CO2024010803A2 - Compuestos de tienopirrolotriazina, su preparación y su uso terapéutico - Google Patents

Compuestos de tienopirrolotriazina, su preparación y su uso terapéutico

Info

Publication number
CO2024010803A2
CO2024010803A2 CONC2024/0010803A CO2024010803A CO2024010803A2 CO 2024010803 A2 CO2024010803 A2 CO 2024010803A2 CO 2024010803 A CO2024010803 A CO 2024010803A CO 2024010803 A2 CO2024010803 A2 CO 2024010803A2
Authority
CO
Colombia
Prior art keywords
thienopyrrolotriazine
compounds
preparation
therapeutic use
formula
Prior art date
Application number
CONC2024/0010803A
Other languages
English (en)
Spanish (es)
Inventor
Olivier Arnoud
Franck Caussanel
Rommel Dadji-Faihun
Gwladys Langot
Frank Marguet
Olivier Venier
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of CO2024010803A2 publication Critical patent/CO2024010803A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CONC2024/0010803A 2022-02-21 2024-08-08 Compuestos de tienopirrolotriazina, su preparación y su uso terapéutico CO2024010803A2 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP22315036 2022-02-21
PCT/EP2023/054138 WO2023156643A1 (en) 2022-02-21 2023-02-20 Thienopyrrolotriazine compounds, their preparation and their therapeutic use

Publications (1)

Publication Number Publication Date
CO2024010803A2 true CO2024010803A2 (es) 2024-08-20

Family

ID=81326677

Family Applications (1)

Application Number Title Priority Date Filing Date
CONC2024/0010803A CO2024010803A2 (es) 2022-02-21 2024-08-08 Compuestos de tienopirrolotriazina, su preparación y su uso terapéutico

Country Status (11)

Country Link
US (1) US20250129091A1 (https=)
EP (1) EP4482841A1 (https=)
JP (1) JP2025506729A (https=)
KR (1) KR20240151767A (https=)
CN (1) CN118843632A (https=)
AU (1) AU2023222186A1 (https=)
CA (1) CA3244475A1 (https=)
CO (1) CO2024010803A2 (https=)
IL (1) IL314781A (https=)
MX (1) MX2024010216A (https=)
WO (1) WO2023156643A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116375728B (zh) * 2021-12-31 2025-06-10 成都赜灵生物医药科技有限公司 噻吩吡咯并三嗪酮类化合物及其用途
WO2025153532A1 (en) 2024-01-16 2025-07-24 NodThera Limited Nlrp3 inhibitors and glp-1 agonists combination therapies

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20210038877A (ko) * 2018-07-25 2021-04-08 노파르티스 아게 Nlrp3 인플라마좀 억제제
JP2023523418A (ja) * 2020-04-23 2023-06-05 ヤンセン ファーマシューティカ エヌ.ベー. Nlrp3の阻害剤としての三環式化合物

Also Published As

Publication number Publication date
IL314781A (en) 2024-10-01
KR20240151767A (ko) 2024-10-18
US20250129091A1 (en) 2025-04-24
JP2025506729A (ja) 2025-03-13
MX2024010216A (es) 2024-09-02
CN118843632A (zh) 2024-10-25
EP4482841A1 (en) 2025-01-01
CA3244475A1 (en) 2023-08-24
WO2023156643A1 (en) 2023-08-24
AU2023222186A1 (en) 2024-10-10

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