CN115103670A - 转录增强相关结构域(tead)转录因子抑制剂及其用途 - Google Patents

转录增强相关结构域(tead)转录因子抑制剂及其用途 Download PDF

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CN115103670A
CN115103670A CN202080096940.9A CN202080096940A CN115103670A CN 115103670 A CN115103670 A CN 115103670A CN 202080096940 A CN202080096940 A CN 202080096940A CN 115103670 A CN115103670 A CN 115103670A
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optionally substituted
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alkyl
formula
cancer
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N.S.格雷
T.张
J.车
N.P.奎亚特科夫斯基
M.范
W.卢
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Dana Farber Cancer Institute Inc
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    • C07C311/38Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring having sulfur atoms of sulfonamide groups and amino groups bound to carbon atoms of six-membered rings of the same carbon skeleton
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CN202080096940.9A 2019-12-24 2020-12-23 转录增强相关结构域(tead)转录因子抑制剂及其用途 Pending CN115103670A (zh)

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Cited By (8)

* Cited by examiner, † Cited by third party
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CN116287270A (zh) * 2023-03-17 2023-06-23 复旦大学附属中山医院 Klf11在检测肺腺癌铁死亡和化疗敏感性中的应用
CN116535379A (zh) * 2023-06-29 2023-08-04 希格生科(深圳)有限公司 化合物及其医药用途
CN117487816A (zh) * 2023-11-03 2024-02-02 中山大学孙逸仙纪念医院 Znf709基因在制备治疗pbc的药物中的应用
CN117625791A (zh) * 2024-01-23 2024-03-01 杭州华得森生物技术有限公司 用于结直肠癌诊断和预后判断的生物标志物及其应用
WO2024120519A1 (zh) * 2022-12-09 2024-06-13 捷思英达控股有限公司 Tead抑制剂、其制备方法和在医学上的应用
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CN117625791B (zh) * 2024-01-23 2024-04-16 杭州华得森生物技术有限公司 用于结直肠癌诊断和预后判断的生物标志物及其应用
CN118584109A (zh) * 2024-03-26 2024-09-03 首都医科大学附属北京胸科医院 一种筛选耐药性肺癌的生物标志物
CN120624647A (zh) * 2025-05-30 2025-09-12 山西省肿瘤医院 鼻咽癌诊断或预测的甲基化标志物组合及应用、试剂盒和计算机可读存储介质
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