CN1086220A - 雄甾-4-烯酮[4，5-b]吡咯衍生物及制备方法 - Google Patents

雄甾-4-烯酮[4，5-b]吡咯衍生物及制备方法 Download PDF

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Publication number
CN1086220A
CN1086220A CN93109285A CN93109285A CN1086220A CN 1086220 A CN1086220 A CN 1086220A CN 93109285 A CN93109285 A CN 93109285A CN 93109285 A CN93109285 A CN 93109285A CN 1086220 A CN1086220 A CN 1086220A
Authority
CN
China
Prior art keywords
compound
general formula
logical formula
definition
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN93109285A
Other languages
English (en)
Chinese (zh)
Inventor
F·布泽蒂
A·隆格
E·D·萨勒
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL filed Critical Farmitalia Carlo Erba SRL
Publication of CN1086220A publication Critical patent/CN1086220A/zh
Pending legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0036—Nitrogen-containing hetero ring
    • C07J71/0042—Nitrogen only
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
    • C07J7/008—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms substituted in position 21
    • C07J7/0085—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms substituted in position 21 by an halogen atom

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Fats And Perfumes (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CN93109285A 1992-08-11 1993-08-10 雄甾-4-烯酮[4，5-b]吡咯衍生物及制备方法 Pending CN1086220A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB929217035A GB9217035D0 (en) 1992-08-11 1992-08-11 Androst-4-eno(4,5-b)pyrrole derivatives and process for their preparation
GB9217035.6 1992-08-11

Publications (1)

Publication Number Publication Date
CN1086220A true CN1086220A (zh) 1994-05-04

Family

ID=10720180

Family Applications (1)

Application Number Title Priority Date Filing Date
CN93109285A Pending CN1086220A (zh) 1992-08-11 1993-08-10 雄甾-4-烯酮[4，5-b]吡咯衍生物及制备方法

Country Status (21)

Country Link
US (1) US5457097A (https=)
EP (1) EP0608404B1 (https=)
JP (1) JPH07500119A (https=)
CN (1) CN1086220A (https=)
AT (1) ATE136036T1 (https=)
AU (1) AU662077B2 (https=)
CA (1) CA2120726A1 (https=)
DE (1) DE69302007T2 (https=)
DK (1) DK0608404T3 (https=)
ES (1) ES2088289T3 (https=)
FI (1) FI941635A0 (https=)
GB (1) GB9217035D0 (https=)
GR (1) GR3019729T3 (https=)
HU (1) HUT67662A (https=)
IL (1) IL106597A (https=)
MX (1) MX9304852A (https=)
MY (1) MY108957A (https=)
NZ (1) NZ254805A (https=)
TW (1) TW276257B (https=)
WO (1) WO1994004554A1 (https=)
ZA (1) ZA935769B (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5510340A (en) * 1992-06-12 1996-04-23 Sri International Antihypercholesterolemic compounds and related pharmaceutical compositions and methods of use
CA2794565C (en) 2010-04-08 2018-08-21 Emory University Substituted androst-4-ene diones

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3032551A (en) * 1961-05-25 1962-05-01 Syntex Sa Pyrrolo(3', 2'-2, 3)-androstanes and process therefor
US3282928A (en) * 1964-04-23 1966-11-01 American Cyanamid Co 1, 11-iminoestratetraenes
GB8503940D0 (en) * 1985-02-15 1985-03-20 Erba Farmitalia 4-substituted androstendione derivatives
GB8617107D0 (en) * 1986-07-14 1986-08-20 Erba Farmitalia 6-/7-methylenandrosta-1 4-diene-3 17-dione derivatives
GB8622330D0 (en) * 1986-09-17 1986-10-22 Erba Farmitalia 4-substituted 6-alkylidenandrostene-3,17-dione derivatives
GB8721384D0 (en) * 1987-09-11 1987-10-21 Erba Farmitalia 17-substituted andro-sta-1 4-dien-3-one derivatives

Also Published As

Publication number Publication date
CA2120726A1 (en) 1994-03-03
GB9217035D0 (en) 1992-09-23
AU4707293A (en) 1994-03-15
US5457097A (en) 1995-10-10
AU662077B2 (en) 1995-08-17
ATE136036T1 (de) 1996-04-15
EP0608404B1 (en) 1996-03-27
HU9401003D0 (en) 1994-07-28
DE69302007D1 (de) 1996-05-02
GR3019729T3 (en) 1996-07-31
FI941635A7 (fi) 1994-04-08
WO1994004554A1 (en) 1994-03-03
EP0608404A1 (en) 1994-08-03
FI941635A0 (fi) 1994-04-08
MX9304852A (es) 1994-02-28
IL106597A (en) 1997-09-30
MY108957A (en) 1996-11-30
DK0608404T3 (da) 1996-04-29
ES2088289T3 (es) 1996-08-01
NZ254805A (en) 1995-11-27
IL106597A0 (en) 1993-12-08
TW276257B (https=) 1996-05-21
JPH07500119A (ja) 1995-01-05
DE69302007T2 (de) 1996-08-29
HUT67662A (en) 1995-04-28
ZA935769B (en) 1994-03-08

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