CN112920193B - 一种灰黄霉素四唑衍生物及其制备方法 - Google Patents
一种灰黄霉素四唑衍生物及其制备方法 Download PDFInfo
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- CN112920193B CN112920193B CN202110169263.5A CN202110169263A CN112920193B CN 112920193 B CN112920193 B CN 112920193B CN 202110169263 A CN202110169263 A CN 202110169263A CN 112920193 B CN112920193 B CN 112920193B
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/20—Spiro-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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CN112933098B (zh) * | 2021-02-07 | 2021-10-26 | 南通大学 | 一种灰黄霉素四唑衍生物在制备抗肿瘤药物中的应用 |
CN113861144B (zh) * | 2021-08-04 | 2022-06-21 | 南通大学 | 一种灰黄霉素开环衍生物及其制备方法 |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
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CN102712606A (zh) * | 2009-11-17 | 2012-10-03 | 田边三菱制药株式会社 | 联苯基衍生物的制备方法 |
CN103635446A (zh) * | 2011-05-04 | 2014-03-12 | 巴兰斯医疗公司 | 戊四唑衍生物 |
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WO2019169389A1 (en) * | 2018-03-02 | 2019-09-06 | Epicentrx, Inc. | Methods and compositions for treating cancer and sensitizing tumor cells to kinase inhibitors |
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Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
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CN102712606A (zh) * | 2009-11-17 | 2012-10-03 | 田边三菱制药株式会社 | 联苯基衍生物的制备方法 |
CN103635446A (zh) * | 2011-05-04 | 2014-03-12 | 巴兰斯医疗公司 | 戊四唑衍生物 |
Non-Patent Citations (2)
Title |
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"Remodeling and Enhancing Schmidt Reaction Pathways in Hexafluoroisopropanol";Hashim F. Motiwala etal.;《Journal of Organic Chemistry》;20160122;第81卷;第1593-1609页 * |
"Synthesis and structure of azole-fused indeno[2,1-c]quinolines and their anti-mycobacterial properties";Ram Shankar Upadhayaya etal.;《Organic & Biomolecular Chemistry》;20101007;第8卷;第5661-5673页 * |
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Application publication date: 20210608 Assignee: NANTONG HAOYOU FOOD ADDITIVES Co.,Ltd. Assignor: NANTONG University Contract record no.: X2023320000032 Denomination of invention: A griseofulvin tetrazole derivative and its preparation method Granted publication date: 20211116 License type: Common License Record date: 20230111 |
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Effective date of registration: 20230816 Address after: 226000 Jiangsu city of Nantong province sik Road No. 9 Patentee after: Nantong University Technology Transfer Center Co.,Ltd. Address before: 226019 Jiangsu city of Nantong province sik Road No. 9 Patentee before: NANTONG University |
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