CN1328272C - 一种工业化生产霉酚酸莫啡酯的方法 - Google Patents
一种工业化生产霉酚酸莫啡酯的方法 Download PDFInfo
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- CN1328272C CN1328272C CNB200510044285XA CN200510044285A CN1328272C CN 1328272 C CN1328272 C CN 1328272C CN B200510044285X A CNB200510044285X A CN B200510044285XA CN 200510044285 A CN200510044285 A CN 200510044285A CN 1328272 C CN1328272 C CN 1328272C
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- mycophenolic acid
- reaction
- morpholino ethanol
- acid
- industrial production
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- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
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Priority Applications (1)
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CNB200510044285XA CN1328272C (zh) | 2005-08-22 | 2005-08-22 | 一种工业化生产霉酚酸莫啡酯的方法 |
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CNB200510044285XA CN1328272C (zh) | 2005-08-22 | 2005-08-22 | 一种工业化生产霉酚酸莫啡酯的方法 |
Publications (2)
Publication Number | Publication Date |
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CN1733749A CN1733749A (zh) | 2006-02-15 |
CN1328272C true CN1328272C (zh) | 2007-07-25 |
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CNB200510044285XA Active CN1328272C (zh) | 2005-08-22 | 2005-08-22 | 一种工业化生产霉酚酸莫啡酯的方法 |
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Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
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CN1974564B (zh) * | 2006-12-15 | 2010-05-12 | 丽珠集团新北江制药股份有限公司 | 一种霉酚酸莫啡酯的制备方法 |
CN100484930C (zh) * | 2007-03-16 | 2009-05-06 | 重庆大新药业股份有限公司 | 一种吗替麦考酚酯的制备方法 |
CN103265514B (zh) * | 2013-06-08 | 2016-01-13 | 重庆理工大学 | 一种制备吗替麦考酚酯的方法 |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5247083A (en) * | 1992-07-10 | 1993-09-21 | Syntex (U.S.A.) Inc. | Direct esterification of mycophenolic acid |
US6709846B1 (en) * | 1998-12-09 | 2004-03-23 | Biocon India Limited | Methods of producing esters of mycophenolate |
CN1520411A (zh) * | 2001-06-08 | 2004-08-11 | ����˹��ҩ�﹫˾ | 霉酚酸莫啡酯的制备方法 |
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2005
- 2005-08-22 CN CNB200510044285XA patent/CN1328272C/zh active Active
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5247083A (en) * | 1992-07-10 | 1993-09-21 | Syntex (U.S.A.) Inc. | Direct esterification of mycophenolic acid |
US6709846B1 (en) * | 1998-12-09 | 2004-03-23 | Biocon India Limited | Methods of producing esters of mycophenolate |
CN1520411A (zh) * | 2001-06-08 | 2004-08-11 | ����˹��ҩ�﹫˾ | 霉酚酸莫啡酯的制备方法 |
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CN1733749A (zh) | 2006-02-15 |
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Date | Code | Title | Description |
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C06 | Publication | ||
PB01 | Publication | ||
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SE01 | Entry into force of request for substantive examination | ||
C14 | Grant of patent or utility model | ||
GR01 | Patent grant | ||
EE01 | Entry into force of recordation of patent licensing contract |
Assignee: Shandong Xinshidai Pharmaceutical Industry Co., Ltd. Assignor: Lunan Pharmaceutical Group Co., Ltd. Contract record no.: 2010370000508 Denomination of invention: Industrial production method of mycophenolic acid morpholine ester Granted publication date: 20070725 License type: Exclusive License Open date: 20060215 Record date: 20100908 |
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EC01 | Cancellation of recordation of patent licensing contract |
Assignee: Shandong Xinshidai Pharmaceutical Industry Co., Ltd. Assignor: Lunan Pharmaceutical Group Co., Ltd. Contract record no.: 2010370000508 Date of cancellation: 20121226 |
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EE01 | Entry into force of recordation of patent licensing contract |
Application publication date: 20060215 Assignee: Lunan New Era Biological Technology Co., Ltd. Assignor: Lunan Pharmaceutical Group Co., Ltd. Contract record no.: 2012370000303 Denomination of invention: Industrial production method of mycophenolic acid morpholine ester Granted publication date: 20070725 License type: Exclusive License Record date: 20121226 |
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LICC | Enforcement, change and cancellation of record of contracts on the licence for exploitation of a patent or utility model |