CN116836178A - 噻吩衍生物的晶型 - Google Patents
噻吩衍生物的晶型 Download PDFInfo
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- CN116836178A CN116836178A CN202310701814.7A CN202310701814A CN116836178A CN 116836178 A CN116836178 A CN 116836178A CN 202310701814 A CN202310701814 A CN 202310701814A CN 116836178 A CN116836178 A CN 116836178A
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- Prior art keywords
- methoxyphenyl
- ethoxy
- pyrrol
- acetamide
- ethyl
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Landscapes
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| WO2025103428A1 (zh) * | 2023-11-14 | 2025-05-22 | 赣州和美药业股份有限公司 | 中重度斑块型银屑病的治疗 |
Citations (4)
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| CN101885731A (zh) * | 2009-05-14 | 2010-11-17 | 天津和美生物技术有限公司 | 噻吩衍生物 |
| JP2017521500A (ja) * | 2014-07-18 | 2017-08-03 | グリーン・クロス・コーポレイションＧｒｅｅｎ Ｃｒｏｓｓ Ｃｏｒｐ． | ５−クロロ−ｎ−（｛（５ｓ）−２−オキソ−３−［４−（５，６−ジヒドロ−４ｈ−［１，２，４］トリアジン−１−イル）フェニル］−１，３−オキサゾリジン−５−イル｝メチル）チオフェン−２−カルボキシアミド メタンスルホネートの新規結晶形態および前記結晶形態を含む医薬組成物 |
| US20180354967A1 (en) * | 2017-06-13 | 2018-12-13 | Biotheryx, Inc. | Bicylic compounds and methods of use |
| CN110437251B (zh) * | 2018-05-02 | 2023-07-21 | 天津合美医药科技有限公司 | 噻吩衍生物的晶型 |
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| US6020358A (en) | 1998-10-30 | 2000-02-01 | Celgene Corporation | Substituted phenethylsulfones and method of reducing TNFα levels |
| WO2003091260A1 (en) * | 2002-04-23 | 2003-11-06 | Dr. Reddy's Laboratories Limited | Novel crystalline polymorph form-vi of olanzapine and a process for preparation thereof |
| CN101186612B (zh) | 2006-11-15 | 2012-10-03 | 天津和美生物技术有限公司 | 可抑制细胞释放肿瘤坏死因子的吡咯啉衍生物及其制备和应用 |
| JP5968881B2 (ja) * | 2010-06-30 | 2016-08-10 | レオ ファーマ アクティーゼルスカブ | カルシウム模倣化合物の新規多形 |
| WO2015082583A1 (en) * | 2013-12-05 | 2015-06-11 | F. Hoffmann-La Roche Ag | Heteroaryl pyridone and aza-pyridone compounds with electrophilic functionality |
| EP3144393A1 (en) * | 2015-09-18 | 2017-03-22 | LEK Pharmaceuticals d.d. | A synthetic pathway towards apremilast |
| CN107417626B (zh) * | 2016-05-23 | 2020-01-24 | 江苏奥赛康药业有限公司 | 一种2-氨基嘧啶类化合物的多晶型形式 |
| CN107474057B (zh) * | 2016-06-07 | 2021-03-12 | 天津药物研究院有限公司 | (5-(2-腈基苄基)-4,5,6,7-四氢噻吩并[3,2-c]吡啶-2-基)乙酸酯盐酸盐的晶型及其制备方法和用途 |
| JP7074782B2 (ja) * | 2017-06-30 | 2022-05-24 | トロフィー エスアーエス | 患者位置決めアクセサリ検出を伴う口腔外歯科用撮像装置 |
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| CN101885731A (zh) * | 2009-05-14 | 2010-11-17 | 天津和美生物技术有限公司 | 噻吩衍生物 |
| JP2017521500A (ja) * | 2014-07-18 | 2017-08-03 | グリーン・クロス・コーポレイションＧｒｅｅｎ Ｃｒｏｓｓ Ｃｏｒｐ． | ５−クロロ−ｎ−（｛（５ｓ）−２−オキソ−３−［４−（５，６−ジヒドロ−４ｈ−［１，２，４］トリアジン−１−イル）フェニル］−１，３−オキサゾリジン−５−イル｝メチル）チオフェン−２−カルボキシアミド メタンスルホネートの新規結晶形態および前記結晶形態を含む医薬組成物 |
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