CN114286816B - 赖氨酰氧化酶的二氟卤代烯丙胺砜衍生物抑制剂、其制备方法和用途 - Google Patents

赖氨酰氧化酶的二氟卤代烯丙胺砜衍生物抑制剂、其制备方法和用途 Download PDF

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CN114286816B
CN114286816B CN202080060323.3A CN202080060323A CN114286816B CN 114286816 B CN114286816 B CN 114286816B CN 202080060323 A CN202080060323 A CN 202080060323A CN 114286816 B CN114286816 B CN 114286816B
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CN114286816A (zh
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D·W·汉佩特
艾莉森·桃乐丝·芬得利
克雷格·伊旺·特纳
曼达·迪奥达
A·E·格雷克
沃尔夫冈·杰洛利梅克
周文斌
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Pharmaxis Ltd
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CN202080060323.3A 2019-07-25 2020-07-24 赖氨酰氧化酶的二氟卤代烯丙胺砜衍生物抑制剂、其制备方法和用途 Active CN114286816B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
AU2019902641A AU2019902641A0 (en) 2019-07-25 Difluorohaloallylamine sulfone derivative inhibitors of lysyl oxidases, methods of preparation, and uses thereof
AU2019902641 2019-07-25
PCT/AU2020/050759 WO2021012014A1 (en) 2019-07-25 2020-07-24 Difluorohaloallylamine sulfone derivative inhibitors of lysyl oxidases, methods of preparation, and uses thereof

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CN114286816A CN114286816A (zh) 2022-04-05
CN114286816B true CN114286816B (zh) 2024-08-20

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WO2021261601A1 (ja) 2020-06-26 2021-12-30 ラクオリア創薬株式会社 レチノイドとがん治療薬との併用療法が有効ながん患者の選択方法およびレチノイドとがん治療薬との併用医薬
CN113440477B (zh) * 2021-08-12 2022-10-11 海南海神同洲制药有限公司 一种低粘度酮康唑乳膏及其制备方法
US12233056B2 (en) 2022-04-06 2025-02-25 Syntara Limited Lysyl oxidase inhibitors for treating myeloid malignancies
GB202209624D0 (en) 2022-06-30 2022-08-17 Institute Of Cancer Res Royal Cancer Hospital Prodrugs
GB202209622D0 (en) 2022-06-30 2022-08-17 Institute Of Cancer Res Royal Cancer Hospital Compounds

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EP3589619A4 (en) * 2017-03-02 2020-12-16 Pharmaxis Ltd. LYSYL OXIDASE INHIBITORS, HALOGENOALLYLAMINE PYRAZOLE DERIVATIVES AND THEIR USES
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JP2022544031A (ja) 2022-10-17
US20220251036A1 (en) 2022-08-11
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AU2020317374A1 (en) 2022-02-03
TW202114991A (zh) 2021-04-16
KR20220040480A (ko) 2022-03-30
MX2022001031A (es) 2022-02-23
CA3145738A1 (en) 2021-01-28
EP4003952A4 (en) 2023-08-23
BR112022000782A2 (pt) 2022-03-15
ZA202202376B (en) 2023-11-29
EP4003952A1 (en) 2022-06-01

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