CN1658873A - 基于抗胆碱能剂和p38激酶抑制剂的新颖药物组合物 - Google Patents

基于抗胆碱能剂和p38激酶抑制剂的新颖药物组合物 Download PDF

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Publication number
CN1658873A
CN1658873A CN038134217A CN03813421A CN1658873A CN 1658873 A CN1658873 A CN 1658873A CN 038134217 A CN038134217 A CN 038134217A CN 03813421 A CN03813421 A CN 03813421A CN 1658873 A CN1658873 A CN 1658873A
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alkyl
amino
group
phenyl
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CN038134217A
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Chinese (zh)
Inventor
伯吉特·琼
米歇尔·佩雷特
迈克尔·P·皮珀
汉斯·C·赖泽
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Boehringer Ingelheim Pharma GmbH and Co KG
Boehringer Ingelheim Pharmaceuticals Inc
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Boehringer Ingelheim Pharma GmbH and Co KG
Boehringer Ingelheim Pharmaceuticals Inc
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Publication of CN1658873A publication Critical patent/CN1658873A/zh
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    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/007—Pulmonary tract; Aromatherapy
    • A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/537—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines spiro-condensed or forming part of bridged ring systems
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    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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  • Otolaryngology (AREA)
  • Emergency Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
CN038134217A 2002-04-10 2003-04-08 基于抗胆碱能剂和p38激酶抑制剂的新颖药物组合物 Pending CN1658873A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US37151402P 2002-04-10 2002-04-10
US60/371,514 2002-04-10

Publications (1)

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CN1658873A true CN1658873A (zh) 2005-08-24

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US (1) US20030225089A1 (enExample)
EP (1) EP1496900A2 (enExample)
JP (1) JP2005529098A (enExample)
KR (1) KR20050006149A (enExample)
CN (1) CN1658873A (enExample)
AR (1) AR039273A1 (enExample)
AU (1) AU2003224048A1 (enExample)
BR (1) BR0309099A (enExample)
CA (1) CA2479522A1 (enExample)
MX (1) MXPA04009772A (enExample)
PE (1) PE20040325A1 (enExample)
PL (1) PL372620A1 (enExample)
RU (1) RU2004133034A (enExample)
TW (1) TW200307681A (enExample)
UY (1) UY27755A1 (enExample)
WO (1) WO2003084539A2 (enExample)
ZA (1) ZA200407058B (enExample)

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BR0309099A (pt) 2005-03-29
RU2004133034A (ru) 2006-06-20
PL372620A1 (en) 2005-07-25
KR20050006149A (ko) 2005-01-15
MXPA04009772A (es) 2004-12-13
TW200307681A (en) 2003-12-16
AR039273A1 (es) 2005-02-16
WO2003084539A3 (en) 2004-09-02
PE20040325A1 (es) 2004-07-08
EP1496900A2 (en) 2005-01-19
JP2005529098A (ja) 2005-09-29
WO2003084539A2 (en) 2003-10-16
CA2479522A1 (en) 2003-10-16
US20030225089A1 (en) 2003-12-04
UY27755A1 (es) 2003-11-28
AU2003224048A1 (en) 2003-10-20

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