CO6210733A2 - Asociacion de compuestos inhibidores de melanogenesis y su uso en cosmeticos y dermatologia - Google Patents

Asociacion de compuestos inhibidores de melanogenesis y su uso en cosmeticos y dermatologia

Info

Publication number
CO6210733A2
CO6210733A2 CO09074062A CO09074062A CO6210733A2 CO 6210733 A2 CO6210733 A2 CO 6210733A2 CO 09074062 A CO09074062 A CO 09074062A CO 09074062 A CO09074062 A CO 09074062A CO 6210733 A2 CO6210733 A2 CO 6210733A2
Authority
CO
Colombia
Prior art keywords
cosmetic
inhibitor
vitamin
receptor antagonist
composition according
Prior art date
Application number
CO09074062A
Other languages
English (en)
Inventor
Marc Criton
Hamon Veronique Lemellay
Yves Leblond
Original Assignee
Lab Mayoly Spindler Sas
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lab Mayoly Spindler Sas filed Critical Lab Mayoly Spindler Sas
Publication of CO6210733A2 publication Critical patent/CO6210733A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
    • A61K31/375Ascorbic acid, i.e. vitamin C; Salts thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/455Nicotinic acids, e.g. niacin; Derivatives thereof, e.g. esters, amides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/64Proteins; Peptides; Derivatives or degradation products thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/67Vitamins
    • A61K8/673Vitamin B group
    • A61K8/675Vitamin B3 or vitamin B3 active, e.g. nicotinamide, nicotinic acid, nicotinyl aldehyde
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/67Vitamins
    • A61K8/676Ascorbic acid, i.e. vitamin C
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin
    • A61Q19/02Preparations for care of the skin for chemically bleaching or whitening the skin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/40Chemical, physico-chemical or functional or structural properties of particular ingredients
    • A61K2800/59Mixtures
    • A61K2800/592Mixtures of compounds complementing their respective functions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/70Biological properties of the composition as a whole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/74Biological properties of particular ingredients
    • A61K2800/78Enzyme modulators, e.g. Enzyme agonists
    • A61K2800/782Enzyme inhibitors; Enzyme antagonists

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Birds (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Cosmetics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

1.- Una combinación que comprende por lo menos un antagonista del receptor de MC1-R, un inhibidor de tirosinasa derivado de vitamina C y un inhibidor de transferencia de melanosoma a los queratinocitos, caracterizada porque el antagonista del receptor de MC1-R es MELANOSTATINE® 5. 2.- La combinación de acuerdo con la reivindicación 1, caracterizada porque el inhibidor de tirosinasa derivado de vitamina C es 2-glucósido de ácido ascórbico. 3.- La combinación de acuerdo con cualquiera de las reivindicaciones anteriores, caracterizada porque el inhibidor de transferencia de melanosoma a los queratinocitos es nicotinamida. 4.- Una composición cosmética y/o dermatológica que comprende una combinación de acuerdo con cualquiera de las reivindicaciones anteriores en un portador cosmética o dermatológicamente aceptable. 5.- La composición cosmética y/o dermatológica de acuerdo con la reivindicación 4, caracterizada porque comprende: - 0.01% a 5% de inhibidor de transferencia de melanosoma, - 0.01% a 5% de inhibidor de tirosinasa derivado de vitamina C, - 0.1 a 40 ppm de antagonista del receptor de MC1-R. 6.- La composición cosmética y/o dermatológica de acuerdo con la reivindicación 5, caracterizada porque comprende: - 0.01% a 5% de niconamida, - 0.01% a 5% de 2-glucósido de ácido ascórbico, - 0.1 a 40 ppm de MELANOSTATINE®.7.- El uso cosmético de una composición de acuerdo con cualquiera de las reivindicaciones 4 a 6, para prevenir y/o tratar la aparición de pigmentación excesiva de la piel y/o brotes corporales superficiales.
CO09074062A 2007-01-16 2009-07-16 Asociacion de compuestos inhibidores de melanogenesis y su uso en cosmeticos y dermatologia CO6210733A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0700279A FR2911280B1 (fr) 2007-01-16 2007-01-16 Association de composes inhibiteurs de la melanogenese et leurs utilisations en cosmetique et en dermatologie

Publications (1)

Publication Number Publication Date
CO6210733A2 true CO6210733A2 (es) 2010-10-20

Family

ID=38472980

Family Applications (1)

Application Number Title Priority Date Filing Date
CO09074062A CO6210733A2 (es) 2007-01-16 2009-07-16 Asociacion de compuestos inhibidores de melanogenesis y su uso en cosmeticos y dermatologia

Country Status (16)

Country Link
US (1) US20100055059A1 (es)
EP (1) EP2109440B1 (es)
JP (1) JP5358456B2 (es)
CN (1) CN101631532A (es)
BR (1) BRPI0806775B1 (es)
CA (1) CA2675463A1 (es)
CO (1) CO6210733A2 (es)
EA (1) EA016034B1 (es)
FR (1) FR2911280B1 (es)
IL (1) IL199830A0 (es)
MA (1) MA31083B1 (es)
MX (1) MX2009007575A (es)
MY (1) MY162582A (es)
TN (1) TN2009000297A1 (es)
WO (1) WO2008107533A2 (es)
ZA (1) ZA200904399B (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101389529B1 (ko) 2012-02-03 2014-04-29 주식회사 스킨앤테크 가용화된 4-메톡시칼콘을 함유하는 피부 미백 조성물 및 이의 제조방법
WO2014088296A1 (ko) * 2012-12-04 2014-06-12 재단법인 경기과학기술진흥원 산유자 추출물을 이용한 피부 미백용 조성물
EP2969030B1 (en) * 2013-03-12 2021-01-13 Avon Products, Inc. A topical lightening composition and methods of use thereof
EP2875806A1 (en) 2013-11-20 2015-05-27 Infinitec Activos, S.L. Targeted capsules for the delivery of whitening agents in the skin
JP6820645B2 (ja) * 2014-02-26 2021-01-27 共栄化学工業株式会社 美白用組成物及び化粧料
US9949913B2 (en) * 2016-03-14 2018-04-24 Jan Marini Skin Research Luminate face lotion
CN108324590A (zh) * 2018-05-17 2018-07-27 云南白药清逸堂实业有限公司 一种美白护理液及其制备方法
EP3599046A1 (de) 2018-07-27 2020-01-29 FRONIUS INTERNATIONAL GmbH Lichtbogenschweissverfahren mit einem abschmelzenden schweissdraht
JP2021004215A (ja) * 2019-06-27 2021-01-14 小林製薬株式会社 Mc1r発現抑制剤
CN111450250A (zh) * 2020-03-12 2020-07-28 中南大学湘雅三医院 Enst00000606533的增强剂或抑制剂在制备治疗色素性皮肤病药物中的应用
FR3137284A1 (fr) * 2022-06-29 2024-01-05 Laboratoires Nigy Composition pour la prevention et le traitement de l’hyperpigmentation de la peau a base de niacinamide ou de l’un de ses derives et d’un extrait d’algue cystoseira

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006102289A2 (en) * 2005-03-23 2006-09-28 Mary Kay Inc. Skin lightening compositions
US20060263309A1 (en) * 2005-05-17 2006-11-23 Bissett Donald L Regulation of mammalian keratinous tissue using personal care compositions comprising tetrahydrocurcumin
US9265792B2 (en) * 2005-11-16 2016-02-23 Patricia A. Riley Integument cell regeneration formulation

Also Published As

Publication number Publication date
EA200970688A1 (ru) 2009-12-30
BRPI0806775B1 (pt) 2016-12-06
JP5358456B2 (ja) 2013-12-04
TN2009000297A1 (fr) 2010-12-31
ZA200904399B (en) 2010-07-28
WO2008107533A2 (fr) 2008-09-12
FR2911280A1 (fr) 2008-07-18
FR2911280B1 (fr) 2012-06-22
MA31083B1 (fr) 2010-01-04
CA2675463A1 (fr) 2008-09-12
JP2010515768A (ja) 2010-05-13
MX2009007575A (es) 2009-07-22
EA016034B1 (ru) 2012-01-30
EP2109440B1 (fr) 2016-01-13
IL199830A0 (en) 2010-04-15
BRPI0806775A2 (pt) 2011-09-13
WO2008107533A3 (fr) 2009-04-09
CN101631532A (zh) 2010-01-20
EP2109440A2 (fr) 2009-10-21
MY162582A (en) 2017-06-30
US20100055059A1 (en) 2010-03-04

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