CN1325838A - 制备间苯二酚衍生物的方法 - Google Patents

制备间苯二酚衍生物的方法 Download PDF

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Publication number
CN1325838A
CN1325838A CN01119693A CN01119693A CN1325838A CN 1325838 A CN1325838 A CN 1325838A CN 01119693 A CN01119693 A CN 01119693A CN 01119693 A CN01119693 A CN 01119693A CN 1325838 A CN1325838 A CN 1325838A
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CN
China
Prior art keywords
alkyl
aryl
formula
compound
acyl
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Pending
Application number
CN01119693A
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English (en)
Chinese (zh)
Inventor
S·E·布莱德利
J·基钦
G·M·温尼
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Pfizer Products Inc
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Pfizer Products Inc
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Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc
Publication of CN1325838A publication Critical patent/CN1325838A/zh
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C37/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring
    • C07C37/06—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring by conversion of non-aromatic six-membered rings or of such rings formed in situ into aromatic six-membered rings, e.g. by dehydrogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/72—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 spiro-condensed with carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C37/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring
    • C07C37/06—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring by conversion of non-aromatic six-membered rings or of such rings formed in situ into aromatic six-membered rings, e.g. by dehydrogenation
    • C07C37/07—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring by conversion of non-aromatic six-membered rings or of such rings formed in situ into aromatic six-membered rings, e.g. by dehydrogenation with simultaneous reduction of C=O group in that ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/56—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds
    • C07C45/57—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with oxygen as the only heteroatom
    • C07C45/59—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with oxygen as the only heteroatom in five-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/70—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form
    • C07C45/71—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form being hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/703—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups
    • C07C49/747—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/18—Systems containing only non-condensed rings with a ring being at least seven-membered
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S977/00—Nanotechnology
    • Y10S977/902—Specified use of nanostructure
    • Y10S977/904—Specified use of nanostructure for medical, immunological, body treatment, or diagnosis
    • Y10S977/926—Topical chemical, e.g. cosmetic or sunscreen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
CN01119693A 2000-03-15 2001-03-15 制备间苯二酚衍生物的方法 Pending CN1325838A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US18970400P 2000-03-15 2000-03-15
US60/189,704 2000-03-15

Publications (1)

Publication Number Publication Date
CN1325838A true CN1325838A (zh) 2001-12-12

Family

ID=22698426

Family Applications (1)

Application Number Title Priority Date Filing Date
CN01119693A Pending CN1325838A (zh) 2000-03-15 2001-03-15 制备间苯二酚衍生物的方法

Country Status (18)

Country Link
US (3) US6504037B2 (enExample)
EP (1) EP1134207A1 (enExample)
JP (1) JP2001294549A (enExample)
KR (1) KR100432303B1 (enExample)
CN (1) CN1325838A (enExample)
AR (1) AR030055A1 (enExample)
AU (1) AU782397B2 (enExample)
BR (1) BR0100982A (enExample)
CA (1) CA2340486A1 (enExample)
CZ (1) CZ2001930A3 (enExample)
HK (1) HK1040987A1 (enExample)
ID (1) ID29673A (enExample)
IL (1) IL141915A0 (enExample)
IN (1) IN192530B (enExample)
PL (1) PL346463A1 (enExample)
RU (1) RU2213087C2 (enExample)
YU (1) YU18601A (enExample)
ZA (1) ZA200102070B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1293857C (zh) * 2002-03-22 2007-01-10 荷兰联合利华有限公司 间苯二酚衍生物在化妆品组合物中的稳定

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6828460B2 (en) * 1999-03-22 2004-12-07 Pfizer Inc. Resorcinol derivatives
JP4228605B2 (ja) 2002-07-02 2009-02-25 住友化学株式会社 改変型還元酵素、その遺伝子及びそれらの利用
JP4228606B2 (ja) 2002-07-03 2009-02-25 住友化学株式会社 改変型還元酵素、その遺伝子及びそれらの利用
US6852310B2 (en) 2002-08-23 2005-02-08 Unilever Home & Personal Care Usa Division Of Conopco, Inc. Skin lightening agents, compositions and methods
CN100383573C (zh) * 2002-12-02 2008-04-23 3M创新有限公司 多光源照明系统
US6875425B2 (en) 2002-12-12 2005-04-05 Unilever Home & Personal Care Usa Skin lightening agents, compositions and methods
US7524485B2 (en) 2002-12-12 2009-04-28 Unilever Home & Personal Care, Usa, Division Of Conopco, Inc. Skin lightening agents, compositions and methods
US7338979B2 (en) 2003-02-11 2008-03-04 Warner-Lambert Company Depigmentation agents
US7300646B2 (en) 2004-02-27 2007-11-27 Unilever Home & Personal Care Usa, Division Of Conopco, Inc. Skin lightening agents, compositions and methods
US20060062865A1 (en) * 2004-09-17 2006-03-23 Nebojsa Ilic Tyrosinase inhibitor and method for preparation
US20060210497A1 (en) * 2005-03-18 2006-09-21 Unilever Home & Personal Care Usa, Division Of Conopco, Inc. Novel resorcinol derivatives
US20060210498A1 (en) * 2005-03-18 2006-09-21 Unilever Home & Personal Care Usa, Division Of Conopco, Inc. Novel resorcinol derivatives for skin
US7250158B1 (en) 2006-03-30 2007-07-31 Conopco, Inc. Skin lightening agents, compositions and methods
US7247294B1 (en) 2006-03-30 2007-07-24 Conopco, Inc. Skin lightening agents, compositions and methods
US7270805B1 (en) 2006-03-30 2007-09-18 Conopco, Inc. Skin lightening agents, compositions and methods
EP2964182B1 (en) 2013-03-08 2018-02-14 Unilever PLC, a company registered in England and Wales under company no. 41424 of Resorcinol compounds for dermatological use
WO2017215863A1 (en) 2016-06-15 2017-12-21 Unilever N.V. Method and cosmetic composition for enhanced transdermal delivery of alkyl substituted resorcinol
CN111909012B (zh) * 2020-08-24 2022-10-21 浙江工业大学台州研究院 一种高选择性、高转化制备1,3-环己二酮的方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0651619B2 (ja) * 1988-05-09 1994-07-06 株式会社クラレ 美白剤
US5059438A (en) * 1990-02-05 1991-10-22 Enzytech, Inc. Compositions and methods for inhibiting browning in foods using resorcinol derivatives
FR2704753B1 (fr) * 1993-05-06 1995-06-30 Oreal Utilisation de derives de la 4-thio resorcine ou 4-thio 1-3-dihydroxybenzene, dans des compositions cosmetiques ou dermopharmaceutiques a action depigmentante.
FR2714601B1 (fr) * 1993-12-30 1996-02-09 Oreal Composition dépigmentante pour le traitement simultané des couches superficielles et profondes, son utilisation.
BR9803596A (pt) * 1997-09-23 2000-04-25 Pfizer Prod Inc Derivados do resorcinol.
PA8469601A1 (es) * 1998-04-10 2000-09-29 Pfizer Prod Inc Procedimiento para alquilar sulfonamidas impedidas estericamente
SI1165495T1 (en) * 1999-03-22 2005-08-31 Pfizer Resorcinol derivatives

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1293857C (zh) * 2002-03-22 2007-01-10 荷兰联合利华有限公司 间苯二酚衍生物在化妆品组合物中的稳定

Also Published As

Publication number Publication date
AU2647701A (en) 2001-09-20
AU782397B2 (en) 2005-07-21
IN192530B (enExample) 2004-04-24
US20050143594A1 (en) 2005-06-30
ID29673A (id) 2001-09-20
US6861564B2 (en) 2005-03-01
US20030088113A1 (en) 2003-05-08
CA2340486A1 (en) 2001-09-15
BR0100982A (pt) 2001-12-04
KR20010096608A (ko) 2001-11-07
US6504037B2 (en) 2003-01-07
IL141915A0 (en) 2002-03-10
AR030055A1 (es) 2003-08-13
KR100432303B1 (ko) 2004-05-20
YU18601A (sh) 2003-07-07
RU2213087C2 (ru) 2003-09-27
HK1040987A1 (zh) 2002-06-28
US20020032352A1 (en) 2002-03-14
PL346463A1 (en) 2001-09-24
EP1134207A1 (en) 2001-09-19
JP2001294549A (ja) 2001-10-23
CZ2001930A3 (cs) 2001-10-17
ZA200102070B (en) 2002-09-13

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