butene
JPS53104631A (en) Method of making 22stilbenyll44stilylltriazole
CS180581B2 (en) Method of producing new 2-pyridazinyl-3-/4-methyl-piperazinocarbonyloxy/-3-isoindolines
CS193477B2 (en) Method of producing 15 alpha,16 alpha-methylene-4-pregnenes
IL39028A0 (en) Method of producing n-trihalogenoalkylthio derivatives
JPS5387361A (en) Method of producing 22*22aminobenzoyl*pyridine
CS193013B2 (en) Method of producing 6-beta-amino-2,2-dimethylpenam-3-alpha-carboxylic acid
GB1403409A (en) Substituted 3,4-dihydropyrimido-4-5-d- pyridazine derivatives and process for producing them