CN1248692C - 玻璃体结合蛋白受体拮抗剂在制备用于抑制粘连形成的药物中的用途 - Google Patents
玻璃体结合蛋白受体拮抗剂在制备用于抑制粘连形成的药物中的用途 Download PDFInfo
- Publication number
- CN1248692C CN1248692C CNB028097874A CN02809787A CN1248692C CN 1248692 C CN1248692 C CN 1248692C CN B028097874 A CNB028097874 A CN B028097874A CN 02809787 A CN02809787 A CN 02809787A CN 1248692 C CN1248692 C CN 1248692C
- Authority
- CN
- China
- Prior art keywords
- alkyl
- adhesion
- compound
- adhesions
- adhesion formation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P41/00—Drugs used in surgical methods, e.g. surgery adjuvants for preventing adhesion or for vitreum substitution
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US28269301P | 2001-04-10 | 2001-04-10 | |
| US60/282,693 | 2001-04-10 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN1509170A CN1509170A (zh) | 2004-06-30 |
| CN1248692C true CN1248692C (zh) | 2006-04-05 |
Family
ID=23082703
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNB028097874A Expired - Fee Related CN1248692C (zh) | 2001-04-10 | 2002-04-10 | 玻璃体结合蛋白受体拮抗剂在制备用于抑制粘连形成的药物中的用途 |
Country Status (26)
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR052823A1 (es) * | 2004-12-21 | 2007-04-04 | Smithkline Beecham Corp | Uso de un antagonista del receptor de vitronectina para l a preparacion de una formulacion farmaceutica util para inhibir el exceso de formacion de cicatrices en la piel de a un mamifero y dicha formulacion |
| RU2744540C1 (ru) * | 2020-02-18 | 2021-03-11 | Федеральное государственное бюджетное образовательное учреждение высшего образования "Курский государственный медицинский университет" Министерства здравоохранения Российской Федерации | Способ профилактики спаечного процесса при операциях на брюшной полости в условиях паренхиматозного кровотечения в эксперименте |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA60311C2 (uk) * | 1996-10-02 | 2003-10-15 | Смітклайн Бічам Корпорейшн | Антагоністи рецептора вітронектину, спосіб одержання цих сполук та фармацевтична композиція |
-
2002
- 2002-04-10 WO PCT/US2002/011285 patent/WO2002083125A1/en not_active Ceased
- 2002-04-10 HU HU0303725A patent/HUP0303725A3/hu unknown
- 2002-04-10 CA CA002443734A patent/CA2443734A1/en not_active Abandoned
- 2002-04-10 KR KR10-2003-7013214A patent/KR20030087069A/ko not_active Abandoned
- 2002-04-10 MX MXPA03009344A patent/MXPA03009344A/es active IP Right Grant
- 2002-04-10 CZ CZ20032767A patent/CZ20032767A3/cs unknown
- 2002-04-10 CN CNB028097874A patent/CN1248692C/zh not_active Expired - Fee Related
- 2002-04-10 IL IL15827202A patent/IL158272A0/xx unknown
- 2002-04-10 EA EA200301109A patent/EA006202B1/ru not_active IP Right Cessation
- 2002-04-10 NZ NZ528577A patent/NZ528577A/en unknown
- 2002-04-10 PL PL02364526A patent/PL364526A1/xx not_active Application Discontinuation
- 2002-04-10 BR BR0208789-8A patent/BR0208789A/pt not_active IP Right Cessation
- 2002-04-10 DE DE60230404T patent/DE60230404D1/de not_active Expired - Lifetime
- 2002-04-10 AT AT02733968T patent/ATE417612T1/de not_active IP Right Cessation
- 2002-04-10 AU AU2002305164A patent/AU2002305164B2/en not_active Ceased
- 2002-04-10 ES ES02733968T patent/ES2319877T3/es not_active Expired - Lifetime
- 2002-04-10 JP JP2002580929A patent/JP4394882B2/ja not_active Expired - Fee Related
- 2002-04-10 OA OA1200300271A patent/OA12505A/en unknown
- 2002-04-10 AP APAP/P/2003/002894A patent/AP2003002894A0/en unknown
- 2002-04-10 EP EP02733968A patent/EP1385504B1/en not_active Expired - Lifetime
- 2002-10-04 UA UA2003109182A patent/UA75395C2/uk unknown
-
2003
- 2003-09-30 ZA ZA200307621A patent/ZA200307621B/en unknown
- 2003-10-01 BG BG108217A patent/BG108217A/bg unknown
- 2003-10-06 MA MA27339A patent/MA26159A1/fr unknown
- 2003-10-08 NO NO20034513A patent/NO20034513L/no not_active Application Discontinuation
- 2003-10-09 EC EC2003004799A patent/ECSP034799A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| UA75395C2 (en) | 2006-04-17 |
| KR20030087069A (ko) | 2003-11-12 |
| EP1385504B1 (en) | 2008-12-17 |
| EA006202B1 (ru) | 2005-10-27 |
| BR0208789A (pt) | 2004-03-09 |
| ZA200307621B (en) | 2004-04-21 |
| HUP0303725A3 (en) | 2009-08-28 |
| ES2319877T3 (es) | 2009-05-14 |
| IL158272A0 (en) | 2004-05-12 |
| CN1509170A (zh) | 2004-06-30 |
| NZ528577A (en) | 2005-01-28 |
| MXPA03009344A (es) | 2004-02-12 |
| JP4394882B2 (ja) | 2010-01-06 |
| AP2003002894A0 (en) | 2003-12-31 |
| AU2002305164B2 (en) | 2005-07-28 |
| DE60230404D1 (cg-RX-API-DMAC7.html) | 2009-01-29 |
| CZ20032767A3 (cs) | 2004-12-15 |
| HUP0303725A2 (hu) | 2004-03-01 |
| EA200301109A1 (ru) | 2004-02-26 |
| OA12505A (en) | 2006-05-29 |
| BG108217A (bg) | 2004-12-30 |
| ECSP034799A (es) | 2004-01-28 |
| EP1385504A4 (en) | 2007-03-14 |
| CA2443734A1 (en) | 2002-10-24 |
| PL364526A1 (en) | 2004-12-13 |
| EP1385504A1 (en) | 2004-02-04 |
| NO20034513L (no) | 2003-12-04 |
| ATE417612T1 (de) | 2009-01-15 |
| MA26159A1 (fr) | 2004-07-01 |
| NO20034513D0 (no) | 2003-10-08 |
| WO2002083125A1 (en) | 2002-10-24 |
| JP2004525959A (ja) | 2004-08-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| C06 | Publication | ||
| PB01 | Publication | ||
| C10 | Entry into substantive examination | ||
| SE01 | Entry into force of request for substantive examination | ||
| C14 | Grant of patent or utility model | ||
| GR01 | Patent grant | ||
| C17 | Cessation of patent right | ||
| CF01 | Termination of patent right due to non-payment of annual fee |
Granted publication date: 20060405 |